BR6464371D0 - Processo para fazer benzazois substituidos na posicao 5 - Google Patents

Processo para fazer benzazois substituidos na posicao 5

Info

Publication number
BR6464371D0
BR6464371D0 BR164371/64A BR16437164A BR6464371D0 BR 6464371 D0 BR6464371 D0 BR 6464371D0 BR 164371/64 A BR164371/64 A BR 164371/64A BR 16437164 A BR16437164 A BR 16437164A BR 6464371 D0 BR6464371 D0 BR 6464371D0
Authority
BR
Brazil
Prior art keywords
benzazoles
replaced
making
making benzazoles
benzazoles replaced
Prior art date
Application number
BR164371/64A
Other languages
English (en)
Inventor
& Co Inc Merck
Original Assignee
& Co Inc Merck
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by & Co Inc Merck filed Critical & Co Inc Merck
Publication of BR6464371D0 publication Critical patent/BR6464371D0/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
BR164371/64A 1963-11-19 1964-11-16 Processo para fazer benzazois substituidos na posicao 5 BR6464371D0 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32484763A 1963-11-19 1963-11-19
US33294063A 1963-12-23 1963-12-23
US62939667A 1967-04-10 1967-04-10

Publications (1)

Publication Number Publication Date
BR6464371D0 true BR6464371D0 (pt) 1973-07-26

Family

ID=27406362

Family Applications (1)

Application Number Title Priority Date Filing Date
BR164371/64A BR6464371D0 (pt) 1963-11-19 1964-11-16 Processo para fazer benzazois substituidos na posicao 5

Country Status (11)

Country Link
US (1) US3478046A (pt)
BE (1) BE655925A (pt)
BR (1) BR6464371D0 (pt)
DE (2) DE1470105A1 (pt)
DK (1) DK124263B (pt)
FR (2) FR1453247A (pt)
GB (1) GB1074640A (pt)
IL (1) IL22369A (pt)
NL (1) NL144612B (pt)
NO (1) NO118912B (pt)
SE (1) SE322781B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2028041A1 (en) * 1969-01-15 1970-10-09 Synthelabo N-salicyl 2-chloro 4-nitro aniline - vetinary - anthelmintic and parasiticide
US4053472A (en) * 1969-04-19 1977-10-11 Schering Aktiengesellschaft 2-(5-nitro-2-imidazolyl)-benzimidazoles
US3985755A (en) * 1972-06-02 1976-10-12 E. R. Squibb & Sons, Inc. Pyridine containing isothiocyanobenzoxazoles
US3983130A (en) * 1972-06-02 1976-09-28 E. R. Squibb & Sons, Inc. Anthelmintic isothiocyanobenzoxazoles
US3929814A (en) * 1974-04-01 1975-12-30 Squibb & Sons Inc (Oxadiazolyl) alkyl) benzimidazoles
IT1099589B (it) * 1978-08-04 1985-09-18 Ravizza Spa Processo per la preparazione di derivati dell'acido benzoxazolil propionico
US4281005A (en) * 1979-03-05 1981-07-28 Merck & Co., Inc. Novel 2-pyridylimidazole compounds
US4365019A (en) * 1981-08-06 1982-12-21 Eastman Kodak Company Positive-working resist quinone diazide containing composition and imaging method having improved development rates
GB9605065D0 (en) * 1996-03-11 1996-05-08 Merck Sharp & Dohme Therapeutic agents
AU2005264998A1 (en) 2004-06-17 2006-01-26 Wyeth The present invention relates to methods of making Gonadotropin Releasing Hormone ('GnRH') (also known as Leutinizing Hormone Releasing Hormone) receptor antagonists
US7696210B2 (en) 2004-06-17 2010-04-13 Wyeth Gonadotropin releasing hormone receptor antagonists
US7538113B2 (en) 2005-02-18 2009-05-26 Wyeth 4-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7582634B2 (en) 2005-02-18 2009-09-01 Wyeth 7-substituted imidazo[4,5-c]pyridine antagonists of gonadotropin releasing hormone receptor
US7534796B2 (en) 2005-02-18 2009-05-19 Wyeth Imidazo[4,5-b]pyridine antagonists of gonadotropin releasing hormone receptor
US7531542B2 (en) 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
US7582636B2 (en) 2005-05-26 2009-09-01 Wyeth Piperazinylimidazopyridine and piperazinyltriazolopyridine antagonists of Gonadotropin Releasing Hormone receptor

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2872453A (en) * 1959-02-03 Indole derivatives
US2945030A (en) * 1958-07-24 1960-07-12 Smith Kline French Lab Substituted aralkyl phenothiazinylalkyl piperazines
BE599143A (pt) * 1960-01-18
GB993581A (en) * 1960-03-03 1965-05-26 Wellcome Found Phenoxyalkylguanidines and their synthesis and pharmaceutical preparations containing them

Also Published As

Publication number Publication date
US3478046A (en) 1969-11-11
BE655925A (pt) 1965-05-18
NL144612B (nl) 1975-01-15
DE1770175A1 (de) 1971-10-07
NL6413475A (pt) 1965-05-20
GB1074640A (en) 1967-07-05
DK124263B (da) 1972-10-02
IL22369A (en) 1968-10-24
FR1453247A (fr) 1966-06-03
SE322781B (pt) 1970-04-20
NO118912B (pt) 1970-03-02
DE1470105A1 (de) 1969-11-20
FR4234M (pt) 1966-06-20

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