BR112023023866A2 - Derivado de piperazina e seu uso na medicina - Google Patents
Derivado de piperazina e seu uso na medicinaInfo
- Publication number
- BR112023023866A2 BR112023023866A2 BR112023023866A BR112023023866A BR112023023866A2 BR 112023023866 A2 BR112023023866 A2 BR 112023023866A2 BR 112023023866 A BR112023023866 A BR 112023023866A BR 112023023866 A BR112023023866 A BR 112023023866A BR 112023023866 A2 BR112023023866 A2 BR 112023023866A2
- Authority
- BR
- Brazil
- Prior art keywords
- medicine
- piperazine derivative
- piperazine
- derivative
- manufacture
- Prior art date
Links
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical class C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 title abstract 3
- 239000003814 drug Substances 0.000 abstract 2
- 230000000259 anti-tumor effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 150000004885 piperazines Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
derivado de piperazina e seu uso na medicina. o presente pedido se refere a um composto à base de piperazina e uma composição do mesmo, e ao seu uso na fabricação de um medicamento antitumoral.
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN202110550437 | 2021-05-21 | ||
CN202110562428 | 2021-05-24 | ||
CN202110885041 | 2021-08-03 | ||
CN202111331120 | 2021-11-12 | ||
CN202210084201 | 2022-01-25 | ||
PCT/CN2022/094124 WO2022242750A1 (zh) | 2021-05-21 | 2022-05-20 | 哌嗪衍生物及其在医药上的应用 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112023023866A2 true BR112023023866A2 (pt) | 2024-02-06 |
Family
ID=84141136
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112023023866A BR112023023866A2 (pt) | 2021-05-21 | 2022-05-20 | Derivado de piperazina e seu uso na medicina |
Country Status (9)
Country | Link |
---|---|
US (1) | US20240158406A1 (pt) |
EP (1) | EP4342896A1 (pt) |
JP (1) | JP2024519088A (pt) |
KR (1) | KR20240012534A (pt) |
CN (1) | CN117279917A (pt) |
AU (1) | AU2022277493A1 (pt) |
BR (1) | BR112023023866A2 (pt) |
CA (1) | CA3217941A1 (pt) |
WO (1) | WO2022242750A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2024032409A1 (zh) * | 2022-08-09 | 2024-02-15 | 成都百裕制药股份有限公司 | 哌嗪类化合物在联合放疗治疗肿瘤中的用途 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2013544891A (ja) * | 2010-12-08 | 2013-12-19 | ヴァンダービルト ユニバーシティー | mGLUR5受容体のアロステリック調節剤としての二環式ピラゾール化合物 |
AU2011343477A1 (en) * | 2010-12-17 | 2013-07-04 | Vanderbilt University | Bicyclic triazole and pyrazole lactams as allosteric modulators of mGluR5 receptors |
CN103570725B (zh) * | 2012-08-01 | 2017-03-22 | 中国科学院上海药物研究所 | 哌嗪并三唑类化合物及其制备方法和用途 |
HRP20230458T1 (hr) | 2018-04-30 | 2023-07-21 | Ribon Therapeutics Inc. | Piridazinoni kao inhibitori parp7 |
WO2020223229A1 (en) * | 2019-04-29 | 2020-11-05 | Ribon Therapeutics, Inc. | Solid forms of a parp7 inhibitor |
CN112745312B (zh) * | 2019-10-30 | 2022-08-30 | 沈阳中化农药化工研发有限公司 | 哒嗪酮异恶唑甲醚类化合物及其应用 |
IL292432A (en) * | 2019-10-30 | 2022-06-01 | Ribon Therapeutics Inc | Pyridazinones as parp7 inhibitors |
WO2021087018A1 (en) * | 2019-10-30 | 2021-05-06 | Ribon Therapeutics, Inc. | Pyridazinones as parp7 inhibitors |
-
2022
- 2022-05-20 AU AU2022277493A patent/AU2022277493A1/en active Pending
- 2022-05-20 CN CN202280033063.XA patent/CN117279917A/zh active Pending
- 2022-05-20 EP EP22804069.7A patent/EP4342896A1/en active Pending
- 2022-05-20 CA CA3217941A patent/CA3217941A1/en active Pending
- 2022-05-20 BR BR112023023866A patent/BR112023023866A2/pt unknown
- 2022-05-20 WO PCT/CN2022/094124 patent/WO2022242750A1/zh active Application Filing
- 2022-05-20 JP JP2023571901A patent/JP2024519088A/ja active Pending
- 2022-05-20 KR KR1020237044434A patent/KR20240012534A/ko unknown
-
2023
- 2023-11-21 US US18/515,434 patent/US20240158406A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
TW202246277A (zh) | 2022-12-01 |
EP4342896A1 (en) | 2024-03-27 |
CN117279917A (zh) | 2023-12-22 |
US20240158406A1 (en) | 2024-05-16 |
CA3217941A1 (en) | 2022-11-24 |
JP2024519088A (ja) | 2024-05-08 |
KR20240012534A (ko) | 2024-01-29 |
AU2022277493A1 (en) | 2023-11-23 |
WO2022242750A1 (zh) | 2022-11-24 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CO2023000186A2 (es) | Derivados de quinoxalina como fármacos anti-cáncer | |
BR112023023866A2 (pt) | Derivado de piperazina e seu uso na medicina | |
BR112016026205A8 (pt) | moduladores de entrançamento de gene smn2, seu uso e seu processo de preparação, e composições farmacêuticas | |
UY39027A (es) | Uso de favipiravir en el tratamiento de la infección por coronavirus | |
AR070783A1 (es) | Forma de cristal de derivados de fenilamina-pirimidina | |
BR112021022889A2 (pt) | Derivados heterocíclicos fundidos | |
BR112023018348A2 (pt) | Forma de cristal de composto de óxido de nitrogênio e piridina e uso da mesma | |
BR112022002112A2 (pt) | Composições de probióticos à base de plantas fermentadas e processos de preparação das mesmas | |
BR112021019859A2 (pt) | Vacinas de circovírus suíno tipo 3 (pcv3) e produção e seus usos | |
BR112018008076A2 (pt) | derivados de lapachona contendo dois centros redox e métodos de uso dos mesmos | |
BR112022016286A2 (pt) | Compostos macrocíclicos, processo para sua preparação e composições farmacêuticas contendo-os | |
BR112018070370A2 (pt) | glucono delta-lactona para tratamento de infecções fúngicas vaginais | |
CL2022000045A1 (es) | Derivados de camptotecina con un resto disulfuro y un resto piperazina. | |
BR112021024546A2 (pt) | Compostos tricíclicos e uso dos mesmos | |
BR112022020897A2 (pt) | Forma de dosagem oral sólida compreendendo pomalidomida. | |
UY39257A (es) | Composición farmacéutica acuosa de levilimab y su uso | |
BR112022011919A2 (pt) | Triterpenoides sintéticos com substituintes à base de nitrogênio em c-17 e métodos de uso dos mesmos | |
TWD202991S (zh) | 錶 | |
TWD202982S (zh) | 錶 | |
CL2022002752A1 (es) | Complejos cristalinos | |
BR112021026774A2 (pt) | N-formilhidroxilaminas como inibidores da neprilisina (nep) e, em praticular, como inibidores mistos da aminopeptidase n (apn) e da neprilisina (nep) | |
JP1718770S (ja) | テーブル | |
CL2023001138A1 (es) | Derivados de 2-hidroxicicloalcan-1-carbamoilo inhibidores de galectina-3 | |
CL2023002052A1 (es) | Derivados de pirazolamida | |
JP1731853S (ja) | ベッドサイドテーブル |