BR112021021681A2 - Rebamipida para uso na prevenção e/ou tratamento de sinucleinopatias - Google Patents
Rebamipida para uso na prevenção e/ou tratamento de sinucleinopatiasInfo
- Publication number
- BR112021021681A2 BR112021021681A2 BR112021021681A BR112021021681A BR112021021681A2 BR 112021021681 A2 BR112021021681 A2 BR 112021021681A2 BR 112021021681 A BR112021021681 A BR 112021021681A BR 112021021681 A BR112021021681 A BR 112021021681A BR 112021021681 A2 BR112021021681 A2 BR 112021021681A2
- Authority
- BR
- Brazil
- Prior art keywords
- rebamipide
- prevention
- treatment
- synucleinopathies
- synucleinopathy
- Prior art date
Links
- ALLWOAVDORUJLA-UHFFFAOYSA-N Rebamipida Chemical compound C=1C(=O)NC2=CC=CC=C2C=1CC(C(=O)O)NC(=O)C1=CC=C(Cl)C=C1 ALLWOAVDORUJLA-UHFFFAOYSA-N 0.000 title abstract 4
- 208000032859 Synucleinopathies Diseases 0.000 title abstract 4
- 229950004535 rebamipide Drugs 0.000 title abstract 4
- 230000002265 prevention Effects 0.000 title abstract 3
- 230000003870 intestinal permeability Effects 0.000 abstract 2
- 208000018737 Parkinson disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4704—2-Quinolinones, e.g. carbostyril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Abstract
rebamipida para uso na prevenção e/ou tratamento de sinucleinopatias. a presente invenção refere-se à rebamipida para o uso em um método de prevenção e/ou tratamento de uma sinucleinopatia, em particular, de doença de parkinson. em particular, a rebamipida é usada na prevenção e/ou tratamento de uma sinucleinopatia em uma pessoa que sofre de permeabilidade intestinal aumentada ou em uma pessoa que está em risco de permeabilidade intestinal aumentada.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP19020318.2A EP3741370A1 (en) | 2019-04-30 | 2019-04-30 | Rebamipide for use in prevention and/or treatment of synucleinopathies |
PCT/EP2020/062120 WO2020221892A2 (en) | 2019-04-30 | 2020-04-30 | Rebamipide for use in prevention and/or treatment of synucleinopathies |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112021021681A2 true BR112021021681A2 (pt) | 2021-12-21 |
Family
ID=66396957
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112021021681A BR112021021681A2 (pt) | 2019-04-30 | 2020-04-30 | Rebamipida para uso na prevenção e/ou tratamento de sinucleinopatias |
Country Status (12)
Country | Link |
---|---|
US (1) | US20220202805A1 (pt) |
EP (1) | EP3741370A1 (pt) |
JP (1) | JP2022533005A (pt) |
KR (1) | KR20220003064A (pt) |
CN (1) | CN113784715A (pt) |
AU (1) | AU2020266279A1 (pt) |
BR (1) | BR112021021681A2 (pt) |
CA (1) | CA3138389A1 (pt) |
EA (1) | EA202192961A1 (pt) |
MX (1) | MX2021013360A (pt) |
WO (1) | WO2020221892A2 (pt) |
ZA (1) | ZA202110052B (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN112603899A (zh) * | 2020-12-23 | 2021-04-06 | 南京友杰医药科技有限公司 | 瑞巴派特肠溶片及其制备方法 |
-
2019
- 2019-04-30 EP EP19020318.2A patent/EP3741370A1/en active Pending
-
2020
- 2020-04-30 WO PCT/EP2020/062120 patent/WO2020221892A2/en active Application Filing
- 2020-04-30 KR KR1020217039133A patent/KR20220003064A/ko unknown
- 2020-04-30 CN CN202080032289.9A patent/CN113784715A/zh active Pending
- 2020-04-30 JP JP2021564279A patent/JP2022533005A/ja active Pending
- 2020-04-30 CA CA3138389A patent/CA3138389A1/en active Pending
- 2020-04-30 EA EA202192961A patent/EA202192961A1/ru unknown
- 2020-04-30 US US17/607,048 patent/US20220202805A1/en active Pending
- 2020-04-30 BR BR112021021681A patent/BR112021021681A2/pt unknown
- 2020-04-30 MX MX2021013360A patent/MX2021013360A/es unknown
- 2020-04-30 AU AU2020266279A patent/AU2020266279A1/en not_active Abandoned
-
2021
- 2021-12-06 ZA ZA2021/10052A patent/ZA202110052B/en unknown
Also Published As
Publication number | Publication date |
---|---|
JP2022533005A (ja) | 2022-07-21 |
WO2020221892A2 (en) | 2020-11-05 |
ZA202110052B (en) | 2023-11-29 |
AU2020266279A1 (en) | 2021-12-23 |
WO2020221892A3 (en) | 2020-12-24 |
EP3741370A1 (en) | 2020-11-25 |
CA3138389A1 (en) | 2020-11-05 |
EA202192961A1 (ru) | 2022-01-20 |
US20220202805A1 (en) | 2022-06-30 |
KR20220003064A (ko) | 2022-01-07 |
MX2021013360A (es) | 2022-01-31 |
CN113784715A (zh) | 2021-12-10 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BR112017008093A2 (pt) | processos para tratamento de doenças oculares | |
MX2018010693A (es) | Compuestos biciclicos para diagnostico y terapia. | |
EA201000603A1 (ru) | ПРИМЕНЕНИЕ АНТИТЕЛ К TrkB ДЛЯ ЛЕЧЕНИЯ РЕСПИРАТОРНЫХ НАРУШЕНИЙ | |
BR112017026739A2 (pt) | compostos para uso no tratamento de distúrbios neuromusculares | |
MX2022010357A (es) | Anticuerpos inhibidores de anti-pcsk9 para el tratamiento de pacientes con hiperlipidemia que se someten aferesis de lipoproteina. | |
BR112018069515A2 (pt) | uso de masitinibe para tratamento de uma subpopulação de pacientes com esclerose lateral amiotrófica | |
BR112018014675A2 (pt) | novos derivados de cianoindolina substituída como inibidores de nik | |
SG11201903725UA (en) | Composition for promoting differentiation of and protecting neural stem cells and method for inducing neural regeneration using same | |
EP4285993A3 (en) | Growth differentiation factor 15 as biomarker for metformin | |
BR112017025998A2 (pt) | inibidor de eixo igfbp3/tmem219, composição farmacêutica para uso no tratamento e/ou prevenção de diabetes, método para identificar um indivíduo em risco de desenvolver diabetes tipo 1 e/ou tipo 2 ou para monitorar a resposta a um tratamento terapêutico em um indivíduo e kit | |
BR112021021826A8 (pt) | Uso de apremilaste e um inibidor da tirosina quinase 2 no tratamento de uma doença ou um transtorno responsivo à inibição da fosfodiesterase tipo 4 | |
MX2020001164A (es) | Composicion para su uso en la prevencion y/o el tratamiento de la mucositis orogastrointestinal inducida por un tratamiento oncologico. | |
BR112021018262A2 (pt) | Tratamento de doenças e distúrbios mitocondriais associados, incluindo sintomas dos mesmos usando pridopidina | |
BR112021021681A2 (pt) | Rebamipida para uso na prevenção e/ou tratamento de sinucleinopatias | |
BR0313413A (pt) | Uso da vacinação beta amilóide juntamente com um inibidor da cox-2 seletivo para o tratamento da doença de alzheimer | |
BR112019008241A2 (pt) | tratamento do prurigo nodular | |
NO20073104L (no) | Anvendelse av en 5-HT6 agonist for behandling og forebygging av neurodegenerative forstyrrelser | |
MX2020013100A (es) | Metodos de uso de cd24 para la prevencion y tratamiento de enfermedad de injerto contra hospedero y mucositis. | |
BR112022003918A2 (pt) | Rebamipida para uso na prevenção e tratamento da doença de crohn | |
BR112022019168A2 (pt) | Tratamento de distúrbios respiratórios | |
MX2022000783A (es) | Inhibidores de la ferroportina para el uso en la prevencion y el tratamiento de lesiones renales. | |
BR112018012126A2 (pt) | ?adjuvante, método para prevenir e/ou tratar uma doença autoimune, e, uso de um adjuvante? | |
BR112017027298A2 (pt) | método de tratamento e/ou prevenção de drea ou asma em pacientes humanos; e método de prevenção, reversão ou tratamento de sintoma(s) de dessensibilização à aspirina em pacientes com drea | |
MX2022002625A (es) | Rebamipida para usarse en la profilaxis y tratamiento de enfermedad celiaca. | |
CL2021003602A1 (es) | Métodos para tratar o prevenir la atrofia muscular espinal |