BR112012032540A2 - formulação de solução de lactona macrocíclica, e, uso da formulação veterinária - Google Patents
formulação de solução de lactona macrocíclica, e, uso da formulação veterináriaInfo
- Publication number
- BR112012032540A2 BR112012032540A2 BR112012032540A BR112012032540A BR112012032540A2 BR 112012032540 A2 BR112012032540 A2 BR 112012032540A2 BR 112012032540 A BR112012032540 A BR 112012032540A BR 112012032540 A BR112012032540 A BR 112012032540A BR 112012032540 A2 BR112012032540 A2 BR 112012032540A2
- Authority
- BR
- Brazil
- Prior art keywords
- formulation
- macrocyclic lactone
- veterinary
- lactone solution
- solution formulation
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
formulação de solução de lactona macrocíclica, e, uso da formulação veterinária.a presente invenção refere-se a formulações para controlar parasitas, compreendendo a combinação de um composto de lactona macrocíclica e levamisol em que o levamisol está em forma particulada em suspensão em um solvente não aquoso.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10167222 | 2010-06-24 | ||
US42084910P | 2010-12-08 | 2010-12-08 | |
PCT/EP2011/060535 WO2011161209A1 (en) | 2010-06-24 | 2011-06-23 | Injectable formulation of a macrocyclic lactone and levamisole |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112012032540A2 true BR112012032540A2 (pt) | 2016-11-22 |
Family
ID=44628008
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012032540A BR112012032540A2 (pt) | 2010-06-24 | 2011-06-23 | formulação de solução de lactona macrocíclica, e, uso da formulação veterinária |
Country Status (9)
Country | Link |
---|---|
US (1) | US20130090296A1 (pt) |
EP (1) | EP2585062A1 (pt) |
AR (1) | AR081970A1 (pt) |
AU (1) | AU2011268899C1 (pt) |
BR (1) | BR112012032540A2 (pt) |
MX (1) | MX336924B (pt) |
NZ (1) | NZ603775A (pt) |
WO (1) | WO2011161209A1 (pt) |
ZA (1) | ZA201209445B (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2010101089B4 (en) * | 2010-10-06 | 2013-03-07 | Jurox Pty Limited | Parasiticidal Composition |
AU2010101389C4 (en) * | 2010-12-08 | 2017-03-02 | Jurox Pty Ltd | Anthelmintic formulation |
AU2012227241C1 (en) * | 2011-09-23 | 2017-01-19 | Virbac (Australia) Pty Limited | Veterinary Topical Formulation |
NZ701697A (en) | 2014-03-24 | 2016-05-27 | Donaghys Ltd | Stable veterinary anthelmintic formulations |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3950360A (en) | 1972-06-08 | 1976-04-13 | Sankyo Company Limited | Antibiotic substances |
US3984564A (en) | 1972-06-08 | 1976-10-05 | Sankyo Company Limited | Antibiotic substances B-41, their production and their use as insecticides and acaricides |
SE434277B (sv) | 1976-04-19 | 1984-07-16 | Merck & Co Inc | Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis |
US4199569A (en) | 1977-10-03 | 1980-04-22 | Merck & Co., Inc. | Selective hydrogenation products of C-076 compounds and derivatives thereof |
ES8800986A1 (es) | 1985-07-27 | 1987-12-01 | Pfizer | Un procedimiento para la produccion de un nuevo derivado de avermectina |
US4916154A (en) | 1986-09-12 | 1990-04-10 | American Cyanamid Company | 23-Imino derivatives of LL-F28249 compounds |
IL98599A (en) | 1990-06-28 | 1995-06-29 | Merck & Co Inc | Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them |
NZ335166A (en) | 1999-04-14 | 2001-11-30 | Ashmont Holdings Ltd | Anthelmintic composition containing triclabendazole in at least one solvent |
US5399717A (en) | 1993-09-29 | 1995-03-21 | Merck & Co., Inc. | Glycosidation route to 4"-epi-methylamino-4"-deoxyavermectin B1 |
AU772988B2 (en) | 1999-06-04 | 2004-05-13 | Elanco Tiergesundheit Ag | Stable biocidal compositions |
CN1375291A (zh) * | 2001-03-16 | 2002-10-23 | 王玉万 | 一种含左旋咪唑或其盐类的兽用复方注射剂 |
NZ520295A (en) * | 2002-07-19 | 2005-04-29 | Ashmont Holdings Ltd | Anthelmintic formulations comprising levamisole and either an avermectin or milbemycin |
NZ552040A (en) * | 2006-12-13 | 2009-04-30 | Bomac Research Ltd | Veterinary formulation comprising an anthelmintic compound and glyceryl acetate |
CA2734459A1 (en) * | 2008-08-18 | 2010-02-25 | Intervet International B.V. | Anthelmintic compositions |
-
2011
- 2011-06-22 AR ARP110102154A patent/AR081970A1/es not_active Application Discontinuation
- 2011-06-23 MX MX2012015193A patent/MX336924B/es active IP Right Grant
- 2011-06-23 NZ NZ603775A patent/NZ603775A/en unknown
- 2011-06-23 US US13/703,941 patent/US20130090296A1/en not_active Abandoned
- 2011-06-23 WO PCT/EP2011/060535 patent/WO2011161209A1/en active Application Filing
- 2011-06-23 AU AU2011268899A patent/AU2011268899C1/en active Active
- 2011-06-23 EP EP11729597.2A patent/EP2585062A1/en not_active Withdrawn
- 2011-06-23 BR BR112012032540A patent/BR112012032540A2/pt not_active Application Discontinuation
-
2012
- 2012-12-12 ZA ZA2012/09445A patent/ZA201209445B/en unknown
Also Published As
Publication number | Publication date |
---|---|
AU2011268899C1 (en) | 2020-03-05 |
ZA201209445B (en) | 2013-08-28 |
AU2011268899A1 (en) | 2012-12-13 |
US20130090296A1 (en) | 2013-04-11 |
MX2012015193A (es) | 2013-01-24 |
EP2585062A1 (en) | 2013-05-01 |
NZ603775A (en) | 2015-01-30 |
MX336924B (es) | 2016-02-05 |
AU2011268899B2 (en) | 2016-07-07 |
AR081970A1 (es) | 2012-10-31 |
WO2011161209A1 (en) | 2011-12-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07G | Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette] |
Free format text: NOTIFICACAO DE DEVOLUCAO DO PEDIDO POR NAO SE ENQUADRAR NO ART. 229-C DA LPI. |
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B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
B06I | Publication of requirement cancelled [chapter 6.9 patent gazette] |
Free format text: ANULADA A PUBLICACAO CODIGO 6.20 NA RPI NO 2516 DE 26/03/2019 POR TER SIDO INDEVIDA. |
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B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] | ||
B12B | Appeal against refusal [chapter 12.2 patent gazette] |