BR0112121A - Process for preparing 4-bromoaniline derivatives - Google Patents
Process for preparing 4-bromoaniline derivativesInfo
- Publication number
- BR0112121A BR0112121A BR0112121-9A BR0112121A BR0112121A BR 0112121 A BR0112121 A BR 0112121A BR 0112121 A BR0112121 A BR 0112121A BR 0112121 A BR0112121 A BR 0112121A
- Authority
- BR
- Brazil
- Prior art keywords
- preparing
- derivatives
- bromoaniline
- cycloalkyl
- alkoxy
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 3
- WDFQBORIUYODSI-IDEBNGHGSA-N 4-bromoaniline Chemical class N[13C]1=[13CH][13CH]=[13C](Br)[13CH]=[13CH]1 WDFQBORIUYODSI-IDEBNGHGSA-N 0.000 title abstract 2
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 1
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 1
- WDFQBORIUYODSI-UHFFFAOYSA-N 4-bromoaniline Chemical class NC1=CC=C(Br)C=C1 WDFQBORIUYODSI-UHFFFAOYSA-N 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
Abstract
"PROCESSO PARA PREPARAR DERIVADOS DE 4-BROMO-ANILINA". é descrito um processo para preparar derivados de 4-bromo-anilina de fórmula I na qual os substituintes têm os seguintes significados: R^ 1^ é C~ 1~-C~ 6~-alquila, C~ 1~-C~ 6~-halo-alquila, C~ 1~-C~ 6~-alcóxi, C~ 1~-C~ 6~halo-alcóxi., C~ 3~-C~ 8~-cicloalquila, halogênio. R^ 2^ é C~ 1~-C~ 6~-alquila, C~ 1~-C~ 6~-alcóxi, C~ 3~-C~ 8~-cicloalquila, C~ 2~-C~ 6~alquenila, ciano ou um radical heterocíclico."PROCESS FOR PREPARING 4-BROMO-ANILINE DERIVATIVES". A process for preparing 4-bromoaniline derivatives of formula I is described in which the substituents have the following meanings: R 1 is C 1 -C 6 alkyl, C 1 -C 6 -haloalkyl, C1-C6-alkoxy, C1-C6-haloalkoxy, C3-C8-cycloalkyl, halogen. R 2 is C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 3 -C 8 -cycloalkyl, C 2 -C 6 alkenyl, cyano or a heterocyclic radical.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10030975 | 2000-06-30 | ||
PCT/EP2001/007482 WO2002002537A1 (en) | 2000-06-30 | 2001-06-29 | Method for producing 4-bromine-aniline derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
BR0112121A true BR0112121A (en) | 2003-05-13 |
BRPI0112121B1 BRPI0112121B1 (en) | 2015-09-01 |
Family
ID=7646770
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0112121-9A BRPI0112121B1 (en) | 2000-06-30 | 2001-06-29 | Process for preparing 4-bromoaniline derivatives |
Country Status (22)
Country | Link |
---|---|
EP (1) | EP1296965B1 (en) |
JP (1) | JP4937485B2 (en) |
KR (1) | KR100779315B1 (en) |
CN (1) | CN1182124C (en) |
AT (1) | ATE305928T1 (en) |
AU (2) | AU6911101A (en) |
BR (1) | BRPI0112121B1 (en) |
CA (1) | CA2413723C (en) |
CZ (1) | CZ301413B6 (en) |
DE (1) | DE50107619D1 (en) |
DK (1) | DK1296965T3 (en) |
EA (1) | EA006293B1 (en) |
ES (1) | ES2250425T3 (en) |
HU (1) | HUP0301741A3 (en) |
IL (2) | IL153412A0 (en) |
MX (1) | MXPA02012483A (en) |
NO (1) | NO324408B1 (en) |
NZ (1) | NZ523825A (en) |
PL (1) | PL206026B1 (en) |
SK (1) | SK285627B6 (en) |
WO (1) | WO2002002537A1 (en) |
ZA (1) | ZA200300816B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8975431B2 (en) * | 2010-05-19 | 2015-03-10 | Rhodia Operations | Process for preparing an ortho-substituted 5-halophenol and a synthesis intermediate thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6377844A (en) * | 1986-09-18 | 1988-04-08 | Nippon Kayaku Co Ltd | Production of p-bromoanilines |
JPH0816085B2 (en) * | 1988-06-07 | 1996-02-21 | 日本化薬株式会社 | Method for producing 2-bromo-4-fluoroaniline |
IL108630A0 (en) * | 1993-02-18 | 1994-05-30 | Fmc Corp | Insecticidal substituted 2,4-diaminoquinazolines |
EP0923509A1 (en) * | 1996-08-30 | 1999-06-23 | Aventis Research & Technologies GmbH & Co. KG | Bromination of aromatic compounds with ozone |
DE59914392D1 (en) * | 1998-05-11 | 2007-08-09 | Basf Ag | PROCESS FOR THE PREPARATION OF ISOXAZOLIN-3-YL-ACYLBENZOLENE |
-
2001
- 2001-06-29 EA EA200300012A patent/EA006293B1/en not_active IP Right Cessation
- 2001-06-29 CA CA002413723A patent/CA2413723C/en not_active Expired - Fee Related
- 2001-06-29 EP EP01947430A patent/EP1296965B1/en not_active Expired - Lifetime
- 2001-06-29 SK SK1797-2002A patent/SK285627B6/en not_active IP Right Cessation
- 2001-06-29 DK DK01947430T patent/DK1296965T3/en active
- 2001-06-29 CZ CZ20024177A patent/CZ301413B6/en not_active IP Right Cessation
- 2001-06-29 CN CNB018119417A patent/CN1182124C/en not_active Expired - Lifetime
- 2001-06-29 KR KR1020027017711A patent/KR100779315B1/en not_active IP Right Cessation
- 2001-06-29 ES ES01947430T patent/ES2250425T3/en not_active Expired - Lifetime
- 2001-06-29 AU AU6911101A patent/AU6911101A/en active Pending
- 2001-06-29 NZ NZ523825A patent/NZ523825A/en unknown
- 2001-06-29 JP JP2002507793A patent/JP4937485B2/en not_active Expired - Lifetime
- 2001-06-29 MX MXPA02012483A patent/MXPA02012483A/en active IP Right Grant
- 2001-06-29 HU HU0301741A patent/HUP0301741A3/en unknown
- 2001-06-29 IL IL15341201A patent/IL153412A0/en active IP Right Grant
- 2001-06-29 AU AU2001269111A patent/AU2001269111B2/en not_active Ceased
- 2001-06-29 DE DE50107619T patent/DE50107619D1/en not_active Expired - Lifetime
- 2001-06-29 PL PL359155A patent/PL206026B1/en not_active IP Right Cessation
- 2001-06-29 WO PCT/EP2001/007482 patent/WO2002002537A1/en active IP Right Grant
- 2001-06-29 AT AT01947430T patent/ATE305928T1/en active
- 2001-06-29 BR BRPI0112121-9A patent/BRPI0112121B1/en not_active IP Right Cessation
-
2002
- 2002-12-12 IL IL153412A patent/IL153412A/en unknown
- 2002-12-23 NO NO20026201A patent/NO324408B1/en not_active IP Right Cessation
-
2003
- 2003-01-29 ZA ZA200300816A patent/ZA200300816B/en unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PT1257553E (en) | PIRROLOPYRIMIDINONE DERIVATIVES, PROCESS FOR THE PREPARATION AND USE | |
NO983970D0 (en) | Tricyclic compounds, their preparation and use | |
ES2182234T3 (en) | METALOPROTEASE INHIBITORS. | |
HRP20090162T1 (en) | Quinolinone-carboxamide compounds as 5-ht4 receptor agonists | |
BR0309534A (en) | Compound, pharmaceutical composition, and use of a compound | |
NO902301L (en) | PROCEDURE FOR THE PREPARATION OF DIARYLSTYRYLQINOLINE DISYRES. | |
DK0923554T3 (en) | N-Benzylpiperidine and tetrahydropyridine derivatives | |
BR0112456A (en) | Piperidine compounds for use as ccr-3 inhibitors | |
PT918776E (en) | TOTAL SYNTHESIS OF ANTITUMAL ACILFULVENOS | |
BRPI0510397A (en) | compounds, pharmaceutical compositions containing them, and methods of use thereof | |
DE60330758D1 (en) | CERTAIN PHARMACEUTICALLY VALUABLE SUBSTITUTED AMINO ALKYL HETEROCYCLES | |
NO995963D0 (en) | Carboxamides useful as 5-HTIF agonists | |
BR0013075A (en) | Tetrazolinone derivatives | |
PT1204658E (en) | SEROTONIN BENZOFURILPIPERAZINE AGONISTS | |
BR0112121A (en) | Process for preparing 4-bromoaniline derivatives | |
NZ337362A (en) | Heterocyclically substituted piperidyl-amino-indan-1-ol compounds and uses thereof | |
EA200200523A1 (en) | NEW FORMATED SUBSTITUTED AMINO DERIVATIVES 3-AMINO-1-PHENYL-1H [1,2,4] TRIAZOLE, METHODS FOR THEIR PRODUCTION AND CONTAINING THEIR PHARMACEUTICAL COMPOSITIONS | |
NO20015202D0 (en) | <beta> -hydroxyalkylamides, process for their preparation and use | |
PT1230252E (en) | BETA-D-5-TIOXYLOSE DERIVATIVES PROCESS FOR PREPARATION AND USE IN THERAPEUTICS | |
MY130817A (en) | Herbicides | |
NO20033049D0 (en) | Process for the preparation of (+/-) trans-4-p-fluorophenyl-3-hydroxymethyl-1 | |
DK1000952T3 (en) | New 2-halogen derivatives of 5-O-deosaminyl erythronolide A, process for their preparation and use thereof as pharmaceuticals | |
HUP0300266A2 (en) | 1,3,4-oxadiazole derivatives and process for producing the same | |
DK1140932T3 (en) | Derivatives of benzo-1,8-naphtyridine |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B07G | Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette] |
Free format text: NOTIFICACAO DE DEVOLUCAO DO PEDIDO POR NAO SE ENQUADRAR NO ART. 229-C DA LPI. |
|
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 01/09/2015, OBSERVADAS AS CONDICOES LEGAIS. |
|
B21F | Lapse acc. art. 78, item iv - on non-payment of the annual fees in time |
Free format text: REFERENTE A 19A ANUIDADE. |
|
B24J | Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12) |
Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2594 DE 24-09-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |