BR0009285A - Avermectin derivatives - Google Patents

Avermectin derivatives

Info

Publication number
BR0009285A
BR0009285A BR0009285-1A BR0009285A BR0009285A BR 0009285 A BR0009285 A BR 0009285A BR 0009285 A BR0009285 A BR 0009285A BR 0009285 A BR0009285 A BR 0009285A
Authority
BR
Brazil
Prior art keywords
avermectin derivatives
preparation
derivatives
agents
avermectin
Prior art date
Application number
BR0009285-1A
Other languages
Portuguese (pt)
Inventor
Werner Hallenbach
Achim Harder
Andreas Turberg
Olaf Hansen
Georg Von Samson-Himmelstjerna
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of BR0009285A publication Critical patent/BR0009285A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Patente de Invenção: "DERIVADOS DE AVERMECTINA". A invenção refere-se a novos derivados de avermectina da fórmula (I), na qual R^ 1^, R^ 2~, R^ 3^ e R^ 4^ têm os significados mencionados na descrição, vários processos para a sua preparação, os agentes contendo os mesmos e seu emprego para a preparação de agentes para combater ecto- e endoparasitas no animal.Invention Patent: "AVERMECTIN DERIVATIVES". The invention relates to new avermectin derivatives of formula (I), in which R ^ 1 ^, R ^ 2 ~, R ^ 3 ^ and R ^ 4 ^ have the meanings mentioned in the description, various processes for their preparation , the agents containing them and their use for the preparation of agents to combat ecto- and endoparasites in the animal.

BR0009285-1A 1999-03-25 2000-03-13 Avermectin derivatives BR0009285A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19913534A DE19913534A1 (en) 1999-03-25 1999-03-25 Avermectin derivatives
PCT/EP2000/002189 WO2000058328A2 (en) 1999-03-25 2000-03-13 Avermectin derivatives

Publications (1)

Publication Number Publication Date
BR0009285A true BR0009285A (en) 2002-01-22

Family

ID=7902359

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0009285-1A BR0009285A (en) 1999-03-25 2000-03-13 Avermectin derivatives

Country Status (9)

Country Link
EP (1) EP1169328A2 (en)
JP (1) JP2002540214A (en)
CN (1) CN1345327A (en)
AU (1) AU4394700A (en)
BR (1) BR0009285A (en)
CA (1) CA2368465A1 (en)
DE (1) DE19913534A1 (en)
HK (1) HK1045698A1 (en)
WO (1) WO2000058328A2 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10112318A1 (en) * 2001-02-05 2002-08-14 Henkel Kgaa conditioning
CN102578113A (en) * 2012-01-18 2012-07-18 华南理工大学 Sucrose ester-emamectin benzoate compound microcapsule pesticide and preparation method thereof
JO3626B1 (en) 2012-02-23 2020-08-27 Merial Inc Topical compositions comprising fipronil and permethrin and methods of use
CN103601776A (en) * 2013-11-25 2014-02-26 京博农化科技股份有限公司 Preparation method of emamectin benzoate midbody
CN103833811A (en) * 2014-03-25 2014-06-04 武汉大学 Abamectin derivative and preparation method thereof
CN109824745A (en) * 2019-01-24 2019-05-31 南开大学 A kind of synthesis and application of ivermectin derivative
CN113817008B (en) * 2021-07-15 2023-05-23 湖州师范学院 Preparation method and application of novel succinyl hexadecanoic macrolide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8800986A1 (en) * 1985-07-27 1987-12-01 Pfizer Antiparasitic avermectin and milbemycin derivatives and process for their preparation.
CH669382A5 (en) * 1986-05-21 1989-03-15 Ciba Geigy Ag 13-0-substd. milbemycin derivs. - with insecticidal, acaricidal, nematocidal and anthelmintic activity, prepd. by etherification of 13-0 unsubstituted cpds
GB8807280D0 (en) * 1988-03-26 1988-04-27 Pfizer Ltd Antiparasitic agents

Also Published As

Publication number Publication date
WO2000058328A3 (en) 2001-04-26
HK1045698A1 (en) 2002-12-06
WO2000058328A2 (en) 2000-10-05
CN1345327A (en) 2002-04-17
EP1169328A2 (en) 2002-01-09
JP2002540214A (en) 2002-11-26
CA2368465A1 (en) 2000-10-05
AU4394700A (en) 2000-10-16
DE19913534A1 (en) 2000-10-05

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BR0009285A (en) Avermectin derivatives

Legal Events

Date Code Title Description
B08F Application fees: dismissal - article 86 of industrial property law

Free format text: REFERENTE A 5A, 6A E 7A ANUIDADES.

B08K Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87)

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1925 DE 27/11/2007.