BG22833A3 - Метод за получаване на n-(фурил-метил)-морфинани и техните присъединителни с киселини соли - Google Patents

Метод за получаване на n-(фурил-метил)-морфинани и техните присъединителни с киселини соли

Info

Publication number
BG22833A3
BG22833A3 BG021205A BG2120572A BG22833A3 BG 22833 A3 BG22833 A3 BG 22833A3 BG 021205 A BG021205 A BG 021205A BG 2120572 A BG2120572 A BG 2120572A BG 22833 A3 BG22833 A3 BG 22833A3
Authority
BG
Bulgaria
Prior art keywords
morphinanes
furyl
methyl
preparation
acid
Prior art date
Application number
BG021205A
Other languages
Bulgarian (bg)
English (en)
Inventor
Herbert Merz
Adolf Langbein
Helmut Wick
Klaus Stockhaus
Original Assignee
C.H.Boehringer Sohn
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by C.H.Boehringer Sohn filed Critical C.H.Boehringer Sohn
Publication of BG22833A3 publication Critical patent/BG22833A3/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG021205A 1971-02-19 1972-02-17 Метод за получаване на n-(фурил-метил)-морфинани и техните присъединителни с киселини соли BG22833A3 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19712107989 DE2107989A1 (de) 1971-02-19 1971-02-19 N-(Furyl-methy])-morphinane, deren Säureadditionssalze sowie Verfahren zu deren Herstellung

Publications (1)

Publication Number Publication Date
BG22833A3 true BG22833A3 (bg) 1977-04-20

Family

ID=5799263

Family Applications (4)

Application Number Title Priority Date Filing Date
BG021205A BG22833A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-(фурил-метил)-морфинани и техните присъединителни с киселини соли
BG019747A BG20584A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-<фурил-метил,порфинани и на техни присъединителни с киселинни соли
BG021203A BG20356A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-(фурил-метил)- морфани и техни присъединителни с киселини соли
BG021204A BG20357A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-(фурил-метил)-морфинани и техни присъединителни с киселини соли

Family Applications After (3)

Application Number Title Priority Date Filing Date
BG019747A BG20584A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-<фурил-метил,порфинани и на техни присъединителни с киселинни соли
BG021203A BG20356A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-(фурил-метил)- морфани и техни присъединителни с киселини соли
BG021204A BG20357A3 (bg) 1971-02-19 1972-02-17 Метод за получаване на n-(фурил-метил)-морфинани и техни присъединителни с киселини соли

Country Status (25)

Country Link
US (1) US3793329A (US20100154137A1-20100624-C00004.png)
AT (3) AT318600B (US20100154137A1-20100624-C00004.png)
AU (1) AU468490B2 (US20100154137A1-20100624-C00004.png)
BE (1) BE779582A (US20100154137A1-20100624-C00004.png)
BG (4) BG22833A3 (US20100154137A1-20100624-C00004.png)
CA (1) CA969180A (US20100154137A1-20100624-C00004.png)
CH (2) CH567501A5 (US20100154137A1-20100624-C00004.png)
CS (4) CS166806B2 (US20100154137A1-20100624-C00004.png)
DD (1) DD96484A5 (US20100154137A1-20100624-C00004.png)
DE (1) DE2107989A1 (US20100154137A1-20100624-C00004.png)
DK (1) DK136721C (US20100154137A1-20100624-C00004.png)
ES (4) ES399875A1 (US20100154137A1-20100624-C00004.png)
FR (1) FR2125599B1 (US20100154137A1-20100624-C00004.png)
GB (1) GB1379781A (US20100154137A1-20100624-C00004.png)
HU (1) HU162947B (US20100154137A1-20100624-C00004.png)
IE (1) IE36116B1 (US20100154137A1-20100624-C00004.png)
IL (1) IL38788A (US20100154137A1-20100624-C00004.png)
NL (1) NL7202153A (US20100154137A1-20100624-C00004.png)
NO (1) NO134055C (US20100154137A1-20100624-C00004.png)
PH (1) PH10385A (US20100154137A1-20100624-C00004.png)
PL (1) PL77393B1 (US20100154137A1-20100624-C00004.png)
RO (4) RO63019A (US20100154137A1-20100624-C00004.png)
SE (1) SE363826B (US20100154137A1-20100624-C00004.png)
SU (3) SU481155A3 (US20100154137A1-20100624-C00004.png)
ZA (1) ZA721072B (US20100154137A1-20100624-C00004.png)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2229770A1 (de) * 1972-06-19 1974-01-10 Boehringer Sohn Ingelheim N-(heteroarylmethyl)-7alpha-acyl6,14-endoaethenotetrahydro-nororipavine und -thebaine, deren hydrierungsprodukte und saeureadditionssalze sowie verfahren zu deren herstellung
DE2230154A1 (de) * 1972-06-21 1974-01-17 Boehringer Sohn Ingelheim N-(heteroaryl-methyl)-6,14-endoaetheno7alpha-hydroxyalkyl-tetrahydro-nororipavine und -thebaine, deren hydrierungsprodukte und saeureadditionssalze sowie verfahren zu deren herstellung
DE2238839A1 (de) * 1972-08-07 1974-02-14 Boehringer Sohn Ingelheim Neue morphinon-derivate, deren saeureadditionssalze, verfahren zu ihrer herstellung sowie ihre verwendung zur herstellung von arzneimitteln
US3923987A (en) * 1972-08-07 1975-12-02 Boehringer Sohn Ingelheim Pharmaceutical compositions containing an n-furyl-or thienyl-methyl)- -oxy-7,8 -dihydro-normorphinone or norcodeinone and method of use
US3975368A (en) * 1972-09-14 1976-08-17 Boehringer Ingelheim Gmbh Pharmaceutical compositions containing an N-(furyl- or thienyl-methyl)-desoxy-normorphine or norcodeine and method of use
DE2245141A1 (de) * 1972-09-14 1974-03-21 Boehringer Sohn Ingelheim Neue n-(heteroarylmethyl)-desoxynormorphine und -norcodeine, deren saeureadditionssalze, verfahren zu deren herstellung sowie deren verwendung als arzneimittel
US4232026A (en) * 1978-07-20 1980-11-04 Merck & Co., Inc. Diazaditwistanes, and pharmaceutical compositions for treating pain in warm blooded animals containing them
US7923454B2 (en) * 2002-05-17 2011-04-12 Jenken Biosciences, Inc. Opioid and opioid-like compounds and uses thereof
GB0421687D0 (en) * 2004-09-30 2004-11-03 Johnson Matthey Plc Preparation of opiate analgesics
GB2438399A (en) * 2006-05-25 2007-11-28 Alpharma Aps Preparation of N-alkylated morphinans by reduction of an iminium group
CA2652849A1 (en) * 2006-05-25 2007-12-06 Alpharma (Bermuda) Investments Ltd. Process useful in the preparation of morphinan antagonists
KR100780932B1 (ko) * 2006-05-30 2007-11-30 엠텍비젼 주식회사 컬러 보간 방법 및 장치
US10766864B2 (en) 2015-05-08 2020-09-08 Nektar Therapeutics Morphinan derivatives for the treatment of neuropathic pain

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE573099A (US20100154137A1-20100624-C00004.png) * 1957-12-04

Also Published As

Publication number Publication date
DE2107989A1 (de) 1972-09-07
CS166805B2 (US20100154137A1-20100624-C00004.png) 1976-03-29
ZA721072B (en) 1973-10-31
SU481155A3 (ru) 1975-08-15
BG20584A3 (bg) 1975-12-05
SU440837A3 (US20100154137A1-20100624-C00004.png) 1974-08-25
BE779582A (fr) 1972-08-18
IL38788A (en) 1975-05-22
AT318599B (de) 1974-10-25
US3793329A (en) 1974-02-19
PH10385A (en) 1977-03-02
NO134055B (US20100154137A1-20100624-C00004.png) 1976-05-03
CS166807B2 (US20100154137A1-20100624-C00004.png) 1976-03-29
AU3914072A (en) 1973-08-23
ES399875A1 (es) 1974-12-01
ES420628A1 (es) 1976-05-01
BG20356A3 (bg) 1975-11-05
CH567503A5 (US20100154137A1-20100624-C00004.png) 1975-10-15
CS166806B2 (US20100154137A1-20100624-C00004.png) 1976-03-29
IE36116B1 (en) 1976-08-18
IE36116L (en) 1972-08-19
RO62412A (fr) 1978-03-15
HU162947B (US20100154137A1-20100624-C00004.png) 1973-05-28
FR2125599B1 (US20100154137A1-20100624-C00004.png) 1975-10-31
CH567501A5 (US20100154137A1-20100624-C00004.png) 1975-10-15
DK136721C (da) 1978-04-24
DD96484A5 (US20100154137A1-20100624-C00004.png) 1973-03-20
GB1379781A (en) 1975-01-08
RO63012A (fr) 1978-05-15
AT312588B (de) 1974-01-10
CS166808B2 (US20100154137A1-20100624-C00004.png) 1976-03-29
FR2125599A1 (US20100154137A1-20100624-C00004.png) 1972-09-29
DK136721B (da) 1977-11-14
SU488411A3 (ru) 1975-10-15
CA969180A (en) 1975-06-10
AT318600B (de) 1974-10-25
NL7202153A (US20100154137A1-20100624-C00004.png) 1972-08-22
IL38788A0 (en) 1972-04-27
AU468490B2 (en) 1976-01-15
BG20357A3 (bg) 1975-11-05
NO134055C (US20100154137A1-20100624-C00004.png) 1976-08-11
RO63262A (fr) 1978-06-15
ES420629A1 (es) 1976-05-01
RO63019A (fr) 1978-05-15
PL77393B1 (US20100154137A1-20100624-C00004.png) 1975-04-30
ES420630A1 (es) 1976-05-01
SE363826B (US20100154137A1-20100624-C00004.png) 1974-02-04
ATA136472A (US20100154137A1-20100624-C00004.png) 1973-12-15
SU466658A3 (ru) 1975-04-05

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