BE884671A - Composes intermediaires pour la preparation de derives de la morphine - Google Patents
Composes intermediaires pour la preparation de derives de la morphineInfo
- Publication number
- BE884671A BE884671A BE0/201677A BE201677A BE884671A BE 884671 A BE884671 A BE 884671A BE 0/201677 A BE0/201677 A BE 0/201677A BE 201677 A BE201677 A BE 201677A BE 884671 A BE884671 A BE 884671A
- Authority
- BE
- Belgium
- Prior art keywords
- preparation
- intermediate compounds
- morphine derivatives
- morphine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US6527579A | 1979-08-09 | 1979-08-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE884671A true BE884671A (fr) | 1980-12-01 |
Family
ID=22061564
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/201677A BE884671A (fr) | 1979-08-09 | 1980-08-07 | Composes intermediaires pour la preparation de derives de la morphine |
Country Status (16)
Country | Link |
---|---|
JP (1) | JPS56501010A (sv) |
AU (1) | AU6116580A (sv) |
BE (1) | BE884671A (sv) |
DD (1) | DD154541A5 (sv) |
DK (1) | DK151781A (sv) |
ES (1) | ES494122A0 (sv) |
FI (1) | FI802479A (sv) |
FR (1) | FR2465735A1 (sv) |
GB (1) | GB2066256A (sv) |
IL (1) | IL60783A0 (sv) |
IT (1) | IT8068267A0 (sv) |
NL (1) | NL8020319A (sv) |
NO (1) | NO802139L (sv) |
PL (1) | PL226162A1 (sv) |
SE (1) | SE8102214L (sv) |
WO (1) | WO1981000409A1 (sv) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4795813A (en) * | 1981-08-17 | 1989-01-03 | The Florida Board Of Regents On Behalf Of The Florida State University | Synthesis of derivatives of codeine and other 3-O-alkylmorphines |
US5668285A (en) * | 1986-10-31 | 1997-09-16 | The United States Of America As Represented By The Department Of Health And Human Services | Total synthesis of northebaine, normophine, noroxymorphone enantiomers and derivatives via N-Nor intermediates |
ATE178329T1 (de) * | 1989-10-16 | 1999-04-15 | Us Health | Totale synthese von northebain-, normorphin-, noroxymorphon-enantiomeren und -derivaten via n- nor-zwischenverbindungen |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3249616A (en) * | 1966-05-03 | Ix-dfflydroxy-g-oxo-n-phenethylmor- phinan (cis) and production thereof | ||
CA913077A (en) * | 1972-10-24 | J. Pachter Irwin | Process of preparing n-substituted 14-hydroxydihydronormorphines | |
US2772270A (en) * | 1954-10-21 | 1956-11-27 | M J Lewenstein | 14-hydroxymorphinone and 8, 14-dihydroxydihydromorphinone |
US2806033A (en) * | 1955-08-03 | 1957-09-10 | Lewenstein | Morphine derivative |
BE638369A (sv) * | 1962-10-10 | |||
US3332950A (en) * | 1963-03-23 | 1967-07-25 | Endo Lab | 14-hydroxydihydronormorphinone derivatives |
NL7106612A (en) * | 1971-05-13 | 1972-11-15 | N-cycloalkylalkyl-14-hydroxy-dihydronormorphines - - by o-demethylation of 14-methoxy cpds | |
US3775414A (en) * | 1972-05-10 | 1973-11-27 | Bristol Myers Co | Process for the preparation of 14-hydroxymorphinan derivatives |
US4161597A (en) * | 1976-12-20 | 1979-07-17 | Research Corporation | N-alkyl-14-hydroxymorphinans and derivatives |
-
1980
- 1980-07-16 NO NO802139A patent/NO802139L/no unknown
- 1980-08-07 AU AU61165/80A patent/AU6116580A/en not_active Abandoned
- 1980-08-07 NL NL8020319A patent/NL8020319A/nl not_active Application Discontinuation
- 1980-08-07 IL IL60783A patent/IL60783A0/xx unknown
- 1980-08-07 JP JP50198480A patent/JPS56501010A/ja active Pending
- 1980-08-07 FI FI802479A patent/FI802479A/fi not_active Application Discontinuation
- 1980-08-07 BE BE0/201677A patent/BE884671A/fr unknown
- 1980-08-07 GB GB8107295A patent/GB2066256A/en not_active Withdrawn
- 1980-08-07 IT IT8068267A patent/IT8068267A0/it unknown
- 1980-08-07 WO PCT/US1980/000998 patent/WO1981000409A1/en active Application Filing
- 1980-08-08 ES ES494122A patent/ES494122A0/es active Granted
- 1980-08-08 FR FR8017530A patent/FR2465735A1/fr not_active Withdrawn
- 1980-08-09 PL PL22616280A patent/PL226162A1/xx unknown
- 1980-09-08 DD DD80223221A patent/DD154541A5/de unknown
-
1981
- 1981-04-03 DK DK151781A patent/DK151781A/da not_active Application Discontinuation
- 1981-04-07 SE SE8102214A patent/SE8102214L/sv unknown
Also Published As
Publication number | Publication date |
---|---|
ES8104296A1 (es) | 1981-04-16 |
AU6116580A (en) | 1981-02-12 |
DK151781A (da) | 1981-04-03 |
WO1981000409A1 (en) | 1981-02-19 |
FR2465735A1 (fr) | 1981-03-27 |
DD154541A5 (de) | 1982-03-31 |
GB2066256A (en) | 1981-07-08 |
PL226162A1 (sv) | 1981-04-24 |
NL8020319A (nl) | 1981-07-01 |
SE8102214L (sv) | 1981-04-07 |
FI802479A (fi) | 1981-02-10 |
JPS56501010A (sv) | 1981-07-23 |
NO802139L (no) | 1981-02-10 |
IL60783A0 (en) | 1980-10-26 |
ES494122A0 (es) | 1981-04-16 |
IT8068267A0 (it) | 1980-08-07 |
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