BE884653A - Nouveaux composes de purine, leur procede de production et composition pharmaceutique les contenant - Google Patents

Nouveaux composes de purine, leur procede de production et composition pharmaceutique les contenant

Info

Publication number
BE884653A
BE884653A BE0/201667A BE201667A BE884653A BE 884653 A BE884653 A BE 884653A BE 0/201667 A BE0/201667 A BE 0/201667A BE 201667 A BE201667 A BE 201667A BE 884653 A BE884653 A BE 884653A
Authority
BE
Belgium
Prior art keywords
producing
pharmaceutical composition
same
composition containing
purine compounds
Prior art date
Application number
BE0/201667A
Other languages
English (en)
French (fr)
Inventor
S Nakagawa
T Naito
T Okita
T Yamasaki
H Yamahita
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of BE884653A publication Critical patent/BE884653A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE0/201667A 1979-08-06 1980-08-06 Nouveaux composes de purine, leur procede de production et composition pharmaceutique les contenant BE884653A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/064,240 US4241063A (en) 1979-08-06 1979-08-06 Purine derivatives and their use as bronchodilators

Publications (1)

Publication Number Publication Date
BE884653A true BE884653A (fr) 1981-02-06

Family

ID=22054538

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/201667A BE884653A (fr) 1979-08-06 1980-08-06 Nouveaux composes de purine, leur procede de production et composition pharmaceutique les contenant

Country Status (5)

Country Link
US (1) US4241063A (en, 2012)
JP (1) JPS57163382A (en, 2012)
AU (1) AU520583B2 (en, 2012)
BE (1) BE884653A (en, 2012)
ZA (1) ZA804701B (en, 2012)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4743689A (en) * 1984-11-20 1988-05-10 Nippon Kayaku Kabushiki Kaisha Antibiotic derivative of adenine
DE3529497A1 (de) * 1985-08-17 1987-02-26 Boehringer Mannheim Gmbh N(pfeil hoch)6(pfeil hoch)-disubstituierte purinderivate, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
US4916225A (en) * 1986-11-25 1990-04-10 Institut Organicheskogo Sinteza Akademii Nauk Latviiskoi Ssr 9-substituted guanines
GB9312853D0 (en) * 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US5591776A (en) * 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
AU695032B2 (en) * 1994-10-05 1998-08-06 Darwin Discovery Limited Purine and guanine compounds as inhibitors of PNP
US6166041A (en) * 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) * 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
US6294541B1 (en) 1996-06-06 2001-09-25 Euro-Celtique S.A. Purine derivatives having phosphodiesterase IV inhibition activity
US5864037A (en) * 1996-06-06 1999-01-26 Euro-Celtique, S.A. Methods for the synthesis of chemical compounds having PDE-IV inhibitory activity
US6057445A (en) 1997-12-12 2000-05-02 Euro-Celtique S.A. Purine compounds having PDE IV inhibitory activity and methods of synthesis
US6319928B1 (en) 1998-11-30 2001-11-20 Euro-Celtique, S.A. Purine derivatives having phosphodiesterase IV inhibition activity
JP2002541078A (ja) 1999-04-02 2002-12-03 ユーロ−セルティーク,エス.エー. ホスホジエステラーゼiv阻害活性を有するプリン誘導体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3228937A (en) * 1963-07-17 1966-01-11 Shell Oil Co Adenine derivative
US3930005A (en) * 1973-06-15 1975-12-30 Squibb & Sons Inc Antiinflammatory agents and their use
US3862189A (en) * 1973-08-14 1975-01-21 Warner Lambert Co Aralkyl-substituted purines and pyrimidines as antianginal bronchodilator agents
US3917837A (en) * 1974-10-21 1975-11-04 American Cyanamid Co Method of using trans-2-(6-amino-9H-purin-9-yl)-cyclopentanol
JPS5271492A (en) * 1975-12-10 1977-06-14 Kohjin Co Ltd Synthesis of 9-substituted-2-substituted thioadenines

Also Published As

Publication number Publication date
JPH0222075B2 (en, 2012) 1990-05-17
JPS57163382A (en) 1982-10-07
AU6102180A (en) 1981-02-12
US4241063A (en) 1980-12-23
AU520583B2 (en) 1982-02-11
ZA804701B (en) 1981-10-28

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