BE871401A - Azetidinones monocycliques antibiotiques - Google Patents

Azetidinones monocycliques antibiotiques

Info

Publication number
BE871401A
BE871401A BE1009107A BE1009107A BE871401A BE 871401 A BE871401 A BE 871401A BE 1009107 A BE1009107 A BE 1009107A BE 1009107 A BE1009107 A BE 1009107A BE 871401 A BE871401 A BE 871401A
Authority
BE
Belgium
Prior art keywords
azetidinones
monocyclic
antibiotics
monocyclic antibiotics
azetidinones monocyclic
Prior art date
Application number
BE1009107A
Other languages
English (en)
Inventor
D K Herron
C A Whitesitt
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BE871401A publication Critical patent/BE871401A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
BE1009107A 1977-10-26 1978-10-20 Azetidinones monocycliques antibiotiques BE871401A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/845,766 US4195021A (en) 1977-10-26 1977-10-26 1,3-Disubstituted 2-azetidinone antibitotics

Publications (1)

Publication Number Publication Date
BE871401A true BE871401A (fr) 1979-04-20

Family

ID=25296053

Family Applications (1)

Application Number Title Priority Date Filing Date
BE1009107A BE871401A (fr) 1977-10-26 1978-10-20 Azetidinones monocycliques antibiotiques

Country Status (7)

Country Link
US (1) US4195021A (fr)
EP (1) EP0001715A3 (fr)
JP (1) JPS5470256A (fr)
BE (1) BE871401A (fr)
FR (1) FR2407203A1 (fr)
GB (1) GB2008574A (fr)
IL (1) IL55779A0 (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4472300A (en) * 1977-12-07 1984-09-18 Fujisawa Pharmaceutical Co., Ltd. Azetidinone derivatives and process for preparation thereof
US4263306A (en) * 1979-08-01 1981-04-21 Merck & Co., Inc. 3-N-Pyridinium nocardicin and antibiotic composition thereof
US4337197A (en) 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates
NZ199981A (en) * 1981-04-09 1985-08-16 Squibb & Sons Inc 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines
US4595532A (en) * 1983-02-02 1986-06-17 University Of Notre Dame Du Lac N-(substituted-methyl)-azetidin-2-ones
IL70782A (en) * 1983-02-02 1991-03-10 Univ Notre Dame Du Lac N-dicarboxymethyl azetidin-2-ones
UA77200C2 (en) 2001-08-07 2006-11-15 Wyeth Corp Antineoplastic combination of cci-779 and bkb-569
CL2004000016A1 (es) * 2003-01-21 2005-04-15 Wyeth Corp Compuesto derivado de cloruro de 4-amino-2-butenoilo o una sal farmaceuticamente aceptable del mismo; procedimiento para preparar dicho compuesto, util como intermediario en la sintesis de compuestos inhibidores de proteina quinasa tirosina.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2143211B1 (fr) * 1971-06-24 1975-10-31 Fujisawa Pharmaceutical Co
FR2278335A1 (fr) 1974-07-04 1976-02-13 Fujisawa Pharmaceutical Co Derives d'azetidinones et leurs procedes de preparation
CH618161A5 (en) * 1974-07-04 1980-07-15 Fujisawa Pharmaceutical Co Process for the preparation of azetidinone derivatives
GB1570278A (en) * 1975-10-06 1980-06-25 Fujisawa Pharmaceutical Co O-substituted-2-azetidinone derivatives and the preparation thereof
JPS6019315B2 (ja) * 1976-01-23 1985-05-15 塩野義製薬株式会社 アゼチジノン化合物

Also Published As

Publication number Publication date
EP0001715A3 (fr) 1979-05-16
FR2407203A1 (fr) 1979-05-25
US4195021A (en) 1980-03-25
GB2008574A (en) 1979-06-06
EP0001715A2 (fr) 1979-05-02
JPS5470256A (en) 1979-06-05
IL55779A0 (en) 1978-12-17

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