BE844449A - Procede d'obtention de preparation pharmaceutiques stables pour usage oral, contenant des derives d'homopyrimidazole - Google Patents

Procede d'obtention de preparation pharmaceutiques stables pour usage oral, contenant des derives d'homopyrimidazole

Info

Publication number
BE844449A
BE844449A BE169173A BE169173A BE844449A BE 844449 A BE844449 A BE 844449A BE 169173 A BE169173 A BE 169173A BE 169173 A BE169173 A BE 169173A BE 844449 A BE844449 A BE 844449A
Authority
BE
Belgium
Prior art keywords
pharmaceutical preparations
oral use
stable pharmaceutical
obtaining stable
homopyrimidazole
Prior art date
Application number
BE169173A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE844449A publication Critical patent/BE844449A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BE169173A 1975-07-25 1976-07-23 Procede d'obtention de preparation pharmaceutiques stables pour usage oral, contenant des derives d'homopyrimidazole BE844449A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU75CI1596A HU173823B (hu) 1975-07-25 1975-07-25 Sposob poluchenija stabil'nogo lechebnogo preparata dlja oral'noj dozirovki, kotoryj soderzhit proizvodnyj gomopirimidazola

Publications (1)

Publication Number Publication Date
BE844449A true BE844449A (fr) 1976-11-16

Family

ID=10994575

Family Applications (1)

Application Number Title Priority Date Filing Date
BE169173A BE844449A (fr) 1975-07-25 1976-07-23 Procede d'obtention de preparation pharmaceutiques stables pour usage oral, contenant des derives d'homopyrimidazole

Country Status (6)

Country Link
JP (1) JPS5215813A (de)
AT (1) AT342761B (de)
BE (1) BE844449A (de)
FI (1) FI762087A (de)
FR (1) FR2318636A1 (de)
HU (1) HU173823B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU183408B (en) * 1981-04-28 1984-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing oral ratard pharmaceutical compositions
JPS59112594A (ja) * 1982-12-17 1984-06-29 松下電器産業株式会社 加熱装置
HU222489B1 (hu) * 1990-07-25 2003-07-28 Novartis Ag. Stabilizált gyógyszerkészítmények és eljárás az előállításukra
FR2665834B1 (fr) * 1991-07-24 2001-02-23 Sandoz Sa Composition pharmaceutique stabilisee par un donneur d'acide chlorhydrique, et sa preparation.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH538494A (de) * 1966-11-02 1973-06-30 Chinoin Gyogyszer Es Vegyeszet Verfahren zur Herstellung neuer Homopyrimidazol-Derivate

Also Published As

Publication number Publication date
FR2318636A1 (fr) 1977-02-18
ATA529576A (de) 1977-08-15
JPS5215813A (en) 1977-02-05
FR2318636B1 (de) 1979-01-12
FI762087A (de) 1977-01-26
HU173823B (hu) 1979-08-28
AT342761B (de) 1978-04-25

Similar Documents

Publication Publication Date Title
NL930110I2 (nl) Carbazolyl-(4)-oxypropanolamine-derivaten, werkwijze ter bereiding daarvan en geneesmiddelen, die deze verbindingen bevatten.
BE896986A (fr) Derives d'indole, procedes pour leur preparation et composition pharmaceutiques les contenant
FR2290912A1 (fr) Formulations pharmaceutiques contenant de la l-dopa ou ses derives
FR2595351B1 (fr) Derives d'indole, procede pour leur preparation et compositions pharmaceutiques les contenant
DE2861289D1 (en) Imidazolidine derivatives, process for their preparation, intermediates for use in this process, pharmaceutical compositions containing them and the use of the active compounds
MA18829A1 (fr) Derives de la pyrimidine,procedes pour leur preparation,compositions pharmaceutiques contenant ces composes et leur utilisation therapeutique
ZA79154B (en) New derivatives of tetrahydropyridinyl indole and their salts,the process for preparing,and the pharmaceutical compositions containing,these new products
BE865851A (fr) Dipyrido(4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant
BE849810A (fr) Nouvelles pyrimidones, procede pour les preparation et compositions pharmaceutiques les contenant
LU81132A1 (fr) 2-(2-thenoylthio)-propionylglycine,procede pour sa preparation et compositions pharmaceutiques la contenant
FR2411839B1 (fr) Derives de l'acide cephalosporanique, procedes pour leur preparation et composition pharmaceutique les contenant
BE839932A (fr) Derives de nitrofurylpyrazole, procedes pour leur preparation, et medicaments contenant ces compose
FR2485537B2 (fr) Dipyrido(4,3-b)(3,4-f)indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant
BE837848A (fr) Thiourees et thiocarbamates, procede pour les preparer et compositions pharmaceutiques les contenant
BE874252A (fr) Nouvelles 2-phenylimino-imidazolidines substituees, leurs sels d'addition avec des acides, medicaments les renfermant et procedes pour leur preparation
BE842118A (fr) Nouvelles propargyl-2-phenylamino-imidazolines-(2), leurs sels d'addition avec des acides, les medicaments les renfermant et procedes pour leur preparation
BE809179A (fr) Nouvelles cyclopropylamines, leur procede d'obtention et les compositions pharmaceutiques en contenant
BE874253A (fr) Nouvelles 2-phenylimino-imidazolidines substituees, leurs sels d'addition avec des acides, medicaments les renfermant et procedes pour leur preparation
BE844449A (fr) Procede d'obtention de preparation pharmaceutiques stables pour usage oral, contenant des derives d'homopyrimidazole
FR2321888A1 (fr) N-tetrahydrofurfuryl-noroxymorphones, leurs sels d'addition avec des acides, procedes pour leur preparation et medicaments en renfermant
RO77772A (ro) Procedeu pentru prepararea unor derivati de acizi 2,2-dimetilciclo‡ropancarboxilici
BE884101A (fr) Derives d'isoquinoleine contenant du soufre, procedes pour leur preparation et composition pharmaceutiques les contenant
MA18628A1 (fr) Procede d'obtention de nouvelles compositions pharmaceutiques a base d'aryltrigluoroethanol
BE875091A (fr) Derives de substitution de spirooxazolidinone steroidienne, leur procede de preparation et compositions pharmaceutiques les contenant
PT65151A (fr) Procede pour la preparation de nouvelles solutions pharmaceutiques stables

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT

Effective date: 19860731