BE802233A - Procede pour la preparation de derives de benzodiazepine - Google Patents

Procede pour la preparation de derives de benzodiazepine

Info

Publication number
BE802233A
BE802233A BE133378A BE133378A BE802233A BE 802233 A BE802233 A BE 802233A BE 133378 A BE133378 A BE 133378A BE 133378 A BE133378 A BE 133378A BE 802233 A BE802233 A BE 802233A
Authority
BE
Belgium
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
BE133378A
Other languages
English (en)
French (fr)
Inventor
A Walser
L H Sternbach
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BE802233A publication Critical patent/BE802233A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
BE133378A 1972-07-13 1973-07-12 Procede pour la preparation de derives de benzodiazepine BE802233A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US271434A US3879406A (en) 1972-07-13 1972-07-13 Preparation of triazolobenzodiazepines

Publications (1)

Publication Number Publication Date
BE802233A true BE802233A (fr) 1974-01-14

Family

ID=23035548

Family Applications (1)

Application Number Title Priority Date Filing Date
BE133378A BE802233A (fr) 1972-07-13 1973-07-12 Procede pour la preparation de derives de benzodiazepine

Country Status (13)

Country Link
US (1) US3879406A (ja)
JP (1) JPS50100093A (ja)
AU (1) AU5803673A (ja)
BE (1) BE802233A (ja)
CH (1) CH580605A5 (ja)
DD (1) DD107692A5 (ja)
DE (1) DE2335281A1 (ja)
FR (2) FR2192827B1 (ja)
GB (2) GB1442222A (ja)
IL (1) IL42721A0 (ja)
LU (1) LU68005A1 (ja)
NL (1) NL7309733A (ja)
ZA (1) ZA734256B (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3954728A (en) * 1972-07-13 1976-05-04 Hoffman-La Roche Inc. Preparation of triazolo benzodiazepines and novel compounds
JPS58427B2 (ja) * 1974-07-25 1983-01-06 武田薬品工業株式会社 4−(ピリジンカルボニル)フェニル−1,2,4−トリアゾ−ル誘導体の製造法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE412325A (ja) * 1961-02-10 1900-01-01
US3182065A (en) * 1964-04-09 1965-05-04 Hoffmann La Roche 2-acetamidobenzoyl-pyridines
JPS4837280B1 (ja) * 1969-03-08 1973-11-09
JPS4927880B1 (ja) * 1969-10-23 1974-07-22
US3734922A (en) * 1971-05-11 1973-05-22 Upjohn Co Certain 4h-s-triazolo(4,3-a)(1,4)benzodiazepines
US3681343A (en) * 1971-05-11 1972-08-01 Upjohn Co 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines
US3701782A (en) * 1972-02-10 1972-10-31 Upjohn Co 1-carbolower alkoxy - 6 - phenyl-4h-s-triazolo(1,4)benzodiazepine compounds

Also Published As

Publication number Publication date
IL42721A0 (en) 1973-10-25
CH580605A5 (ja) 1976-10-15
GB1442222A (en) 1976-07-14
NL7309733A (ja) 1974-01-15
FR2192827B1 (ja) 1977-12-16
DD107692A5 (ja) 1974-08-12
AU5803673A (en) 1975-01-16
GB1442221A (en) 1976-07-14
DE2335281A1 (de) 1974-01-31
ZA734256B (en) 1974-02-27
FR2192827A1 (ja) 1974-02-15
JPS50100093A (ja) 1975-08-08
FR2275464B1 (ja) 1977-07-22
FR2275464A1 (fr) 1976-01-16
LU68005A1 (ja) 1975-04-11
US3879406A (en) 1975-04-22

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