BE762711A - Pyrazolopyridine carboxylic acids antimicro - bial tranquillising anti asthma agents - Google Patents

Pyrazolopyridine carboxylic acids antimicro - bial tranquillising anti asthma agents

Info

Publication number
BE762711A
BE762711A BE762711A BE762711A BE762711A BE 762711 A BE762711 A BE 762711A BE 762711 A BE762711 A BE 762711A BE 762711 A BE762711 A BE 762711A BE 762711 A BE762711 A BE 762711A
Authority
BE
Belgium
Prior art keywords
lower alkyl
phenyl
tranquillising
carboxylic acids
antimicro
Prior art date
Application number
BE762711A
Other languages
French (fr)
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR707022122A external-priority patent/FR2052975B1/fr
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of BE762711A publication Critical patent/BE762711A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Pyrazolopyridine carboxylic acids - antimicrobial, tranquillising, anti-asthma agents Cpds. of general formula (I) : (where R = aliphatic 1-12 C radical or phenyl-lower alkyl; R1 = H or lower alkyl; R2 = lower alkyl, phenyl-lower alkyl, substd. phenyl-lower alkyl or cycloalkyl-lower alkyl; R3 = H, lower alkyl, phenyl or substd. phenyl. (I) have antimicrobial activity and may be used against infections caused by Trichomonas vaginalis, Staphylococcus aureus and Trichophyton mentagrophytes. They may also be used as surface-disinfectants in water, powders, sprays, soaps, detergents etc. (I) have CNS- inhibitory activity and may be used as tranquillisers. (I) increase the intracellular concn. of adenosine-31, 51-cyclic monophosphate and may be used in the treatment of asthma. Intermediates (II) have bloodsugar-lowering activity in mammals.
BE762711A 1969-06-16 1971-02-09 Pyrazolopyridine carboxylic acids antimicro - bial tranquillising anti asthma agents BE762711A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83367369A 1969-06-16 1969-06-16
FR707022122A FR2052975B1 (en) 1969-06-16 1970-06-16

Publications (1)

Publication Number Publication Date
BE762711A true BE762711A (en) 1971-07-16

Family

ID=26215797

Family Applications (1)

Application Number Title Priority Date Filing Date
BE762711A BE762711A (en) 1969-06-16 1971-02-09 Pyrazolopyridine carboxylic acids antimicro - bial tranquillising anti asthma agents

Country Status (1)

Country Link
BE (1) BE762711A (en)

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