BE750524A - Nouveaux derives de benzodiazephine et leurs sels - Google Patents

Nouveaux derives de benzodiazephine et leurs sels

Info

Publication number
BE750524A
BE750524A BE750524DA BE750524A BE 750524 A BE750524 A BE 750524A BE 750524D A BE750524D A BE 750524DA BE 750524 A BE750524 A BE 750524A
Authority
BE
Belgium
Prior art keywords
benzodiazephine
derivatives
salts
new
new benzodiazephine
Prior art date
Application number
Other languages
English (en)
Inventor
H Yamamoto
S Inaba
T Hirohashi
M Yamamoto
K Ishizumi
M Akatsu
I Maruyama
Y Kume
K Mori
T Izumi
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of BE750524A publication Critical patent/BE750524A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/26Preparation from compounds already containing the benzodiazepine skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/30Preparation including building-up the benzodiazepine skeleton from compounds already containing hetero rings
    • C07D243/36Preparation including building-up the benzodiazepine skeleton from compounds already containing hetero rings containing an indole or hydrogenated indole ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE750524D 1969-05-16 1970-05-15 Nouveaux derives de benzodiazephine et leurs sels BE750524A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP44038183A JPS4811718B1 (fr) 1969-05-16 1969-05-16

Publications (1)

Publication Number Publication Date
BE750524A true BE750524A (fr) 1970-10-16

Family

ID=12518255

Family Applications (1)

Application Number Title Priority Date Filing Date
BE750524D BE750524A (fr) 1969-05-16 1970-05-15 Nouveaux derives de benzodiazephine et leurs sels

Country Status (12)

Country Link
JP (1) JPS4811718B1 (fr)
AT (2) AT300815B (fr)
BE (1) BE750524A (fr)
CA (1) CA946844A (fr)
CH (1) CH537396A (fr)
CS (1) CS169804B2 (fr)
ES (2) ES379701A1 (fr)
FR (1) FR2051534B1 (fr)
GB (1) GB1272887A (fr)
NL (1) NL161749C (fr)
SE (1) SE372269B (fr)
ZA (1) ZA703130B (fr)

Also Published As

Publication number Publication date
NL7007057A (fr) 1970-11-18
NL161749B (nl) 1979-10-15
DE2023182A1 (de) 1970-11-19
CA946844A (en) 1974-05-07
NL161749C (nl) 1980-03-17
ES379701A1 (es) 1972-08-01
FR2051534B1 (fr) 1974-04-12
JPS4811718B1 (fr) 1973-04-14
GB1272887A (en) 1972-05-03
ES383587A1 (es) 1973-01-01
CH537396A (de) 1973-05-31
ZA703130B (en) 1971-01-27
CS169804B2 (fr) 1976-07-29
SE372269B (fr) 1974-12-16
FR2051534A1 (fr) 1971-04-09
AT308125B (de) 1973-06-25
AT300815B (de) 1972-08-10
DE2023182B2 (de) 1975-08-28

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