BE1003340A3 - Nouvelle utilisation therapeutique des alpha-aminofluorocetones. - Google Patents
Nouvelle utilisation therapeutique des alpha-aminofluorocetones. Download PDFInfo
- Publication number
- BE1003340A3 BE1003340A3 BE9000075A BE9000075A BE1003340A3 BE 1003340 A3 BE1003340 A3 BE 1003340A3 BE 9000075 A BE9000075 A BE 9000075A BE 9000075 A BE9000075 A BE 9000075A BE 1003340 A3 BE1003340 A3 BE 1003340A3
- Authority
- BE
- Belgium
- Prior art keywords
- alpha
- aminofluorocetones
- therapeutic use
- new therapeutic
- phenylalanylalanylfluoromethylketone
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/005—Enzyme inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pyrrole Compounds (AREA)
Abstract
La présente invention a pour objet l'utilisation d'alpha-aminofluorocétones, spécialement la benzyloxycarbonyl-1-phénylalanylalanylfluorométhylcétone, pour la préparation de médicaments ayant une activité cardiovasculaire et anti-hypertensive.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH23889 | 1989-01-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE1003340A3 true BE1003340A3 (fr) | 1992-03-03 |
Family
ID=4182438
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE9000075A BE1003340A3 (fr) | 1989-01-26 | 1990-01-22 | Nouvelle utilisation therapeutique des alpha-aminofluorocetones. |
Country Status (6)
Country | Link |
---|---|
JP (1) | JPH02247123A (fr) |
BE (1) | BE1003340A3 (fr) |
DE (1) | DE4001087A1 (fr) |
FR (1) | FR2641972A1 (fr) |
GB (1) | GB2227411A (fr) |
IT (1) | IT1239745B (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5101068A (en) * | 1990-02-16 | 1992-03-31 | Prototek Inc. | Magnesium fluoromalonates |
JP3228347B2 (ja) * | 1991-06-25 | 2001-11-12 | 三菱化学株式会社 | シクロプロペノン誘導体 |
US5395958A (en) * | 1992-09-30 | 1995-03-07 | Mitsubishi Kasei Corporation | Cyclopropene derivatives |
ATE197591T1 (de) * | 1995-03-31 | 2000-12-15 | Naeja Pharmaceutical Inc | 4-substituierte-3-peptidyl-azetidin-2-on-deriva e als cystein-proteinase inhibitoren |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4518528A (en) * | 1983-05-19 | 1985-05-21 | Rasnick David W | α Amino fluoro ketones |
-
1990
- 1990-01-17 DE DE4001087A patent/DE4001087A1/de not_active Withdrawn
- 1990-01-22 GB GB9001453A patent/GB2227411A/en not_active Withdrawn
- 1990-01-22 FR FR9000777A patent/FR2641972A1/fr active Pending
- 1990-01-22 BE BE9000075A patent/BE1003340A3/fr not_active IP Right Cessation
- 1990-01-22 IT IT47551A patent/IT1239745B/it active IP Right Grant
- 1990-01-25 JP JP2015948A patent/JPH02247123A/ja active Pending
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4518528A (en) * | 1983-05-19 | 1985-05-21 | Rasnick David W | α Amino fluoro ketones |
Non-Patent Citations (2)
Title |
---|
CHEMICAL ABSTRACTS, vol. 108, no. 17, 25 avril 1988, page 798, abr�g� no. 150981h, Columbus, Ohio, US; & ZA-A-86 06 642 (MERCK & CO., INC.) 29-04-1987 * |
CHEMICAL ABSTRACTS, vol. 86, no. 11, 14 mars 1977, page 186, abr�g� no. 67205q, Columbus, Ohio, US; V.N. OREKHOVICH et al.: "Enzymological factors in vascular tension regulation", & VESTN. AKAD. MED. NAUK. SSSR 1976, (9), 42-7 * |
Also Published As
Publication number | Publication date |
---|---|
IT1239745B (it) | 1993-11-15 |
JPH02247123A (ja) | 1990-10-02 |
DE4001087A1 (de) | 1990-08-02 |
IT9047551A0 (it) | 1990-01-22 |
GB9001453D0 (en) | 1990-03-21 |
GB2227411A (en) | 1990-08-01 |
FR2641972A1 (fr) | 1990-07-27 |
IT9047551A1 (it) | 1990-07-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: S.A. SANDOZ Effective date: 19920131 |