AU9144491A - Method of preparing "syn" derivatives of propanamide - Google Patents

Method of preparing "syn" derivatives of propanamide

Info

Publication number
AU9144491A
AU9144491A AU91444/91A AU9144491A AU9144491A AU 9144491 A AU9144491 A AU 9144491A AU 91444/91 A AU91444/91 A AU 91444/91A AU 9144491 A AU9144491 A AU 9144491A AU 9144491 A AU9144491 A AU 9144491A
Authority
AU
Australia
Prior art keywords
propanamide
syn
preparing
derivatives
camphosultam
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU91444/91A
Other versions
AU652018B2 (en
Inventor
Thierry Aubert
Xavier Radisson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Rhone Poulenc Rorer SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer SA filed Critical Rhone Poulenc Rorer SA
Publication of AU9144491A publication Critical patent/AU9144491A/en
Application granted granted Critical
Publication of AU652018B2 publication Critical patent/AU652018B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Abstract

Method for preparing a 'syn' derivative of propanamide of forumula (I) by the action of a derivative of camphosultam of general formula (II) or (III) on aldehyde of formula (IV) in the presence of a Lewis acid and an organic base. In formulae (I) to (IV), X is a halogen atom, R is an alkyl, aryl or heteroaryl radical, R1? is the residue of one or other of the camphosultam enantiomers. The products obtained by the method may be used in the preparation of therapeutically active products.
AU91444/91A 1990-12-18 1991-12-17 Method of preparing "SYN" derivatives of propanamide Ceased AU652018B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9015814A FR2670490B1 (en) 1990-12-18 1990-12-18 PROCESS FOR THE PREPARATION OF "SYN" DERIVATIVES OF PROPANAMIDE.
FR9015814 1990-12-18
PCT/FR1991/001019 WO1992011250A1 (en) 1990-12-18 1991-12-17 Method of preparing 'syn' derivatives of propanamide

Publications (2)

Publication Number Publication Date
AU9144491A true AU9144491A (en) 1992-07-22
AU652018B2 AU652018B2 (en) 1994-08-11

Family

ID=9403335

Family Applications (1)

Application Number Title Priority Date Filing Date
AU91444/91A Ceased AU652018B2 (en) 1990-12-18 1991-12-17 Method of preparing "SYN" derivatives of propanamide

Country Status (22)

Country Link
EP (1) EP0563219B1 (en)
JP (1) JPH06503572A (en)
KR (1) KR930703277A (en)
AT (1) ATE114646T1 (en)
AU (1) AU652018B2 (en)
CA (1) CA2098583A1 (en)
CZ (1) CZ115393A3 (en)
DE (1) DE69105524D1 (en)
ES (1) ES2065163T3 (en)
FI (1) FI932812A (en)
FR (1) FR2670490B1 (en)
GR (1) GR3014892T3 (en)
HU (1) HUT68144A (en)
IE (1) IE914396A1 (en)
MX (1) MX9102629A (en)
NO (1) NO931918L (en)
NZ (1) NZ241025A (en)
PT (1) PT99854A (en)
SK (1) SK62093A3 (en)
WO (1) WO1992011250A1 (en)
YU (1) YU195391A (en)
ZA (1) ZA919882B (en)

Also Published As

Publication number Publication date
WO1992011250A1 (en) 1992-07-09
KR930703277A (en) 1993-11-29
NO931918D0 (en) 1993-05-26
MX9102629A (en) 1992-10-01
FI932812A0 (en) 1993-06-17
FI932812A (en) 1993-06-17
DE69105524D1 (en) 1995-01-12
CA2098583A1 (en) 1992-06-19
FR2670490A1 (en) 1992-06-19
CZ115393A3 (en) 1994-02-16
ES2065163T3 (en) 1995-02-01
GR3014892T3 (en) 1995-05-31
ZA919882B (en) 1992-09-30
HU9301770D0 (en) 1993-09-28
IE914396A1 (en) 1992-07-01
NO931918L (en) 1993-05-26
FR2670490B1 (en) 1994-09-23
JPH06503572A (en) 1994-04-21
EP0563219B1 (en) 1994-11-30
YU195391A (en) 1994-01-20
PT99854A (en) 1992-12-31
ATE114646T1 (en) 1994-12-15
AU652018B2 (en) 1994-08-11
SK62093A3 (en) 1993-11-10
NZ241025A (en) 1993-04-28
EP0563219A1 (en) 1993-10-06
HUT68144A (en) 1995-05-29

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