AU7869081A - Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates - Google Patents

Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates

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Publication number
AU7869081A
AU7869081A AU78690/81A AU7869081A AU7869081A AU 7869081 A AU7869081 A AU 7869081A AU 78690/81 A AU78690/81 A AU 78690/81A AU 7869081 A AU7869081 A AU 7869081A AU 7869081 A AU7869081 A AU 7869081A
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AU
Australia
Prior art keywords
carbon atoms
alkyl
optionally substituted
case
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU78690/81A
Other versions
AU547689B2 (en
Inventor
Wilhelm Brandes
Karl Heinz Buchel
Hans-Ludwig Elbe
Paul-Ernst Frohberger
Udo Kraatz
Wolfgang Kramer
Erik Regel
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Bayer AG
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Bayer AG
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Application filed by Bayer AG filed Critical Bayer AG
Publication of AU7869081A publication Critical patent/AU7869081A/en
Application granted granted Critical
Publication of AU547689B2 publication Critical patent/AU547689B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/04—Saturated compounds containing keto groups bound to acyclic carbon atoms
    • C07C49/16—Saturated compounds containing keto groups bound to acyclic carbon atoms containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Abstract

1. Substituted 1-azolyl-butan-2-ones of the formula see diagramm : EP0054865,P68,F1 in which Az represents 1,2,4-triazol-1-yl and 4-yl or imidazol-1-yl ; R**1 represents hydrogen, alkyl with 1 to 12 and alkenyl and alkinyl with in each case 2 to 12 carbon atoms, and represents optionally C1 -C4 -alkyl-substituted cycloalkyl with 3 to 7 carbon atoms or cycloalkylalkyl with 3 to 7 carbon atoms in the cycloalkyl part and 1 to 4 carbon atoms in the alkyl part, and represents optionally substituted phenoxyalkyl with 1 to 4 carbon atoms in the alkyl part or optionally substituted phenylalkyl with 1 to 4 carbon atoms in the alkyl part, the phenyl substituents to be mentioned in each case being : halogen ; alkyl, alkoxy and alkylthio with in each case 1 to 6 carbon atoms ; cyclohexyl ; dialkylamino with in each case 1 to 4 carbon atoms in each alkyl part ; halogenoalkyl, halogenoalkoxy and halogenoalkylthio with in each case 1 to 4 carbon atoms and 1 to 5 identical or different halogen atoms ; nitro ; cyano ; alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl part ; and optionally halogensubstituted phenyl and phenoxy ; and the grouping -CO-NR**6 R**7 ; n represents the numbers 0 or 1, R**2 represents cyano or the groupings -X-R**3 and -CO-NR**4 R**5 , and, in the case where n does not represent 0 at the same time as R**1 represents hydrogen and Az represents 1,2,4-triazolyl, also additionally represents optionally substituted aryl with 6 to 10 carbon atoms, possible substituents being the aryl substituents already mentioned under R**1 , and represents alkoxycarbonyl with 1 to 4 carbon atoms in the alkyl part ; X represents oxygen, sulphur, or the SO or SO2 group, R**3 represents alkyl with 1 to 6 carbon atoms, halogenoalkyl with 1 to 4 carbon atoms and 1 to 5 identical or different halogen atoms, and represents optionally substituted aryl with 6 to 10 carbon atoms and aralkyl with 6 to 10 carbon atoms in the aryl part and 1 to 2 carbon atoms in the alkyl part, possible substituents being the aryl substituents already mentioned under R**1 ; R**4 represents hydrogen, alkyl with 1 to 4 carbon atoms or optionally substituted aryl with 1 to 10 carbon atoms, possible substituents being the aryl substituents already mentioned under R**1 ; R**5 represents hydrogen or alkyl with 1 to 4 carbon atoms ; and R**6 and R**7 represent hydrogen, alkyl with 1 to 4 carbon atoms, phenyl which is optionally substituted by halogen and alkyl with 1 to 4 carbon atoms, or both together with the adjacent nitrogen atom represent a saturated 5- or 6-membered ring system which can contain nitrogen or oxygen as additional hetero atoms ; and plant-tolerated acid addition salts and metal salt complexes thereof.
AU78690/81A 1980-12-20 1981-12-21 Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates Ceased AU547689B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19803048266 DE3048266A1 (en) 1980-12-20 1980-12-20 SUBSTITUTED 1-AZOLYL-BUTANE-2ONE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS FUNGICIDES AND AS INTERMEDIATE PRODUCTS
DE30482667 1980-12-20

Publications (2)

Publication Number Publication Date
AU7869081A true AU7869081A (en) 1982-07-01
AU547689B2 AU547689B2 (en) 1985-10-31

Family

ID=6119802

Family Applications (1)

Application Number Title Priority Date Filing Date
AU78690/81A Ceased AU547689B2 (en) 1980-12-20 1981-12-21 Substituted 1-azolyl-butan-2-ones, their starting compounds and their intermediates

Country Status (15)

Country Link
EP (1) EP0054865B1 (en)
JP (1) JPS57128676A (en)
AT (1) ATE18213T1 (en)
AU (1) AU547689B2 (en)
BR (1) BR8108274A (en)
CA (1) CA1178587A (en)
DE (2) DE3048266A1 (en)
DK (1) DK563081A (en)
EG (1) EG15306A (en)
ES (1) ES8300712A1 (en)
GR (1) GR77634B (en)
HU (1) HU189549B (en)
IL (1) IL64572A (en)
PT (1) PT74109B (en)
ZA (1) ZA818757B (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3209431A1 (en) * 1982-03-16 1983-09-22 Bayer Ag, 5090 Leverkusen PHENOXYPROPYLTRIAZOLYL KETONES AND CARBINOLS, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS FUNGICIDES
DE3229274A1 (en) * 1982-08-05 1984-02-09 Bayer Ag, 5090 Leverkusen SUBSTITUTED AZOLYLVINYL KETONES AND CARBINOLS
DE3229273A1 (en) * 1982-08-05 1984-02-09 Bayer Ag, 5090 Leverkusen SUBSTITUTED AZOLYLALLYL KETONES AND CARBINOLS
DE3313941A1 (en) * 1983-04-15 1984-10-18 Schering AG, 1000 Berlin und 4709 Bergkamen 4-AZOLYL-PENTANNITRILE, METHOD FOR THE PRODUCTION OF THESE COMPOUNDS AND THE BIOCIDES CONTAINING THEM
DE3322526A1 (en) * 1983-06-23 1985-01-10 Basf Ag, 6700 Ludwigshafen FUNGICIDAL AZOL COMPOUNDS, THEIR PRODUCTION AND USE
DE3329128A1 (en) * 1983-08-11 1985-02-28 Bayer Ag, 5090 Leverkusen 3-CYCLOALKYL-1- (1,3-DIOXAN-5-YL) -2- (1,2,4-TRIAZOL-1-YL) -PROPAN-1-ONE AND -PROPAN-1-OLE
DE3336861A1 (en) * 1983-10-11 1985-04-25 Bayer Ag, 5090 Leverkusen AZOLYL-TETRAHYDROFURAN-2-YLIDEN-METHANE DERIVATIVES
DE3434158A1 (en) * 1984-09-18 1986-03-20 Bayer Ag, 5090 Leverkusen SUBSTITUTED 1,1-BIS-AZOLYL-BUTAN-2-ONE AND -OLE
DE3702962A1 (en) * 1987-01-31 1988-08-11 Bayer Ag PYRIMIDINE DERIVATIVE-BASED PEST CONTROL
DE3725397A1 (en) * 1987-07-31 1989-02-09 Bayer Ag 1,4-DISUBSTITUTED 1-AZOLYL-3,3-DIMETHYLBUTANE DERIVATIVES
DE3813253A1 (en) * 1988-04-20 1989-11-02 Bayer Ag SUBSTITUTED TRIAZOLYL METHYLCARBINOLS
USRE37303E1 (en) * 1992-01-10 2001-07-31 Institut National Del La Sante Et De La Recherche Medicale Imidazole compounds and their therapeutic applications
FR2686084B1 (en) * 1992-01-10 1995-12-22 Bioprojet Soc Civ NEW IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATIONS.
DE4222542A1 (en) * 1992-07-09 1994-01-13 Bayer Ag Triazolyl butane derivatives
DE4222541A1 (en) * 1992-07-09 1994-01-13 Bayer Ag Triazolyl butane derivatives
DE4318916A1 (en) * 1993-06-07 1994-12-08 Bayer Ag Cyclobutylazole

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2842137A1 (en) * 1978-09-28 1980-04-17 Bayer Ag HALOGENED 1-AZOLYL-1-FLUORPHENOXYBUTANE DERIVATIVES, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE AS FUNGICIDES
DE2951164A1 (en) * 1979-12-19 1981-07-16 Bayer Ag, 5090 Leverkusen SUBSTITUTED TRIAZOLYL METHYL-TERT.-BUTYL-KETONE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A PLANT PROTECTANT AND AS AN INTERMEDIATE PRODUCT

Also Published As

Publication number Publication date
EG15306A (en) 1986-09-30
ATE18213T1 (en) 1986-03-15
PT74109B (en) 1983-05-16
IL64572A (en) 1985-05-31
DK563081A (en) 1982-06-21
ZA818757B (en) 1982-11-24
IL64572A0 (en) 1982-03-31
ES508134A0 (en) 1982-11-01
PT74109A (en) 1982-01-01
GR77634B (en) 1984-09-25
EP0054865A1 (en) 1982-06-30
EP0054865B1 (en) 1986-02-26
DE3173926D1 (en) 1986-04-03
JPS57128676A (en) 1982-08-10
CA1178587A (en) 1984-11-27
DE3048266A1 (en) 1982-07-29
AU547689B2 (en) 1985-10-31
BR8108274A (en) 1982-10-05
ES8300712A1 (en) 1982-11-01
HU189549B (en) 1986-07-28

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