AU6653996A - Solution synthesis of peripheral acting analgesic opioid tetrapeptides - Google Patents

Solution synthesis of peripheral acting analgesic opioid tetrapeptides

Info

Publication number
AU6653996A
AU6653996A AU66539/96A AU6653996A AU6653996A AU 6653996 A AU6653996 A AU 6653996A AU 66539/96 A AU66539/96 A AU 66539/96A AU 6653996 A AU6653996 A AU 6653996A AU 6653996 A AU6653996 A AU 6653996A
Authority
AU
Australia
Prior art keywords
tetrapeptides
solution synthesis
acting analgesic
analgesic opioid
peripheral acting
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU66539/96A
Inventor
Nicholas Rinaldi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shire Canada Inc
Original Assignee
IAF BioChem International Inc
Biochem Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by IAF BioChem International Inc, Biochem Pharma Inc filed Critical IAF BioChem International Inc
Publication of AU6653996A publication Critical patent/AU6653996A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU66539/96A 1995-08-18 1996-08-15 Solution synthesis of peripheral acting analgesic opioid tetrapeptides Abandoned AU6653996A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9516994.2A GB9516994D0 (en) 1995-08-18 1995-08-18 Solution synthesis of peripheral acting analgestic opioid tetrapeptides
GB9516994 1995-08-18
PCT/CA1996/000552 WO1997007129A1 (en) 1995-08-18 1996-08-15 Solution synthesis of peripheral acting analgesic opioid tetrapeptides

Publications (1)

Publication Number Publication Date
AU6653996A true AU6653996A (en) 1997-03-12

Family

ID=10779465

Family Applications (1)

Application Number Title Priority Date Filing Date
AU66539/96A Abandoned AU6653996A (en) 1995-08-18 1996-08-15 Solution synthesis of peripheral acting analgesic opioid tetrapeptides

Country Status (3)

Country Link
AU (1) AU6653996A (en)
GB (1) GB9516994D0 (en)
WO (1) WO1997007129A1 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1030831A4 (en) * 1997-10-10 2003-01-02 Aventis Pharm Prod Inc Process for the preparation of azacycloalkylalkanoyl pseudotetrapeptides
SE9800865D0 (en) * 1998-03-16 1998-03-16 Astra Ab New Process
SE9903291D0 (en) * 1999-09-15 1999-09-15 Astra Ab New process
HRP20211911T1 (en) 2013-03-15 2022-03-18 Protagonist Therapeutics, Inc. Hepcidin analogues and uses therof
SI3143037T1 (en) 2014-05-16 2021-11-30 Protagonist Therapeutics, Inc. Alpha4beta7 integrin thioether peptide antagonists
CA2955460A1 (en) 2014-07-17 2016-01-21 Protagonist Therapeutics, Inc. Oral peptide inhibitors of interleukin-23 receptor and their use to treat inflammatory bowel diseases
CA3009834A1 (en) 2015-12-30 2017-07-06 Protagonist Therapeutics, Inc. Analogues of hepcidin mimetics with improved in vivo half lives
WO2017165676A1 (en) * 2016-03-23 2017-09-28 Protagonist Therapeutics, Inc. METHODS FOR SYNTHESIZING α4β7 PEPTIDE ANTAGONISTS
CA3089868A1 (en) 2018-02-08 2019-08-15 Protagonist Therapeutics, Inc. Conjugated hepcidin mimetics
CN113624898B (en) * 2021-08-23 2023-08-25 成都诺和晟泰生物科技有限公司 Purification method of chiral analgesic polypeptide medicine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2359817A1 (en) * 1976-07-27 1978-02-24 Reckitt & Colmann Prod Ltd Peptide cpds. contg. tyrosine, glycine, phenylalanine and d-amino acid - local anaesthetics, smooth muscle relaxants, adrenergic neutron blockers, beta-stimulants etc.
NL8005121A (en) * 1979-09-20 1981-03-24 Erba Farmitalia ORGANICALLY ACTIVE PEPTIDES.
IS4261A (en) * 1994-02-21 1995-08-22 Astra Aktiebolag New peptide opioids for the treatment of pain and their use

Also Published As

Publication number Publication date
WO1997007129A1 (en) 1997-02-27
GB9516994D0 (en) 1995-10-18

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