AU5990480A - Tripeptidic derivatives - Google Patents

Tripeptidic derivatives

Info

Publication number
AU5990480A
AU5990480A AU59904/80A AU5990480A AU5990480A AU 5990480 A AU5990480 A AU 5990480A AU 59904/80 A AU59904/80 A AU 59904/80A AU 5990480 A AU5990480 A AU 5990480A AU 5990480 A AU5990480 A AU 5990480A
Authority
AU
Australia
Prior art keywords
tripeptidic
derivatives
tripeptidic derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU59904/80A
Other versions
AU547872B2 (en
Inventor
L.G. Svendsen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
DSM Nutritional Products AG
Original Assignee
Pentapharm AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pentapharm AG filed Critical Pentapharm AG
Publication of AU5990480A publication Critical patent/AU5990480A/en
Application granted granted Critical
Publication of AU547872B2 publication Critical patent/AU547872B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0808—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0823—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12Q—MEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
    • C12Q1/00—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions
    • C12Q1/34—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving hydrolase
    • C12Q1/37—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving hydrolase involving peptidase or proteinase

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Analytical Chemistry (AREA)
  • Biotechnology (AREA)
  • Immunology (AREA)
  • Microbiology (AREA)
  • Physics & Mathematics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Engineering & Computer Science (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
AU59904/80A 1979-05-11 1980-05-08 Tripeptidic derivatives Ceased AU547872B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH441279 1979-05-11
CH4412/79 1979-05-11
CH351580 1980-05-06
CH3515/80 1980-05-06

Publications (2)

Publication Number Publication Date
AU5990480A true AU5990480A (en) 1980-12-03
AU547872B2 AU547872B2 (en) 1985-11-07

Family

ID=25693215

Family Applications (1)

Application Number Title Priority Date Filing Date
AU59904/80A Ceased AU547872B2 (en) 1979-05-11 1980-05-08 Tripeptidic derivatives

Country Status (6)

Country Link
EP (1) EP0019589B1 (en)
AU (1) AU547872B2 (en)
CA (1) CA1161431A (en)
DE (1) DE3065506D1 (en)
ES (1) ES491376A0 (en)
WO (1) WO1980002559A1 (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2936543A1 (en) * 1979-09-10 1981-04-09 Behringwerke Ag, 3550 Marburg CHROMOGENIC COMPOUNDS
DK155051C (en) * 1980-05-06 1989-07-03 Pentapharm Ag TRIPEPTIDE DERIVATIVES AND PROCEDURES FOR QUANTITATIVE ANALYSIS OF PROTEOLYTIC ENZYMES UNDER USE thereof
DE3244030A1 (en) * 1982-11-27 1984-05-30 Behringwerke Ag, 3550 Marburg CHROMOGENIC COMPOUNDS, METHOD FOR THEIR PRODUCTION AND THEIR USE
DK201084A (en) * 1983-04-28 1984-10-29 Kimberly Clark Co PROCEDURE FOR DETERMINING CATHEPSIN B IN THE PRESENCE OF OTHER PROTEOLYTIC ENZYMES AND RELATIONSHIPS FOR USING THE PROCEDURE
HU192646B (en) * 1984-12-21 1987-06-29 Gyogyszerkutato Intezet Process for preparing new n-alkyl-peptide aldehydes
US5240913A (en) * 1989-08-18 1993-08-31 Biogen, Inc. Inhibitors of thrombin
FI91777C (en) * 1990-04-02 1994-08-10 Elomit Oy Method for determining plasmin activity
JP3486412B2 (en) * 1993-04-30 2004-01-13 メルク エンド カンパニー インコーポレーテッド Thrombin inhibitor
EP0758341B1 (en) * 1994-04-26 2004-03-24 Aventis Pharmaceuticals, Inc. FACTOR Xa INHIBITORS
US5804560A (en) * 1995-01-06 1998-09-08 Sibia Neurosciences, Inc. Peptide and peptide analog protease inhibitors
US6017887A (en) * 1995-01-06 2000-01-25 Sibia Neurosciences, Inc. Peptide, peptide analog and amino acid analog protease inhibitors
HU224315B1 (en) * 1996-06-05 2005-07-28 Gyógyszerkutató Intézet Kft. Peptidyl-arginin-aldehyde derivatives of anticoagulant activity and pharmaceutical compositions containing them
EP1217000A1 (en) * 2000-12-23 2002-06-26 Aventis Pharma Deutschland GmbH Inhibitors of factor Xa and factor VIIa
CN102464701B (en) * 2010-11-08 2015-10-21 上海医药工业研究院 One class novel cpd, Preparation Method And The Use

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE380257B (en) * 1972-05-02 1975-11-03 Bofors Ab NEW DIAGNOSTIC OPERATING SUBSTRATES WITH HIGH SPECIFICITY FOR THROMBIN AND OTHER PROTEOLYTIC ENZYMES OF THE PEPTIDYL-PEPTIDE HYDROLASES
DE2527932C2 (en) * 1974-07-02 1983-04-21 Pentapharm AG, 4052 Basel Acid addition salts of tripeptide derivatives and their use as substrates for the determination of plasma kallikrein
SE407571B (en) * 1975-07-11 1979-04-02 Kabi Ab NEW CHROMOGENA ENZYME SUBSTRATE FOR SERINE PROTEASES
US4061625A (en) * 1975-07-11 1977-12-06 Ab Kabi Novel chromogenic thrombin substrates
CH634662A5 (en) * 1976-05-28 1983-02-15 Pentapharm Ag USE OF TRIPEPTIDE DERIVATIVES FOR THE QUANTITATIVE DETERMINATION OF PLASMINOGEN ACTIVATORS.
US4147692A (en) * 1977-02-26 1979-04-03 Ajinomoto Co., Inc. Novel dipeptide derivatives, and method of measuring enzymatic activity

Also Published As

Publication number Publication date
AU547872B2 (en) 1985-11-07
DE3065506D1 (en) 1983-12-15
WO1980002559A1 (en) 1980-11-27
CA1161431A (en) 1984-01-31
ES8105865A1 (en) 1981-05-16
EP0019589B1 (en) 1983-11-09
EP0019589A1 (en) 1980-11-26
ES491376A0 (en) 1981-05-16

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