AU567332B2 - 1-(2-carbethoxy 4-benzalkylamido phenoxy) 3-amino 2- propanols - Google Patents

1-(2-carbethoxy 4-benzalkylamido phenoxy) 3-amino 2- propanols

Info

Publication number
AU567332B2
AU567332B2 AU25537/84A AU2553784A AU567332B2 AU 567332 B2 AU567332 B2 AU 567332B2 AU 25537/84 A AU25537/84 A AU 25537/84A AU 2553784 A AU2553784 A AU 2553784A AU 567332 B2 AU567332 B2 AU 567332B2
Authority
AU
Australia
Prior art keywords
branched
atom
formula
lower alkyl
alkyl radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU25537/84A
Other versions
AU2553784A (en
Inventor
Etienne Bouley
Jean Lacrampe
Jean-Marie Teulon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
UPSA SAS
Original Assignee
Carpibem SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8304150A external-priority patent/FR2542737B1/en
Priority claimed from FR8318509A external-priority patent/FR2555169B2/en
Application filed by Carpibem SA filed Critical Carpibem SA
Publication of AU2553784A publication Critical patent/AU2553784A/en
Application granted granted Critical
Publication of AU567332B2 publication Critical patent/AU567332B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
    • C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
    • C07D303/22—Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

1. Claims for the Contracting States : BE CH DE FR GB IT LI LU NL SE Compounds characterized in that they respond to formula : see diagramm : EP0122827,P20,F2 in which : - R and R' may each designate an atom of hydrogen, an atom of halogen, a nitro group or alkyl or alkoxy radicals with C1-C5, branched or not, or a SCH3 or CF3 group ; - R1 represents a lower alkyl radical with 1 to 5 carbon atoms, branched or not ; - R2 represents a lower alkyl radical with 1 to 5 carbon atoms, branched or not ; and - n designates an integer less than 5. 1. Claims for the Contracting State : AT A process for preparing novel compounds responding to formula see diagramm : EP0122827,P21,F2 in which : - R and R' may each designate an atom of hydrogen, an atom of halogen, a nitro group or alkyl or alkoxy radicals with C1-C5, branched or not, or a SCH3 or CF3 group ; - R1 represents a lower alkyl radical with C1 -C5 , branched or not ; - R2 represents a lower alkyl radical with C1 -C5 , branched or not ; and - n designates an integer less than 5, characterized in that said process comprises the step of reacting a base of formula NH2 -R2 where R2 is as defined hereinabove, on a compound of formula (II) without solvent or in a conventional organic solvent such as alcohols, at a temperature of between 20 degrees C and 150 degrees C, see diagramm : EP0122827,P21,F3 R, R', R1 and n being as defined hereinabove.
AU25537/84A 1983-03-14 1984-03-13 1-(2-carbethoxy 4-benzalkylamido phenoxy) 3-amino 2- propanols Ceased AU567332B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR8304150A FR2542737B1 (en) 1983-03-14 1983-03-14 NOVELS (CARBETHOXY-2 BENZALKYLAMIDO-4 PHENOXY) -1 AMINO-3 PROPANOLS-2, THEIR PREPARATIONS AND THEIR THERAPEUTIC USES
FR83-04150 1983-03-14
FR8318509A FR2555169B2 (en) 1983-11-21 1983-11-21 NOVEL (CARBETHOXY-2 BENZALKYLAMIDO-4 PHENOXYL) -1 AMINO-3 PROPANOLS-2, THEIR PREPARATIONS AND THEIR THERAPEUTIC USES
FR83-18509 1983-11-21

Publications (2)

Publication Number Publication Date
AU2553784A AU2553784A (en) 1984-09-20
AU567332B2 true AU567332B2 (en) 1987-11-19

Family

ID=26223333

Family Applications (1)

Application Number Title Priority Date Filing Date
AU25537/84A Ceased AU567332B2 (en) 1983-03-14 1984-03-13 1-(2-carbethoxy 4-benzalkylamido phenoxy) 3-amino 2- propanols

Country Status (12)

Country Link
EP (1) EP0122827B1 (en)
KR (1) KR910002945B1 (en)
AT (1) ATE20879T1 (en)
AU (1) AU567332B2 (en)
CA (1) CA1218378A (en)
DE (1) DE3460323D1 (en)
DK (1) DK117484A (en)
ES (1) ES530503A0 (en)
GR (1) GR81821B (en)
IE (1) IE57094B1 (en)
PH (1) PH19184A (en)
PT (1) PT78238B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0617020A1 (en) * 1992-04-02 1994-09-28 Shudo, Koichi, Prof. Dr. Carboxylic acid derivatives having retinoic acid-like activity
JP3854154B2 (en) * 2000-04-19 2006-12-06 ニューロテック カンパニー リミテッド Compounds, compositions and methods for preventing neurodegeneration resulting from acute and chronic damage to the central nervous system
US6573402B1 (en) 2000-04-20 2003-06-03 Neurotech Co., Ltd. Compounds, compositions and methods for preventing neurodegeneration in acute and chronic injuries in the central nervous system
EP1551793B1 (en) 2002-06-19 2016-01-20 AmKor Pharma, Inc. Tetrafluorobenzyl derivatives and pharmaceutical composition for preventing and treating acute and chronic neurodegenerative diseases in central nervous system containing the same
KR101333753B1 (en) 2006-04-13 2013-11-28 주식회사 아라온테크 Pharmaceutical composition for treating or preventing degenerative and inflammatory diseases
KR100852962B1 (en) 2007-11-12 2008-08-20 주식회사 뉴로테크 Manufacturing method of 2-hydroxy-5-phenylalkylaminobenzoic acid derivatives and their salts
CA2708804C (en) 2007-12-14 2016-01-12 3M Innovative Properties Company Fiber aggregate
EA021092B1 (en) 2007-12-14 2015-04-30 Шлюмбергер Текнолоджи Б.В. Method of treating subterranean wells using changeable additives
MX2010006456A (en) 2007-12-14 2010-09-28 Schlumberger Technology Bv Proppants and uses thereof.
KR101204108B1 (en) * 2009-02-09 2012-11-22 주식회사 지엔티파마 Medicinal use of 5-benzylaminosalicylic acid derivative or its salt

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU1699483A (en) * 1982-07-20 1984-02-23 Menarini A. S.A.S. 1-alkylamine-3 (4(p-alkyloxy-benzamide)phenoxy)-2- propanols

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3852468A (en) * 1967-02-27 1974-12-03 Ici Ltd Alkanolamine derivatives as {62 -adrenergic blocking agents

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU1699483A (en) * 1982-07-20 1984-02-23 Menarini A. S.A.S. 1-alkylamine-3 (4(p-alkyloxy-benzamide)phenoxy)-2- propanols

Also Published As

Publication number Publication date
DE3460323D1 (en) 1986-08-28
EP0122827B1 (en) 1986-07-23
DK117484A (en) 1984-09-15
ES8504681A1 (en) 1985-05-01
IE840528L (en) 1984-09-14
CA1218378A (en) 1987-02-24
AU2553784A (en) 1984-09-20
IE57094B1 (en) 1992-04-22
EP0122827A1 (en) 1984-10-24
PH19184A (en) 1986-01-23
PT78238B (en) 1986-04-24
DK117484D0 (en) 1984-02-28
PT78238A (en) 1984-04-01
KR910002945B1 (en) 1991-05-11
GR81821B (en) 1984-12-12
ATE20879T1 (en) 1986-08-15
KR840009078A (en) 1984-12-24
ES530503A0 (en) 1985-05-01

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