AU5663598A - 2,1,3-benzothia(oxa)diazole derivatives and their use as endothelin-receptor antagonists - Google Patents

2,1,3-benzothia(oxa)diazole derivatives and their use as endothelin-receptor antagonists

Info

Publication number
AU5663598A
AU5663598A AU56635/98A AU5663598A AU5663598A AU 5663598 A AU5663598 A AU 5663598A AU 56635/98 A AU56635/98 A AU 56635/98A AU 5663598 A AU5663598 A AU 5663598A AU 5663598 A AU5663598 A AU 5663598A
Authority
AU
Australia
Prior art keywords
benzothia
endothelin
oxa
receptor antagonists
diazole derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU56635/98A
Inventor
Soheila Anzali
Maria Christadler
Dieter Dorsch
Werner Mederski
Mathias Dr Osswald
Claus-Jochen Schmitges
Claudia Wilm
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Patent GmbH
Original Assignee
Merck Patent GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH
Publication of AU5663598A publication Critical patent/AU5663598A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU56635/98A 1996-12-19 1997-12-15 2,1,3-benzothia(oxa)diazole derivatives and their use as endothelin-receptor antagonists Abandoned AU5663598A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19653037 1996-12-19
DE19653037A DE19653037A1 (en) 1996-12-19 1996-12-19 Endothelin receptor antagonists
PCT/EP1997/007045 WO1998027077A1 (en) 1996-12-19 1997-12-15 2,1,3-benzothia(oxa)diazole derivatives and their use as endothelin-receptor antagonists

Publications (1)

Publication Number Publication Date
AU5663598A true AU5663598A (en) 1998-07-15

Family

ID=7815375

Family Applications (1)

Application Number Title Priority Date Filing Date
AU56635/98A Abandoned AU5663598A (en) 1996-12-19 1997-12-15 2,1,3-benzothia(oxa)diazole derivatives and their use as endothelin-receptor antagonists

Country Status (4)

Country Link
AR (1) AR008718A1 (en)
AU (1) AU5663598A (en)
DE (1) DE19653037A1 (en)
WO (1) WO1998027077A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10155076A1 (en) * 2001-11-09 2003-05-22 Merck Patent Gmbh Use of endothelin receptor antagonists for the treatment of tumor diseases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0714391A1 (en) * 1993-08-19 1996-06-05 Warner-Lambert Company Substituted 2(5h)furanone, 2(5h)thiophenone and 2(5h)pyrrolone derivatives, their preparation and their use as endothelin antagonists
AU4547896A (en) * 1995-02-03 1996-08-21 Banyu Pharmaceutical Co., Ltd. 4-oxo-2-butenoic acid derivatives
DE19509950A1 (en) * 1995-03-18 1996-09-19 Merck Patent Gmbh Endothelin receptor antagonists
DE19607096A1 (en) * 1996-02-24 1997-08-28 Merck Patent Gmbh Endothelin receptor antagonists

Also Published As

Publication number Publication date
WO1998027077A1 (en) 1998-06-25
AR008718A1 (en) 2000-02-09
DE19653037A1 (en) 1998-06-25

Similar Documents

Publication Publication Date Title
AU5840396A (en) N-heteroaryl-pyridinesulfonamide derivatives and their use as endothelin antagonists
AU2077795A (en) N-heterocyclyl sulphonamide derivatives and their use as endothelin antagonists
AU2957997A (en) 1,2,4-oxadiazoles as adhesion-receptor antagonists
AU2952997A (en) Thiocyano-triazolyl derivatives and their use as microbicides
HK1018780A1 (en) 6-Phenylpyridine-2-ylamine derivatives, the composition and use thereof.
AU6514196A (en) Heterocyclic compounds, their preparation and use
AU2766097A (en) Acyl mercapto-triazolyl derivatives and the use thereof as microbicides
AU2896597A (en) Sulphonyl-mercapto-triazolyl derivatives and their use as microbicides
AU3460297A (en) Taxane derivatives and drugs containing the same
AU3839895A (en) Heterocyclic compounds, their preparation and use
AU6636598A (en) Novel 3,4-dialkoxyphenyl derivatives and the use thereof
AU7550398A (en) Heterocyclic compounds, their production and use
AU679887B2 (en) Azole derivatives, their use, production and usage
AU6514296A (en) Heterocyclic compounds, their preparation and use
AU6524996A (en) Piperazine derivatives and their use as 5-HT1A antagonists
AU7659998A (en) N-triazolyl-2-indolecarboxamides and their use as cck-a agonists
AU2894297A (en) 2,4-diaminopyrimidine derivatives
HUP0102400A3 (en) Substituted octalydropyrido[1,2a]pyrazin derivatives and pharmaceutical compositions containing the same
AU3440597A (en) N-phenylimino heterocyclic derivatives and their use as herbicides
AU3693797A (en) 1,3-dimethyl-5-fluoro-pyrazole-4-carboxamide derivatives, their preparation and their use as microbicides
AU2654692A (en) Pyrrolobenzoxazine derivatives as 5-ht agonists and antagonists
EP1469001B8 (en) Corroles, including chiral derivatives and the use thereof
AU3467697A (en) 3'-oximino-2',3'-dideoxynucleosides and derivatives of the same
AU9068398A (en) 3-substituted 3,4,5,7-tetrahydro-pyrrolo3',4':4,5 thieno2,3-dpyrimidine derivatives, their preparation and use as 5ht antagonists
AU4991797A (en) Piperazino derivatives as neurokinin antagonists