AU5567080A - Penicillins - Google Patents

Penicillins

Info

Publication number
AU5567080A
AU5567080A AU55670/80A AU5567080A AU5567080A AU 5567080 A AU5567080 A AU 5567080A AU 55670/80 A AU55670/80 A AU 55670/80A AU 5567080 A AU5567080 A AU 5567080A AU 5567080 A AU5567080 A AU 5567080A
Authority
AU
Australia
Prior art keywords
penicillins
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU55670/80A
Other versions
AU535080B2 (en
Inventor
Frederico Arcamone
Giovanni Farnceschi
Maurizio Foglio
Aurora Sanfilippo
Cosimo Scarafile
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Carlo Erba SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL, Carlo Erba SpA filed Critical Farmitalia Carlo Erba SRL
Publication of AU5567080A publication Critical patent/AU5567080A/en
Application granted granted Critical
Publication of AU535080B2 publication Critical patent/AU535080B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568—Four-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
AU55670/80A 1979-02-24 1980-02-19 Penicillins Ceased AU535080B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB7906634 1979-02-24
GB7906634 1979-02-24
GB7932591 1979-09-20
GB7932591 1979-09-20

Publications (2)

Publication Number Publication Date
AU5567080A true AU5567080A (en) 1980-09-11
AU535080B2 AU535080B2 (en) 1984-03-01

Family

ID=26270697

Family Applications (1)

Application Number Title Priority Date Filing Date
AU55670/80A Ceased AU535080B2 (en) 1979-02-24 1980-02-19 Penicillins

Country Status (24)

Country Link
AT (1) AT368506B (en)
AU (1) AU535080B2 (en)
CA (2) CA1154010A (en)
CH (2) CH654831A5 (en)
CS (1) CS226010B2 (en)
DE (1) DE3006273A1 (en)
DK (1) DK159448C (en)
ES (2) ES8200685A1 (en)
FI (1) FI75163C (en)
FR (1) FR2449690B1 (en)
GB (1) GB2043639B (en)
GR (1) GR73623B (en)
HK (1) HK74487A (en)
HU (1) HU182664B (en)
IE (1) IE49407B1 (en)
IT (1) IT1193922B (en)
LU (1) LU82192A1 (en)
NL (1) NL192265C (en)
NO (1) NO161000C (en)
NZ (1) NZ192949A (en)
PT (1) PT70849A (en)
SE (1) SE449489B (en)
UA (1) UA6041A1 (en)
YU (1) YU42964B (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
DE3121510A1 (en) * 1980-07-04 1982-06-16 Farmitalia Carlo Erba S.p.A., 20159 Milano 6-Alkyl-2-subst. penems and process for their preparation
JPS588084A (en) * 1981-07-08 1983-01-18 Takeda Chem Ind Ltd (6r)-substituted-(5r)-penem-3-carboxylic acid derivative and its preparation
EP0070204B1 (en) * 1981-07-15 1987-11-19 Sumitomo Pharmaceuticals Company, Limited Carboxylic beta-lactam compounds and the preparation thereof
US4508649A (en) * 1981-12-11 1985-04-02 Farmitalia Carlo Erba Process for preparing optically active penems
NO831160L (en) * 1982-04-08 1983-10-10 Erba Farmitalia PREPARATION OF SUBSTITUTED PENEM DERIVATIVES
PH21930A (en) * 1982-11-16 1988-04-08 Ciba Geigy Ag 6-hydroxy-lower alkylpenem compounds,pharmaceutical composition containing same and method of use thereof
DE3372968D1 (en) * 1982-11-16 1987-09-17 Ciba Geigy Ag Heterocyclyl-thio compounds, process for their preparation, pharmaceutical compositions containing them and their use
GB8300295D0 (en) * 1983-01-06 1983-02-09 Erba Farmitalia Penem esters
JPS59152387A (en) * 1983-02-10 1984-08-31 Shionogi & Co Ltd Novel penem compound
GB8321677D0 (en) * 1983-08-11 1983-09-14 Erba Farmitalia Preparation of penems
US4656165A (en) * 1983-09-02 1987-04-07 Ciba-Geigy Corporation Aminomethyl penem compounds
US4711886A (en) * 1984-07-02 1987-12-08 Merck & Co., Inc. β-lactam derivatives as anti-inflammatory and antidegenerative agents
US4761408A (en) * 1984-11-02 1988-08-02 Ciba-Geigy Corporation Crystalline aminomethyl compound
DE3882730D1 (en) * 1987-02-11 1993-09-09 Ciba Geigy Ag BICYCLIC BETA LACTAM CARBON ACIDS.
GB2206578B (en) * 1987-07-07 1991-07-03 Erba Carlo Spa Process for the preparation of penems
US5364768A (en) * 1987-07-07 1994-11-15 Farmitalia Carlo Erba S.R.L. Process for the preparation of penems
IT1286558B1 (en) * 1996-02-27 1998-07-15 Menarini Farma Ind PROCESS FOR THE PREPARATION OF 2-HALOGENOMETHYL-PENEMS AND THEIR USE FOR THE PREPARATION OF ANTIBACTERIAL PENEMS
DE69805975T2 (en) 1997-12-29 2002-12-19 Res Corp Technologies Inc 2-BETA-SUBSTITUTED-6-ALKYLIDENPENICILIC ACID DERIVATIVES AS BETA LACTAMASE INHIBITORS
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
US6720445B2 (en) * 2000-12-21 2004-04-13 Beacon Laboratories, Inc. Acetyloxymethyl esters and methods for using the same
CA2454413A1 (en) 2001-07-24 2003-03-13 Alamx, L.L.C. 7-alkylidene-3-substituted-3-cephem-4-carboxylates as beta-lactamase inhibitors
JP2005525399A (en) 2002-04-04 2005-08-25 アラムクス エルエルシー Inhibitors of serine and metallo-β-lactamases

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU77306A1 (en) * 1977-05-09 1979-01-18
EP0000636A1 (en) * 1977-07-13 1979-02-07 Glaxo Group Limited Penem compounds, processes for their preparation, their use in pharmaceutical compositions and azetidinones used in their preparation
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
US4155912A (en) * 1977-12-14 1979-05-22 Bristol-Myers Company 2-Methylpenem-3-carboxylic acid antibiotics
JPS54117459A (en) * 1978-01-20 1979-09-12 Glaxo Group Ltd Novel lactam compound
EP0003960B1 (en) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-substituted thia-aza-compounds, their preparation and pharmaceutical compositions containing them
JPS5559193A (en) * 1978-09-20 1980-05-02 Glaxo Group Ltd Bblactam compound
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
EP0013067A1 (en) * 1978-12-22 1980-07-09 Beecham Group Plc Bicyclic beta-lactam antibacterial agents, their use in pharmaceutical compositions, processes for their preparation and intermediates for use in such processes

Also Published As

Publication number Publication date
HU182664B (en) 1984-02-28
CH654831A5 (en) 1986-03-14
IE49407B1 (en) 1985-10-02
PT70849A (en) 1980-03-01
HK74487A (en) 1987-10-23
NL192265C (en) 1997-04-03
UA6041A1 (en) 1994-12-29
DK77580A (en) 1980-08-25
GR73623B (en) 1984-03-26
FR2449690A1 (en) 1980-09-19
CS226010B2 (en) 1984-03-19
AU535080B2 (en) 1984-03-01
NZ192949A (en) 1984-03-16
GB2043639B (en) 1983-07-20
CH651570A5 (en) 1985-09-30
ES488886A0 (en) 1981-11-16
SE8001424L (en) 1980-08-25
FI75163C (en) 1988-05-09
DK159448C (en) 1991-03-04
FI800493A (en) 1980-08-25
NL192265B (en) 1996-12-02
CA1154010A (en) 1983-09-20
IT8020021A0 (en) 1980-02-19
ATA91980A (en) 1982-02-15
CA1212665B (en) 1986-10-14
IT8020021A1 (en) 1981-08-19
DK159448B (en) 1990-10-15
GB2043639A (en) 1980-10-08
LU82192A1 (en) 1980-06-06
ES8107224A1 (en) 1981-10-01
FI75163B (en) 1988-01-29
NO161000C (en) 1989-06-21
NO800501L (en) 1980-08-25
SE449489B (en) 1987-05-04
ES495977A0 (en) 1981-10-01
ES8200685A1 (en) 1981-11-16
AT368506B (en) 1982-10-25
DE3006273A1 (en) 1980-09-04
NL8001012A (en) 1980-08-26
FR2449690B1 (en) 1986-06-13
IT1193922B (en) 1988-08-31
NO161000B (en) 1989-03-13
YU42964B (en) 1989-02-28
YU46180A (en) 1983-02-28
IE800338L (en) 1980-08-24

Similar Documents

Publication Publication Date Title
AU2489984A (en) Arylsulphonyls
AU535080B2 (en) Penicillins
AU534807B2 (en) 3-thiovinyl cephalosporins
AU529508B2 (en) 6-n-propyl-8alpha-methoxymethyl or -methylmercaptomethyl -ergolines
AU525431B2 (en) Emulsans
AU537785B2 (en) Cephalosporins
AU527992B2 (en) 9-aminoalkylfluorenes
AU528665B2 (en) Breathalyser
AU538836B2 (en) Cephalosporins
AU540402B2 (en) Cephalosporins
AU531808B2 (en) Tetrahydrobenzothiazolylimidazolidinones
AU520127B2 (en) Penicillins
AU528075B2 (en) Z-aza-ergolines
AU541984B2 (en) Penicillins
AU5553780A (en) Penicillins
AU517488B2 (en) Penicillins
JPS5659781A (en) Penicillins
AU540237B2 (en) Cephalosporins
AU541011B2 (en) Cephalosporins
AU3302184A (en) Woolpack
AU4319879A (en) Boat-carrier
AU531779B2 (en) Penicillins
AU530095B2 (en) Cephalosporin
GB2061268B (en) Penicillins
AU523015B2 (en) N-substituted-6-oxamorphinans