AU546961B2 - 2,3-dihydro-2-oxo-1h-imidazole derivatives - Google Patents
2,3-dihydro-2-oxo-1h-imidazole derivativesInfo
- Publication number
- AU546961B2 AU546961B2 AU83177/82A AU8317782A AU546961B2 AU 546961 B2 AU546961 B2 AU 546961B2 AU 83177/82 A AU83177/82 A AU 83177/82A AU 8317782 A AU8317782 A AU 8317782A AU 546961 B2 AU546961 B2 AU 546961B2
- Authority
- AU
- Australia
- Prior art keywords
- dihydro
- oxo
- imidazole derivatives
- imidazole
- carboxylic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- AICIYIDUYNFPRY-UHFFFAOYSA-N 1,3-dihydro-2H-imidazol-2-one Chemical class O=C1NC=CN1 AICIYIDUYNFPRY-UHFFFAOYSA-N 0.000 title 1
- XJSWLMGZMRUNLP-UHFFFAOYSA-N 2-oxo-1,3-dihydroimidazole-4-carboxylic acid Chemical class OC(=O)C1=CNC(=O)N1 XJSWLMGZMRUNLP-UHFFFAOYSA-N 0.000 abstract 1
- MFAPRXKYGWLTNN-UHFFFAOYSA-N 5-(bromomethyl)-2-oxo-1,3-dihydroimidazole-4-carboxylic acid Chemical class OC(=O)C=1NC(=O)NC=1CBr MFAPRXKYGWLTNN-UHFFFAOYSA-N 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 239000003146 anticoagulant agent Substances 0.000 abstract 1
- 239000002220 antihypertensive agent Substances 0.000 abstract 1
- 229940030600 antihypertensive agent Drugs 0.000 abstract 1
- 229960004676 antithrombotic agent Drugs 0.000 abstract 1
- 239000000496 cardiotonic agent Substances 0.000 abstract 1
- 230000003177 cardiotonic effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Cardiology (AREA)
- Veterinary Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/260,447 US4329470A (en) | 1981-05-04 | 1981-05-04 | 5-(4-Phenyl 1-piperidinyl)methyl-2,3-dihydro-2-oxo-1H-imidazole-4-carboxylic acid derivatives |
| US260447 | 1981-05-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU8317782A AU8317782A (en) | 1982-11-11 |
| AU546961B2 true AU546961B2 (en) | 1985-09-26 |
Family
ID=22989202
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU83177/82A Ceased AU546961B2 (en) | 1981-05-04 | 1982-04-30 | 2,3-dihydro-2-oxo-1h-imidazole derivatives |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4329470A (OSRAM) |
| EP (1) | EP0064706B1 (OSRAM) |
| JP (1) | JPS57185280A (OSRAM) |
| AT (1) | ATE14125T1 (OSRAM) |
| AU (1) | AU546961B2 (OSRAM) |
| CA (1) | CA1167850A (OSRAM) |
| DE (1) | DE3264545D1 (OSRAM) |
| ES (1) | ES511871A0 (OSRAM) |
| IL (1) | IL65664A (OSRAM) |
| ZA (1) | ZA822988B (OSRAM) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5159083A (en) * | 1990-12-28 | 1992-10-27 | Neurogen Corporation | Certain aminomethyl phenylimidazole derivatives; a class of dopamine receptor subtype specific ligands |
| US5850564A (en) * | 1995-05-03 | 1998-12-15 | Btr, Inc, | Scalable multiple level tab oriented interconnect architecture |
| US6093737A (en) * | 1996-12-30 | 2000-07-25 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| AU6013998A (en) * | 1996-12-30 | 1998-07-31 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US6127390A (en) * | 1997-10-02 | 2000-10-03 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2441933A (en) * | 1945-07-30 | 1948-05-18 | Hoffmann La Roche | Substituted imidazolones and process of making them |
| US2441936A (en) * | 1946-03-22 | 1948-05-18 | Hoffmann La Roche | Imidazolones and method of preparation |
| US2514380A (en) * | 1946-12-26 | 1950-07-11 | Hoffmann La Roche | Diamines and method of production |
| US3303199A (en) * | 1963-07-15 | 1967-02-07 | Geigy Chem Corp | Certain imidazolone derivatives and process for making same |
| NZ193935A (en) * | 1979-06-18 | 1985-05-31 | Richardson Merrell Inc | 4-aroyl-imidazol-2-one derivatives;pharmaceutical compositions |
-
1981
- 1981-05-04 US US06/260,447 patent/US4329470A/en not_active Expired - Lifetime
-
1982
- 1982-04-30 ZA ZA822988A patent/ZA822988B/xx unknown
- 1982-04-30 CA CA000402069A patent/CA1167850A/en not_active Expired
- 1982-04-30 JP JP57071660A patent/JPS57185280A/ja active Granted
- 1982-04-30 AU AU83177/82A patent/AU546961B2/en not_active Ceased
- 1982-05-02 IL IL65664A patent/IL65664A/xx not_active IP Right Cessation
- 1982-05-03 DE DE8282103742T patent/DE3264545D1/de not_active Expired
- 1982-05-03 EP EP82103742A patent/EP0064706B1/en not_active Expired
- 1982-05-03 AT AT82103742T patent/ATE14125T1/de not_active IP Right Cessation
- 1982-05-03 ES ES511871A patent/ES511871A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| IL65664A (en) | 1986-01-31 |
| EP0064706A1 (en) | 1982-11-17 |
| ES8308870A1 (es) | 1983-10-01 |
| ATE14125T1 (de) | 1985-07-15 |
| EP0064706B1 (en) | 1985-07-03 |
| JPH0261474B2 (OSRAM) | 1990-12-20 |
| CA1167850A (en) | 1984-05-22 |
| ZA822988B (en) | 1983-03-30 |
| DE3264545D1 (en) | 1985-08-08 |
| IL65664A0 (en) | 1982-08-31 |
| JPS57185280A (en) | 1982-11-15 |
| US4329470A (en) | 1982-05-11 |
| ES511871A0 (es) | 1983-10-01 |
| AU8317782A (en) | 1982-11-11 |
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