AU4234193A - Synthesis of nucleotide monomers - Google Patents

Synthesis of nucleotide monomers

Info

Publication number
AU4234193A
AU4234193A AU42341/93A AU4234193A AU4234193A AU 4234193 A AU4234193 A AU 4234193A AU 42341/93 A AU42341/93 A AU 42341/93A AU 4234193 A AU4234193 A AU 4234193A AU 4234193 A AU4234193 A AU 4234193A
Authority
AU
Australia
Prior art keywords
synthesis
deoxyadenosine
contacting
benzoyl
yield
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU42341/93A
Other languages
English (en)
Inventor
Leonid Beigelman
Jasenka Matulic-Academic
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sirna Therapeutics Inc
Original Assignee
Ribozyme Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/882,479 external-priority patent/US5506349A/en
Application filed by Ribozyme Pharmaceuticals Inc filed Critical Ribozyme Pharmaceuticals Inc
Publication of AU4234193A publication Critical patent/AU4234193A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
AU42341/93A 1992-05-13 1993-05-06 Synthesis of nucleotide monomers Abandoned AU4234193A (en)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US88257292A 1992-05-13 1992-05-13
US882572 1992-05-13
US882479 1992-05-13
US07/882,479 US5506349A (en) 1992-05-13 1992-05-13 Chemical synthesis of 2', 3'-dideoxycytidine
US91064992A 1992-07-08 1992-07-08
US910649 1992-07-08
US91954492A 1992-07-24 1992-07-24
US919544 1992-07-24

Publications (1)

Publication Number Publication Date
AU4234193A true AU4234193A (en) 1993-12-13

Family

ID=27505972

Family Applications (1)

Application Number Title Priority Date Filing Date
AU42341/93A Abandoned AU4234193A (en) 1992-05-13 1993-05-06 Synthesis of nucleotide monomers

Country Status (6)

Country Link
EP (1) EP0640091A4 (fr)
JP (1) JPH07508022A (fr)
AU (1) AU4234193A (fr)
CA (1) CA2135498A1 (fr)
MX (1) MX9302761A (fr)
WO (1) WO1993023413A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW374087B (en) * 1993-05-25 1999-11-11 Univ Yale L-2',3'-dideoxy nucleotide analogs as anti-hepatitis B(HBV) and anti-HIV agents
US5627160A (en) * 1993-05-25 1997-05-06 Yale University L-2',3'-dideoxy nucleoside analogs as anti-hepatitis B (HBV) and anti-HIV agents
EP1910393A2 (fr) * 2005-07-05 2008-04-16 Hetero Drugs Limited Nouveau procede de preparation de didanosine au moyen de nouveaux produits intermediaires
CN105884846B (zh) * 2016-06-01 2018-08-28 中南大学 一种2’-脱氧腺苷的合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US64631A (en) * 1867-05-14 Thomas g
US5099010A (en) * 1983-01-17 1992-03-24 Research Corporation Intermediates in the preparation of 3'-amino-2',3'-dideoxycytidine and the pharmacologically acceptable salts thereof
US5084445A (en) * 1986-05-01 1992-01-28 University Of Georgia Research Foundation, Inc. 3'-azido-2',3'-dideoxy-5-methylcytidine
JPS63275597A (ja) * 1987-05-07 1988-11-14 Ajinomoto Co Inc ジデオキシシチジンの製造方法、その製造中間体、およびその製造方法
US4987224A (en) * 1988-08-02 1991-01-22 University Of Georgia Research Foundation, Inc. Method of preparation of 2',3'-dideoxynucleosides

Also Published As

Publication number Publication date
WO1993023413A1 (fr) 1993-11-25
JPH07508022A (ja) 1995-09-07
EP0640091A1 (fr) 1995-03-01
CA2135498A1 (fr) 1993-11-25
MX9302761A (es) 1994-05-31
EP0640091A4 (fr) 1995-07-26

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