AU2849399A - Monobactam enzyme inhibitors - Google Patents

Monobactam enzyme inhibitors

Info

Publication number
AU2849399A
AU2849399A AU28493/99A AU2849399A AU2849399A AU 2849399 A AU2849399 A AU 2849399A AU 28493/99 A AU28493/99 A AU 28493/99A AU 2849399 A AU2849399 A AU 2849399A AU 2849399 A AU2849399 A AU 2849399A
Authority
AU
Australia
Prior art keywords
monobactam
enzyme inhibitors
inhibitors
enzyme
monobactam enzyme
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
AU28493/99A
Inventor
Ronald George Micetich
Andhe Venkat Narender Reddy
Rajeshwar Singh
Nian Zhou
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synphar Laboratories Inc
Original Assignee
Synphar Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synphar Laboratories Inc filed Critical Synphar Laboratories Inc
Publication of AU2849399A publication Critical patent/AU2849399A/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU28493/99A 1998-03-24 1999-03-23 Monobactam enzyme inhibitors Withdrawn AU2849399A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9806287 1998-03-24
GBGB9806287.0A GB9806287D0 (en) 1998-03-24 1998-03-24 Monobactam enzyme inhibitors
PCT/IB1999/000558 WO1999048911A1 (en) 1998-03-24 1999-03-23 Monobactam enzyme inhibitors

Publications (1)

Publication Number Publication Date
AU2849399A true AU2849399A (en) 1999-10-18

Family

ID=10829163

Family Applications (1)

Application Number Title Priority Date Filing Date
AU28493/99A Withdrawn AU2849399A (en) 1998-03-24 1999-03-23 Monobactam enzyme inhibitors

Country Status (3)

Country Link
AU (1) AU2849399A (en)
GB (1) GB9806287D0 (en)
WO (1) WO1999048911A1 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9907683D0 (en) 1999-04-06 1999-05-26 Synphar Lab Inc Substituted azetidin-2-ones as cysteine protease inhibitors
JP4911864B2 (en) 2000-08-14 2012-04-04 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド Substituted pyrazoles
DE60126286T2 (en) 2000-08-14 2007-11-15 Ortho-Mcneil Pharmaceutical, Inc. SUBSTITUTED PYRAZOLE
EP1309593B1 (en) 2000-08-14 2006-03-15 Ortho-McNeil Pharmaceutical, Inc. Substituted pyrazoles
US7332494B2 (en) 2000-08-14 2008-02-19 Janssen Pharmaceutica, N.V. Method for treating allergies using substituted pyrazoles
RU2290179C2 (en) 2000-09-06 2006-12-27 Орто-Макнейл Фармасьютикал, Инк. Method for treatment of allergy by using substituted pyrazoles
WO2002070519A1 (en) * 2001-03-05 2002-09-12 Axys Pharmaceuticals, Inc. Monobactams as cathepsin k inhibitors
JP5587790B2 (en) 2008-01-09 2014-09-10 アミュラ セラピューティクス リミティド Compound
KR20130087002A (en) 2010-06-04 2013-08-05 알바니 몰레큘라 리써치, 인크. Glycine transporter-1 inhibitors, methods of making them, and uses thereof
WO2012151319A1 (en) * 2011-05-02 2012-11-08 Virobay, Inc. Cathepsin inhibitors for the treatment of bone cancer and bone cancer pain

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996032408A1 (en) * 1995-03-31 1996-10-17 Synphar Laboratories, Inc. Novel 4-substituted-3-peptidyl-azetidin-2-one derivatives useful as cysteine proteinase inhibitor
US5905076A (en) * 1996-04-10 1999-05-18 National Research Council Of Canada 6-substituted amino-4-oxa-1-azabicyclo 3,2,0! heptan-7-one derivatives as cysteine protease inhibitors
US5916887A (en) * 1996-09-23 1999-06-29 National Research Council Of Canada 4-substituted-3-(2-amino-2-cycloalkyl methyl)-acetamido azetidin-2-one derivatives as cysteine proteinase regulators
CA2266639A1 (en) * 1996-09-23 1998-03-26 Rajeshwar Singh 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators
WO1998032766A1 (en) * 1997-01-23 1998-07-30 Synphar Laboratories Inc. SUBSTITUTED AMINO BICYCLIC-β-LACTAM PENAM AND CEPHAM DERIVATIVES AS CYSTEINE PROTEASE INHIBITORS

Also Published As

Publication number Publication date
WO1999048911A1 (en) 1999-09-30
GB9806287D0 (en) 1998-05-20

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Legal Events

Date Code Title Description
MK13 Application withdrawn section 141(2)/reg 8.3(2) - pct appl. non-entering nat. phase, withdrawn by applicant