AU2020394131B2 - Cycloalkyl urea derivative - Google Patents

Cycloalkyl urea derivative

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Publication number
AU2020394131B2
AU2020394131B2 AU2020394131A AU2020394131A AU2020394131B2 AU 2020394131 B2 AU2020394131 B2 AU 2020394131B2 AU 2020394131 A AU2020394131 A AU 2020394131A AU 2020394131 A AU2020394131 A AU 2020394131A AU 2020394131 B2 AU2020394131 B2 AU 2020394131B2
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AU
Australia
Prior art keywords
group
alkyl
halogen atom
alkoxy
carboxamide
Prior art date
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Application number
AU2020394131A
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English (en)
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AU2020394131A1 (en
Inventor
Yuta FUNAKOSHI
Eiji IDEUE
Masafumi KOMIYA
Shoukou LEE
Shunichiro Uesugi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Pharma Co Ltd
Original Assignee
Sumitomo Pharmaceuticals Co Ltd
Sumitomo Pharma Co Ltd
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Publication of AU2020394131A1 publication Critical patent/AU2020394131A1/en
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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JP2026501630A (ja) 2022-12-30 2026-01-16 エクソン、ラブズ、インコーポレイテッド ジヒドロ－キナゾリン、－ベンゾチアジンおよび－ベンズオキサジン誘導体ならびに神経疾患を治療または予防するためのオレキシン受容体作動薬としてのそれらの使用
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