AU2009205477A1 - Beta-lactams for the treatment of glaucoma, ocular hypertension, baldness and hair loss - Google Patents
Beta-lactams for the treatment of glaucoma, ocular hypertension, baldness and hair loss Download PDFInfo
- Publication number
- AU2009205477A1 AU2009205477A1 AU2009205477A AU2009205477A AU2009205477A1 AU 2009205477 A1 AU2009205477 A1 AU 2009205477A1 AU 2009205477 A AU2009205477 A AU 2009205477A AU 2009205477 A AU2009205477 A AU 2009205477A AU 2009205477 A1 AU2009205477 A1 AU 2009205477A1
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- Prior art keywords
- compound
- prodrug
- pharmaceutically acceptable
- acceptable salt
- pct
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2217208P | 2008-01-18 | 2008-01-18 | |
| US61/022,172 | 2008-01-18 | ||
| US12/352,903 | 2009-01-13 | ||
| US12/352,903 US8063033B2 (en) | 2008-01-18 | 2009-01-13 | Therapeutic beta-lactams |
| PCT/US2009/030894 WO2009091764A2 (en) | 2008-01-18 | 2009-01-14 | Therapeutic beta-lactams |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2009205477A1 true AU2009205477A1 (en) | 2009-07-23 |
Family
ID=40876971
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2009205477A Abandoned AU2009205477A1 (en) | 2008-01-18 | 2009-01-14 | Beta-lactams for the treatment of glaucoma, ocular hypertension, baldness and hair loss |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8063033B2 (enExample) |
| EP (1) | EP2321304A2 (enExample) |
| JP (1) | JP2011510009A (enExample) |
| AU (1) | AU2009205477A1 (enExample) |
| BR (1) | BRPI0906846A2 (enExample) |
| CA (1) | CA2712264A1 (enExample) |
| WO (1) | WO2009091764A2 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7772392B2 (en) * | 2005-05-06 | 2010-08-10 | Allergan, Inc. | Therapeutic substituted β-lactams |
| BRPI0611257A2 (pt) * | 2005-05-06 | 2010-08-24 | Allergan Inc | beta-lactamas substituÍdas e uso em medicina do mesmo |
| CA2688897A1 (en) * | 2007-05-23 | 2008-11-23 | Allergan, Inc. | Cyclic lactams for the treatment of glaucoma or elevated intraocular pressure |
| US8440819B2 (en) * | 2008-02-22 | 2013-05-14 | Allergan, Inc. | Therapeutic substituted beta-lactams |
| US8202855B2 (en) * | 2008-03-04 | 2012-06-19 | Allergan, Inc | Substituted beta-lactams |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4166452A (en) * | 1976-05-03 | 1979-09-04 | Generales Constantine D J Jr | Apparatus for testing human responses to stimuli |
| US4256108A (en) * | 1977-04-07 | 1981-03-17 | Alza Corporation | Microporous-semipermeable laminated osmotic system |
| US4265874A (en) * | 1980-04-25 | 1981-05-05 | Alza Corporation | Method of delivering drug with aid of effervescent activity generated in environment of use |
| GB8329559D0 (en) * | 1983-11-04 | 1983-12-07 | Erba Farmitalia | Furyl derivatives of 16-substituted prostaglandins preparations |
| CA2151588C (en) | 1992-12-16 | 2002-03-19 | Michael D. Varney | Antiproliferative substituted 5-thiapyrimidinone and 5-selenopyrimidinone |
| US5462968A (en) * | 1994-01-19 | 1995-10-31 | Allergan, Inc. | EP2 -receptor agonists as agents for lowering intraocular pressure |
| US5698598A (en) * | 1995-08-04 | 1997-12-16 | Allergan | EP2 -receptor agonists as agents for lowering intraocular pressure |
| US6090847A (en) * | 1997-11-21 | 2000-07-18 | Allergan Sales, Inc. | EP2 -receptor agonists as neuroprotective agents for the eye |
| US6437146B1 (en) * | 1998-09-25 | 2002-08-20 | Fujisawa Pharmaceutical Co., Ltd. | Oxazole compounds as prostaglandin e2 agonists or antagonists |
| SI1339678T1 (sl) * | 2000-11-27 | 2007-12-31 | Pfizer Prod Inc | Selektivni agonisti EP4 receptorja pri zdravljenju osteoporoze |
| AU2002328855B2 (en) * | 2001-07-16 | 2005-11-24 | F. Hoffmann-La Roche Ag | Prostaglandin Analogues As EP4 Receptor Agonists |
| CN1617868A (zh) * | 2001-11-05 | 2005-05-18 | 阿勒根公司 | 作为EP2－受体激动剂的ω－环烷基17－杂芳基前列腺素E2 类似物 |
| ATE336247T1 (de) * | 2002-03-18 | 2006-09-15 | Pfizer Prod Inc | Verwendung von selektiven ep4 rezeptor agonisten zur behandlung von krankheiten |
| US7091231B2 (en) * | 2004-12-10 | 2006-08-15 | Allergan, Inc. | 12-Aryl prostaglandin analogs |
| US7772392B2 (en) * | 2005-05-06 | 2010-08-10 | Allergan, Inc. | Therapeutic substituted β-lactams |
| BRPI0611257A2 (pt) * | 2005-05-06 | 2010-08-24 | Allergan Inc | beta-lactamas substituÍdas e uso em medicina do mesmo |
| US7674786B2 (en) * | 2005-05-06 | 2010-03-09 | Allergan, Inc. | Therapeutic β-lactams |
| WO2006121822A1 (en) * | 2005-05-06 | 2006-11-16 | Allergan, Inc. | USE OF β-LACTAMS FOR THE TREATMENTOF IBD AND GLAUCOMA |
| US7427685B2 (en) * | 2005-12-06 | 2008-09-23 | Allergan, Inc. | Therapeutic substituted cyclopentanes |
| US20070254920A1 (en) * | 2006-04-26 | 2007-11-01 | Aerie Pharmaceuticals, Inc. | Prodrug derivatives of acids using alcohols with homotopic hydroxy groups and methods for their preparation and use |
| US8202855B2 (en) * | 2008-03-04 | 2012-06-19 | Allergan, Inc | Substituted beta-lactams |
-
2009
- 2009-01-13 US US12/352,903 patent/US8063033B2/en active Active
- 2009-01-14 BR BRPI0906846-5A patent/BRPI0906846A2/pt not_active IP Right Cessation
- 2009-01-14 EP EP09702401A patent/EP2321304A2/en not_active Withdrawn
- 2009-01-14 JP JP2010543200A patent/JP2011510009A/ja active Pending
- 2009-01-14 CA CA2712264A patent/CA2712264A1/en not_active Abandoned
- 2009-01-14 WO PCT/US2009/030894 patent/WO2009091764A2/en not_active Ceased
- 2009-01-14 AU AU2009205477A patent/AU2009205477A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US8063033B2 (en) | 2011-11-22 |
| JP2011510009A (ja) | 2011-03-31 |
| EP2321304A2 (en) | 2011-05-18 |
| US20090186866A1 (en) | 2009-07-23 |
| WO2009091764A2 (en) | 2009-07-23 |
| WO2009091764A3 (en) | 2010-01-21 |
| CA2712264A1 (en) | 2009-07-23 |
| BRPI0906846A2 (pt) | 2015-07-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |