AU2003291322B2 - Methods for treating gastroesophageal reflux disease - Google Patents
Methods for treating gastroesophageal reflux disease Download PDFInfo
- Publication number
- AU2003291322B2 AU2003291322B2 AU2003291322A AU2003291322A AU2003291322B2 AU 2003291322 B2 AU2003291322 B2 AU 2003291322B2 AU 2003291322 A AU2003291322 A AU 2003291322A AU 2003291322 A AU2003291322 A AU 2003291322A AU 2003291322 B2 AU2003291322 B2 AU 2003291322B2
- Authority
- AU
- Australia
- Prior art keywords
- gastroesophageal reflux
- reflux disease
- glucocorticoid receptor
- receptor antagonist
- antagonist
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- A61P5/46—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids
Landscapes
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| CA (2) | CA2504751C (cg-RX-API-DMAC7.html) |
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| US8569277B2 (en) | 2004-08-11 | 2013-10-29 | Palo Alto Investors | Methods of treating a subject for a condition |
| US8324192B2 (en) | 2005-11-12 | 2012-12-04 | The Regents Of The University Of California | Viscous budesonide for the treatment of inflammatory diseases of the gastrointestinal tract |
| US8679545B2 (en) | 2005-11-12 | 2014-03-25 | The Regents Of The University Of California | Topical corticosteroids for the treatment of inflammatory diseases of the gastrointestinal tract |
| US8497258B2 (en) | 2005-11-12 | 2013-07-30 | The Regents Of The University Of California | Viscous budesonide for the treatment of inflammatory diseases of the gastrointestinal tract |
| WO2007131041A2 (en) * | 2006-05-02 | 2007-11-15 | Corcept Therapeutics, Inc. | The use of a glucocorticoid receptor ii antagonist to treat depression in patients taking il-2 |
| PT2114970E (pt) | 2007-02-02 | 2011-09-22 | Pfizer Prod Inc | Compostos tricíclicos e sua utilização como moduladores de receptor de glucocorticóide |
| WO2009050136A2 (en) * | 2007-10-17 | 2009-04-23 | Laboratoire Hra Pharma | Glucocorticoid receptor antagonists such as mifepristone for treating cushing' s syndrome |
| US20090123551A1 (en) * | 2007-11-13 | 2009-05-14 | Meritage Pharma, Inc. | Gastrointestinal delivery systems |
| HRP20180408T1 (hr) | 2007-11-13 | 2018-04-20 | Meritage Pharma, Inc. | Pripravci za liječenje gastrointestinalnih upala |
| US20100216754A1 (en) * | 2007-11-13 | 2010-08-26 | Meritage Pharma, Inc. | Compositions for the treatment of inflammation of the gastrointestinal tract |
| US20090143343A1 (en) * | 2007-11-13 | 2009-06-04 | Meritage Pharma, Inc. | Compositions for the treatment of inflammation of the gastrointestinal tract |
| US20090264392A1 (en) * | 2008-04-21 | 2009-10-22 | Meritage Pharma, Inc. | Treating eosinophilic esophagitis |
| EP2440210A4 (en) * | 2009-06-12 | 2014-01-29 | Meritage Pharma Inc | METHOD FOR THE TREATMENT OF STOMACH DARM DISEASES |
| US10500216B2 (en) | 2011-11-18 | 2019-12-10 | Corcept Therapeutics, Inc. | Optimizing mifepristone absorption |
| US20150209374A1 (en) | 2014-01-29 | 2015-07-30 | Faro Owiesy | Composition and Method for Curing Migraine Headaches |
| US9943526B2 (en) | 2015-04-21 | 2018-04-17 | Corcept Therapeutics, Inc. | Optimizing mifepristone levels for cushing's patients |
| JP6768789B2 (ja) | 2015-08-13 | 2020-10-14 | コーセプト セラピューティクス， インコーポレイテッド | Ａｃｔｈ依存性クッシング症候群を鑑別診断する方法 |
| AU2017210156B2 (en) | 2016-01-19 | 2021-10-28 | Corcept Therapeutics, Inc. | Differential diagnosis of Ectopic Cushing's Syndrome |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4753932A (en) * | 1985-01-14 | 1988-06-28 | Roussel Uclaf | Novel 10-substituted steroids |
| US4912097A (en) * | 1986-05-06 | 1990-03-27 | Roussel Uclaf | Novel 11 β-alkynylphenyl-10-nor-steroids |
| US5468741A (en) * | 1993-05-28 | 1995-11-21 | The Regents Of The University Of California | Use of low levels of mifepristone to treat leiomyomata |
| US6011025A (en) * | 1995-08-17 | 2000-01-04 | Akzo Nobel, N.V. | 11-(substituted phenyl)-estra-4,9-diene derivatives |
Family Cites Families (9)
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|---|---|---|---|---|
| US5250529A (en) * | 1990-02-08 | 1993-10-05 | Kos Pharmaceuticals, Inc. | Method alleviating migraine headache with mast cell degranulation blocking agents |
| US5521166A (en) * | 1994-12-19 | 1996-05-28 | Ortho Pharmaceitical Corporation | Antiprogestin cyclophasic hormonal regimen |
| US5914129A (en) | 1996-07-23 | 1999-06-22 | Mauskop; Alexander | Analgesic composition for treatment of migraine headaches |
| US5697112A (en) * | 1996-11-08 | 1997-12-16 | Glaxo Wellcome Inc. | Therapy pillow useful for treating gastroesophageal reflux disease (gerd) and other applications |
| US6166013A (en) * | 1998-07-30 | 2000-12-26 | Abbott Laboratories | Glucocortiocoid-selective agents |
| EE05584B1 (et) * | 1999-04-30 | 2012-10-15 | Pfizer Products Inc. | Glkokortikoidretseptori modulaatorid |
| IL139197A0 (en) * | 1999-10-29 | 2001-11-25 | Pfizer Prod Inc | Use of corticotropin releasing factor antagonists and related compositions |
| US6579898B2 (en) | 2001-03-01 | 2003-06-17 | Pfizer Inc. | Compositions having improved bioavailability |
| EP1587574A4 (en) * | 2001-12-21 | 2009-03-18 | Rhode Island Hospital | SELECTIVE 11b-HSD HEMMER AND METHOD OF USE THEREOF |
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2003
- 2003-11-05 EP EP03768706A patent/EP1581234A4/en not_active Withdrawn
- 2003-11-05 EP EP03768714A patent/EP1567167A4/en not_active Ceased
- 2003-11-05 CA CA2504751A patent/CA2504751C/en not_active Expired - Fee Related
- 2003-11-05 JP JP2004550521A patent/JP2006508951A/ja active Pending
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2010
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Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4753932A (en) * | 1985-01-14 | 1988-06-28 | Roussel Uclaf | Novel 10-substituted steroids |
| US4912097A (en) * | 1986-05-06 | 1990-03-27 | Roussel Uclaf | Novel 11 β-alkynylphenyl-10-nor-steroids |
| US5468741A (en) * | 1993-05-28 | 1995-11-21 | The Regents Of The University Of California | Use of low levels of mifepristone to treat leiomyomata |
| US6011025A (en) * | 1995-08-17 | 2000-01-04 | Akzo Nobel, N.V. | 11-(substituted phenyl)-estra-4,9-diene derivatives |
Non-Patent Citations (1)
| Title |
|---|
| Agarwal et al, 1996. Pharmacology and Therapeutics. 70(3):183-213. * |
Also Published As
| Publication number | Publication date |
|---|---|
| US8450379B2 (en) | 2013-05-28 |
| JP2011021044A (ja) | 2011-02-03 |
| WO2004041215A3 (en) | 2004-11-04 |
| WO2004041214A2 (en) | 2004-05-21 |
| CA2504697C (en) | 2012-03-13 |
| US7361646B2 (en) | 2008-04-22 |
| AU2003291314A1 (en) | 2004-06-07 |
| JP2006507311A (ja) | 2006-03-02 |
| EP1567167A2 (en) | 2005-08-31 |
| US20040167110A1 (en) | 2004-08-26 |
| WO2004041214A3 (en) | 2004-11-11 |
| AU2003291322A1 (en) | 2004-06-07 |
| EP1581234A4 (en) | 2007-09-12 |
| US20040132703A1 (en) | 2004-07-08 |
| CA2504751A1 (en) | 2004-05-21 |
| AU2003291314C1 (en) | 2004-06-07 |
| WO2004041215A2 (en) | 2004-05-21 |
| CA2504697A1 (en) | 2004-05-21 |
| JP2006508951A (ja) | 2006-03-16 |
| AU2003291314B2 (en) | 2007-07-26 |
| EP1567167A4 (en) | 2007-09-12 |
| CA2504751C (en) | 2013-02-05 |
| EP1581234A2 (en) | 2005-10-05 |
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| FGA | Letters patent sealed or granted (standard patent) | ||
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |