AU2003218273A1 - Stereoselective process for the synthesis of (d)-2-amino-5-phenylpentanoic or alkyl ester thereof - Google Patents

Stereoselective process for the synthesis of (d)-2-amino-5-phenylpentanoic or alkyl ester thereof

Info

Publication number
AU2003218273A1
AU2003218273A1 AU2003218273A AU2003218273A AU2003218273A1 AU 2003218273 A1 AU2003218273 A1 AU 2003218273A1 AU 2003218273 A AU2003218273 A AU 2003218273A AU 2003218273 A AU2003218273 A AU 2003218273A AU 2003218273 A1 AU2003218273 A1 AU 2003218273A1
Authority
AU
Australia
Prior art keywords
phenylpentanoic
synthesis
amino
alkyl ester
stereoselective process
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003218273A
Inventor
Tonya Lynn Combs
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of AU2003218273A1 publication Critical patent/AU2003218273A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88—Nitrogen atoms, e.g. allantoin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AU2003218273A 2002-04-10 2003-03-28 Stereoselective process for the synthesis of (d)-2-amino-5-phenylpentanoic or alkyl ester thereof Abandoned AU2003218273A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US37165102P 2002-04-10 2002-04-10
US60/371,651 2002-04-10
PCT/US2003/008460 WO2003087036A1 (en) 2002-04-10 2003-03-28 Stereoselective process for the synthesis of (d)-2-amino-5-phenylpentanoic or alkyl ester thereof

Publications (1)

Publication Number Publication Date
AU2003218273A1 true AU2003218273A1 (en) 2003-10-27

Family

ID=29250715

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003218273A Abandoned AU2003218273A1 (en) 2002-04-10 2003-03-28 Stereoselective process for the synthesis of (d)-2-amino-5-phenylpentanoic or alkyl ester thereof

Country Status (2)

Country Link
AU (1) AU2003218273A1 (en)
WO (1) WO2003087036A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR086554A1 (en) 2011-05-27 2014-01-08 Novartis Ag DERIVATIVES OF PIPERIDINE 3-ESPIROCICLICA AS AGRONISTS OF GHRELINE RECEPTORS
EP2852591A1 (en) 2012-05-03 2015-04-01 Novartis AG L-malate salt of 2, 7 - diaza - spiro [4.5]dec- 7 - yle derivatives and crystalline forms thereof as ghrelin receptor agonists

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6329342B1 (en) * 1997-08-19 2001-12-11 Eli Lilly And Company Treatment of congestive heart failure with growth hormone secretagogues

Also Published As

Publication number Publication date
WO2003087036A1 (en) 2003-10-23

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase