AU2003212856A1 - Substituted benzopyrans as selective estrogen receptor-beta agonists - Google Patents

Substituted benzopyrans as selective estrogen receptor-beta agonists

Info

Publication number
AU2003212856A1
AU2003212856A1 AU2003212856A AU2003212856A AU2003212856A1 AU 2003212856 A1 AU2003212856 A1 AU 2003212856A1 AU 2003212856 A AU2003212856 A AU 2003212856A AU 2003212856 A AU2003212856 A AU 2003212856A AU 2003212856 A1 AU2003212856 A1 AU 2003212856A1
Authority
AU
Australia
Prior art keywords
estrogen receptor
selective estrogen
beta agonists
substituted benzopyrans
benzopyrans
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003212856A
Other languages
English (en)
Inventor
Jeffrey Alan Dodge
Venkatesh Gary Krishnan
Charles Willis Lugar Iii
Blake Lee Neubauer
Bryan Hurst Norman
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of AU2003212856A1 publication Critical patent/AU2003212856A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • C07D311/60—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with aryl radicals attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2003212856A 2002-03-01 2003-02-13 Substituted benzopyrans as selective estrogen receptor-beta agonists Abandoned AU2003212856A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US36152402P 2002-03-01 2002-03-01
US60/361,524 2002-03-01
PCT/US2003/002678 WO2003074044A1 (fr) 2002-03-01 2003-02-13 Benzopyranes substitues utilises comme agonistes selectifs des recepteurs des oestrogenes beta

Publications (1)

Publication Number Publication Date
AU2003212856A1 true AU2003212856A1 (en) 2003-09-16

Family

ID=27789125

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003212856A Abandoned AU2003212856A1 (en) 2002-03-01 2003-02-13 Substituted benzopyrans as selective estrogen receptor-beta agonists

Country Status (2)

Country Link
AU (1) AU2003212856A1 (fr)
WO (1) WO2003074044A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9623021B2 (en) 2007-01-22 2017-04-18 Gtx, Inc. Nuclear receptor binding agents
US9604931B2 (en) 2007-01-22 2017-03-28 Gtx, Inc. Nuclear receptor binding agents
EP2647376A1 (fr) 2007-01-22 2013-10-09 Gtx, Inc. Agents de liaison de récepteur nucléaire

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH473114A (de) * 1963-08-28 1969-05-31 Merck Ag E Verfahren zur Herstellung von substituierten Flavanoiden
DE1518038C3 (de) * 1965-10-20 1975-01-23 Merck Patent Gmbh, 6100 Darmstadt 3,6-Di*ubstituierte Flavanderivate und Verfahren zu Ihrer Herstellung, sowie diese enthaltende Arzneimittel
CN1358091A (zh) * 1999-04-16 2002-07-10 阿斯特拉曾尼卡有限公司 雌激素受体－β配体
US7214706B2 (en) * 2000-03-01 2007-05-08 Akzo Nobel N.V. Chroman derivatives as estrogenic compounds

Also Published As

Publication number Publication date
WO2003074044A1 (fr) 2003-09-12

Similar Documents

Publication Publication Date Title
AU2003243637A1 (en) Cannabinoid receptor agonists
AU2003239350A1 (en) 7-hydroxy chromones as potent antioxidants
IL163928A0 (en) Pyridinoylpiperidines as 5-htf agonists
AU2003271157A1 (en) Saw blade
AU2002253675A1 (en) Chromene compound
AU2003261613A1 (en) Automatic optical-fiber cutter
AU2002326312A1 (en) Cannabinoids
AU2003266267A1 (en) Birefringent marking
AU2003298659A1 (en) Soluble isoflavone compositions
AU2003220963A1 (en) Chromene compound
AU2002349677A1 (en) Chromene compound
AU2003248537A1 (en) Bushing
AU2002357184A1 (en) SUBSTITUTED 6H-DIBENZO(c,h)CHROMENES AS ESTROGENIC AGENTS
AU2002951388A0 (en) Bookmark
AUPS328902A0 (en) An incendiary
AU2003248356A1 (en) Beta3-adrenergic receptor agonists
AU2003212856A1 (en) Substituted benzopyrans as selective estrogen receptor-beta agonists
AU2003273786A1 (en) An attachment device for an object, such as a cutting board
SI1448544T1 (sl) Substituirani benzopirani kot selektivni agonistiestrogenskega receptorja beta
AU2003214424A1 (en) Network performance indicators
AU2003256785A1 (en) Improved shears
AU2003286316A1 (en) 5-aminophenanthridine derivatives as npy-5 antagonists
AU2002358595A1 (en) Cutting die
AU2003284704A1 (en) Substituted 1h-pyridine-2-one derivatives
AU2002328757A1 (en) Radar support for speed monitoring

Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase