AU2002363366A1 - Derivatives of phenoxy-N- 4-(isothiazolidin-1,1-dioxid-2YL)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor XA in the treatment of thromboembolic diseases and tumors - Google Patents

Derivatives of phenoxy-N- 4-(isothiazolidin-1,1-dioxid-2YL)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor XA in the treatment of thromboembolic diseases and tumors

Info

Publication number
AU2002363366A1
AU2002363366A1 AU2002363366A AU2002363366A AU2002363366A1 AU 2002363366 A1 AU2002363366 A1 AU 2002363366A1 AU 2002363366 A AU2002363366 A AU 2002363366A AU 2002363366 A AU2002363366 A AU 2002363366A AU 2002363366 A1 AU2002363366 A1 AU 2002363366A1
Authority
AU
Australia
Prior art keywords
isothiazolidin
dioxid
valerian
pheny
phenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU2002363366A
Other versions
AU2002363366B2 (en
Inventor
Christopher Barnes
Bertram Cezanne
Dieter Dorsch
Johannes Gleitz
Werner Mederski
Christos Tsaklakidis
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Patent GmbH
Original Assignee
Merck Patent GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10155075A external-priority patent/DE10155075A1/en
Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH
Publication of AU2002363366A1 publication Critical patent/AU2002363366A1/en
Application granted granted Critical
Publication of AU2002363366B2 publication Critical patent/AU2002363366B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

AU2002363366A 2001-11-09 2002-10-10 Derivatives of phenoxy-N- 4-(isothiazolidin-1,1-dioxid-2YL)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor XA in the treatment of thromboembolic diseases and tumors Ceased AU2002363366B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10155075.8 2001-11-09
DE10155075A DE10155075A1 (en) 2001-11-09 2001-11-09 Cyclic sulfonamides
PCT/EP2002/011349 WO2003039543A1 (en) 2001-11-09 2002-10-10 Derivatives of phenoxy-n-'4-(isothiazolidin-1,1-dioxid-2yl)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor xa in the treatment of thromboembolic diseases and tumors

Publications (2)

Publication Number Publication Date
AU2002363366A1 true AU2002363366A1 (en) 2003-07-24
AU2002363366B2 AU2002363366B2 (en) 2007-11-22

Family

ID=7705183

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002363366A Ceased AU2002363366B2 (en) 2001-11-09 2002-10-10 Derivatives of phenoxy-N- 4-(isothiazolidin-1,1-dioxid-2YL)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor XA in the treatment of thromboembolic diseases and tumors

Country Status (21)

Country Link
US (1) US7199133B2 (en)
EP (1) EP1441726B1 (en)
JP (1) JP4447909B2 (en)
KR (1) KR20050035165A (en)
CN (1) CN1582148A (en)
AR (1) AR037342A1 (en)
AT (1) ATE348611T1 (en)
AU (1) AU2002363366B2 (en)
BR (1) BR0213680A (en)
CA (1) CA2465713A1 (en)
DE (2) DE10155075A1 (en)
DK (1) DK1441726T3 (en)
ES (1) ES2277623T3 (en)
HU (1) HUP0401983A2 (en)
MX (1) MXPA04004307A (en)
MY (1) MY134079A (en)
PL (1) PL369737A1 (en)
PT (1) PT1441726E (en)
RU (1) RU2301228C2 (en)
WO (1) WO2003039543A1 (en)
ZA (1) ZA200404549B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1302462A4 (en) * 2000-07-17 2007-07-18 Takeda Pharmaceutical Sulfone derivatives, process for their production and use thereof
US20040152741A1 (en) * 2002-09-09 2004-08-05 Nps Allelix Corporation Arylglycine derivatives and their use as glycine transport inhibitors
WO2004048363A1 (en) * 2002-11-22 2004-06-10 Takeda Pharmaceutical Company Limited Imidazole derivative, process for producing the same, and use
US7371743B2 (en) 2004-02-28 2008-05-13 Boehringer Ingelheim International Gmbh Carboxylic acid amides, the preparation thereof and their use as medicaments
TWI396686B (en) 2004-05-21 2013-05-21 Takeda Pharmaceutical Cyclic amide derivative, and its production and use
DE102004054847A1 (en) * 2004-11-13 2006-05-24 Sanofi-Aventis Deutschland Gmbh Substituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic agent, and medicament containing them
KR101009594B1 (en) * 2007-05-09 2011-01-20 주식회사 레고켐 바이오사이언스 FXa inhibitors with cyclic amidines as P4 subunit, processes for their preparations, and pharmaceutical compositions and derivatives thereof
BRPI0816837B1 (en) * 2007-09-28 2022-10-18 Portola Pharmaceuticals, Inc PHARMACEUTICAL COMPOSITIONS, ISOLATED TWO-CHAIN POLYPEPTIDE AND USE OF A PHARMACEUTICAL COMPOSITION
KR20150105302A (en) 2012-11-05 2015-09-16 난트 홀딩스 아이피, 엘엘씨 Cyclic sulfonamide containing derivatives as inhibitors of hedgehog signaling pathway

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3901814A1 (en) 1988-07-28 1990-02-01 Bayer Ag SUBSTITUTED AMINOMETHYLZETRALINE AND ITS HETEROCYCLIC ANALOG
US5300523A (en) 1988-07-28 1994-04-05 Bayer Aktiengesellschaft Substituted aminomethyltetralins and their heterocyclic analogues
AU4224993A (en) * 1992-08-19 1994-03-15 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles
US5550139A (en) 1994-01-03 1996-08-27 The Wichita State University Serine protease inhibitors
GB9715895D0 (en) * 1997-07-29 1997-10-01 Zeneca Ltd Heterocyclic compounds
US6489300B1 (en) 1997-07-31 2002-12-03 Eugene D. Thorsett Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
AR016133A1 (en) 1997-07-31 2001-06-20 Wyeth Corp CARBAMILOXI COMPOUND INHIBITING THE ADHESION OF LEUKOCYTES THROUGH VLA-4, COMPOUNDS THAT ARE DRUGS OF THESE COMPOUNDS, PHARMACEUTICAL COMPOSITION, METHOD FOR SETTING VLA-4 TO A BIOLOGICAL SAMPLE, METHOD FOR THE TREATMENT OF A TREATMENT
DE19751949A1 (en) 1997-11-24 1999-05-27 Bayer Ag Neuronal regeneration and neurodegenerative disease treatment with aminomethyl-chroman derivatives
DE19754573A1 (en) * 1997-12-09 1999-06-10 Bayer Ag Pharmaceutical composition for the treatment of stroke and traumatic brain injury
US6114532A (en) 1998-02-03 2000-09-05 Boehringer Ingelheim Pharma Kg Bicyclic heterocycles, the preparation thereof, and their use as pharmaceuticals
DE19804085A1 (en) 1998-02-03 1999-08-05 Boehringer Ingelheim Pharma New benzo-condensed heterocyclic compounds useful in treatment of thrombosis and prevention of vascular occlusion
BR0009083B1 (en) 1999-03-17 2011-11-01 an amide derivative comprising a quinazolinone nucleus, process for the preparation of an amide derivative, pharmaceutical composition, and use of an amide derivative.
US20030065176A1 (en) * 2000-01-29 2003-04-03 Myung-Gyun Kang Factor xa inhibitors with aryl-amidines and derivatives, and prodrugs thereof
KR100423899B1 (en) 2000-05-10 2004-03-24 주식회사 엘지생명과학 Indazoles substituted with 1,1-dioxoisothiazolidine useful as inhibitors of cell proliferation
IL155089A0 (en) * 2000-10-12 2003-10-31 Merck & Co Inc Aza and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
US6488154B1 (en) * 2000-10-16 2002-12-03 Ming-Chuan Yeh Chip tray

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