AU2002334103A1 - Azabicyclic spiroether derivatives as receptor antagonists - Google Patents
Azabicyclic spiroether derivatives as receptor antagonistsInfo
- Publication number
- AU2002334103A1 AU2002334103A1 AU2002334103A AU2002334103A AU2002334103A1 AU 2002334103 A1 AU2002334103 A1 AU 2002334103A1 AU 2002334103 A AU2002334103 A AU 2002334103A AU 2002334103 A AU2002334103 A AU 2002334103A AU 2002334103 A1 AU2002334103 A1 AU 2002334103A1
- Authority
- AU
- Australia
- Prior art keywords
- spiroether
- azabicyclic
- derivatives
- receptor antagonists
- antagonists
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- NJLYCNZOTQCQMC-UHFFFAOYSA-N 2-hexa-2,4-diynyl-1,6-dioxaspiro[4.4]non-3-ene Chemical class C1=CC(CC#CC#CC)OC11OCCC1 NJLYCNZOTQCQMC-UHFFFAOYSA-N 0.000 title 1
- 239000002464 receptor antagonist Substances 0.000 title 1
- 229940044551 receptor antagonist Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/20—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/GB2002/004523 WO2004031191A1 (fr) | 2002-10-04 | 2002-10-04 | Derives de spiroether azabicyclique utilises en tant qu'antagonistes du recepteur nk-1 |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2002334103A1 true AU2002334103A1 (en) | 2004-04-23 |
Family
ID=32050695
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002334103A Abandoned AU2002334103A1 (en) | 2002-10-04 | 2002-10-04 | Azabicyclic spiroether derivatives as receptor antagonists |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP1551846A1 (fr) |
JP (1) | JP2006503859A (fr) |
AU (1) | AU2002334103A1 (fr) |
WO (1) | WO2004031191A1 (fr) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ329807A (en) * | 1997-04-23 | 2000-07-28 | Pfizer | NK-1 receptor antagonists and P receptor antagonists 2-Diarylmethyl-3-amino-1-azabicyclo[2.2.2]octane derivatives and amino substituted N-containing rings as agents for treating irritable bowel syndrome |
US6387925B1 (en) * | 1999-06-01 | 2002-05-14 | Pfizer Inc. | Polymorphs of a crystalline azo-bicyclo (2.2.2) oct-3-yl amine citrate and their pharmaceutical compositions |
US6262067B1 (en) * | 1999-06-22 | 2001-07-17 | Pfizer Inc. | Polymorphs of a crystalline azo-bicyclo 2,2,2 OCT-3-yl amine dihydrochloride and their pharmaceutical compositions |
-
2002
- 2002-10-04 AU AU2002334103A patent/AU2002334103A1/en not_active Abandoned
- 2002-10-04 JP JP2004540910A patent/JP2006503859A/ja not_active Withdrawn
- 2002-10-04 EP EP02807882A patent/EP1551846A1/fr not_active Withdrawn
- 2002-10-04 WO PCT/GB2002/004523 patent/WO2004031191A1/fr not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
JP2006503859A (ja) | 2006-02-02 |
WO2004031191A1 (fr) | 2004-04-15 |
EP1551846A1 (fr) | 2005-07-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AU2003261392A1 (en) | M3muscarinic acetylcholine receptor antagonists | |
AU2003241836A1 (en) | Lpa receptor antagonists | |
AP1828A (en) | Muscarinic Acetycholine receptor antagonists | |
AU2003299807A1 (en) | Heteroarylalkanoic acids as integrin receptor antagonists | |
IL198122A0 (en) | Triazole derivatives as tachykinin receptor antagonists | |
AU2003301851A1 (en) | Azacyclic compounds as orexin receptor antagonist | |
AU2005234596A8 (en) | Piperazinylpiperidine derivatives as chemokine receptor antagonists | |
PL356990A1 (en) | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists | |
AU2003255501A1 (en) | Cxcr4 receptor antagonists | |
AU2003215549A1 (en) | Mercaptoimidazoles as ccr2 receptor antagonists | |
AU2003267088A1 (en) | Chemokine receptor antagonists as therapeutic agents | |
PL1636206T3 (pl) | Pochodne imidazolu jako antagoniści receptorów glutaminianu | |
IL164016A0 (en) | Azetidine derivatives as ccr-3 receptor antagonists | |
AU2002356369A1 (en) | Xanthine derivatives as muscarinic receptor antagonists | |
AU2003205964A1 (en) | Substituted azabicyclo hexane derivatives as muscarinic receptor antagonists | |
AU2002347552A1 (en) | 1-substituted-3-pyrrolidine derivatives as muscarinic receptor antagonists | |
AU2003214520A1 (en) | Substituted azabicyclo hexane derivatives as muscarinic receptor antagonists | |
AU2003300904A1 (en) | Antagonists for human prolactin | |
AU2003240705A1 (en) | Morpholinylmethylureas ccr-3 receptor antagonists | |
AU2003223010A1 (en) | Substituted azabicyclo hexane derivatives as muscarinic receptor antagonists | |
GB0203412D0 (en) | 5-HT 2B receptor antagonists | |
AU2003287219A1 (en) | Il-8 receptor antagonists | |
AU1100300A (en) | Piperidyloxadiazoles as dopamine receptor antagonists | |
AU2003267802A1 (en) | Quaternary ammonium compounds as muscarinic receptor antagonists | |
AU2003297408A1 (en) | Thiazole compounds as integrin receptor antagonists derivatives |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |