AU2002319320A1 - Substituted isoxazoles and the use thereof as antibiotics - Google Patents
Substituted isoxazoles and the use thereof as antibioticsInfo
- Publication number
- AU2002319320A1 AU2002319320A1 AU2002319320A AU2002319320A AU2002319320A1 AU 2002319320 A1 AU2002319320 A1 AU 2002319320A1 AU 2002319320 A AU2002319320 A AU 2002319320A AU 2002319320 A AU2002319320 A AU 2002319320A AU 2002319320 A1 AU2002319320 A1 AU 2002319320A1
- Authority
- AU
- Australia
- Prior art keywords
- antibiotics
- substituted isoxazoles
- isoxazoles
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 229940064005 Antibiotic throat preparations Drugs 0.000 title 1
- 229940083879 Antibiotics FOR TREATMENT OF HEMORRHOIDS AND ANAL FISSURES FOR TOPICAL USE Drugs 0.000 title 1
- 229940042052 Antibiotics for systemic use Drugs 0.000 title 1
- 229940042786 Antitubercular Antibiotics Drugs 0.000 title 1
- 229940093922 Gynecological Antibiotics Drugs 0.000 title 1
- 229940024982 Topical Antifungal Antibiotics Drugs 0.000 title 1
- 239000003242 anti bacterial agent Substances 0.000 title 1
- 230000003115 biocidal Effects 0.000 title 1
- 229940079866 intestinal antibiotics Drugs 0.000 title 1
- 150000002545 isoxazoles Chemical class 0.000 title 1
- 229940005935 ophthalmologic Antibiotics Drugs 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES200101793A ES2180456B1 (en) | 2001-07-20 | 2001-07-20 | SUBSTITUTED ISOXAZOLS AND ITS USE AS ANTIBIOTICS. |
ESP200101793 | 2001-07-20 | ||
PCT/ES2002/000358 WO2003008395A1 (en) | 2001-07-20 | 2002-07-17 | Substituted isoxazoles and the use thereof as antibiotics |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002319320A1 true AU2002319320A1 (en) | 2003-05-22 |
AU2002319320B2 AU2002319320B2 (en) | 2008-03-06 |
Family
ID=8498579
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002319320A Ceased AU2002319320B2 (en) | 2001-07-20 | 2002-07-17 | Substituted isoxazoles and the use thereof as antibiotics |
Country Status (14)
Country | Link |
---|---|
US (1) | US20050014806A1 (en) |
EP (1) | EP1437349B9 (en) |
JP (1) | JP2005502634A (en) |
KR (1) | KR100882377B1 (en) |
CN (1) | CN1556797A (en) |
AT (1) | ATE370129T1 (en) |
AU (1) | AU2002319320B2 (en) |
BR (1) | BR0211588A (en) |
CA (1) | CA2453846A1 (en) |
DE (1) | DE60221870T2 (en) |
DK (1) | DK1437349T3 (en) |
ES (2) | ES2180456B1 (en) |
PT (1) | PT1437349E (en) |
WO (1) | WO2003008395A1 (en) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1443930A1 (en) | 2001-10-25 | 2004-08-11 | AstraZeneca AB | Isoxazoline derivatives useful as antimicrobials |
US7842693B2 (en) | 2002-06-12 | 2010-11-30 | Chemocentryx, Inc. | Substituted piperazines |
US7589199B2 (en) | 2002-06-12 | 2009-09-15 | Chemocentryx, Inc. | Substituted piperazines |
AU2003236500B9 (en) * | 2002-06-12 | 2009-07-02 | Chemocentryx, Inc. | 1-aryl-4-substituted piperazine derivatives for use as CCR1 antagonists for the treatment of inflammation and immune disorders |
US20050256130A1 (en) * | 2002-06-12 | 2005-11-17 | Chemocentryx, Inc. | Substituted piperazines |
MXPA04012959A (en) * | 2002-06-29 | 2005-05-16 | Zentaris Gmbh | Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases. |
WO2005082892A2 (en) * | 2004-02-17 | 2005-09-09 | Dr. Reddy's Laboratories Ltd. | Triazole compounds as antibacterial agents and pharmaceutical compositions containing them |
JP4845873B2 (en) | 2004-03-03 | 2011-12-28 | ケモセントリックス インコーポレーティッド | Bicyclic and bridged nitrogen heterocycles |
US7435831B2 (en) | 2004-03-03 | 2008-10-14 | Chemocentryx, Inc. | Bicyclic and bridged nitrogen heterocycles |
US7696352B2 (en) | 2004-06-18 | 2010-04-13 | Millennium Pharmaceuticals, Inc. | Factor Xa inhibitors |
KR101195801B1 (en) | 2004-06-18 | 2012-11-05 | 밀레니엄 파머슈티컬스 인코퍼레이티드 | Factor xa inhibitors |
CN101405277A (en) * | 2006-01-19 | 2009-04-08 | 萨尔瓦特实验室股份有限公司 | Dicarbonylic compounds with antibacterial activity |
EA015942B1 (en) | 2006-05-05 | 2011-12-30 | Милленниум Фамэсьютикэлс, Инк. | Substituted imidazoles, composition based thereon, a method for preventing or treating undesired thrombosis using thereof and method for inhibiting the coagulation of a blood sample |
CA2651700A1 (en) * | 2006-05-22 | 2007-11-29 | Merck Frosst Canada Ltd. | Cyclic amine derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
CN101220000B (en) * | 2007-12-28 | 2010-12-22 | 天津药物研究院 | Acyl chloride and sulfonyl chloride derivant, and uses thereof |
EP2334636A2 (en) | 2008-09-19 | 2011-06-22 | Pfizer Inc. | Hydroxamic acid derivatives useful as antibacterial agents |
CA2782453C (en) | 2009-12-16 | 2015-11-24 | Matthew Frank Brown | N-linked hydroxamic acid derivatives useful as antibacterial agents |
US8742120B2 (en) | 2009-12-17 | 2014-06-03 | Millennium Pharmaceuticals, Inc. | Methods of preparing factor xa inhibitors and salts thereof |
US8530501B2 (en) | 2009-12-17 | 2013-09-10 | Millennium Pharmaceuticals, Inc. | Salts and crystalline forms of a factor Xa inhibitor |
CN101781294B (en) * | 2010-03-10 | 2012-02-01 | 天津药物研究院 | Imidazole derivative, and preparation method and application thereof |
CN101798303B (en) * | 2010-03-10 | 2011-09-07 | 天津药物研究院 | Azole derivatives, preparation method and application thereof |
MX341977B (en) | 2011-03-07 | 2016-09-07 | Pfizer | Fluoro-pyridinone derivatives useful as antibacterial agents. |
CA2830866A1 (en) | 2011-04-08 | 2012-10-11 | Pfizer Inc. | Imidazole, pyrazole, and triazole derivatives useful as antibacterial agents |
CA2830920C (en) * | 2011-04-08 | 2015-07-14 | Pfizer Inc. | Isoxazole derivatives useful as antibacterial agents |
KR101369584B1 (en) * | 2011-04-19 | 2014-03-06 | 일양약품주식회사 | Phenyl-isoxazol derivatives and preparation process thereof |
US9708276B2 (en) | 2011-10-12 | 2017-07-18 | University of Pittsburgh—of the Commonwealth System of Higher Education | Small molecules targeting androgen receptor nuclear localization and/or level in prostate cancer |
ES2753244T3 (en) | 2013-03-15 | 2020-04-07 | Univ Degli Studi Di Milano Bicocca | Novel Compounds 1,2,4 Oxadiazole Active Against Gram Positive Pathogens |
CN103172584A (en) * | 2013-03-15 | 2013-06-26 | 吉林大学 | Biisoxazole methyl ether derivative and preparation method thereof |
US20160257657A1 (en) | 2013-09-20 | 2016-09-08 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer |
JP6564380B2 (en) | 2013-09-20 | 2019-08-21 | ユニバーシティ オブ ピッツバーグ − オブ ザ コモンウェルス システム オブ ハイヤー エデュケイション | Compounds for treating prostate cancer |
US10518196B2 (en) * | 2014-01-29 | 2019-12-31 | General Electric Company | Devices for separation of particulates, associated methods and systems |
US10980806B2 (en) | 2016-03-24 | 2021-04-20 | University of Pittsburgh—of the Commonwealth System of Higher Education | Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer |
CN109369553B (en) * | 2018-10-22 | 2023-04-11 | 上海凌凯医药科技有限公司 | Method for synthesizing N-3-isoxazole carbamic acid tert-butyl ester |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6069141A (en) * | 1998-02-13 | 2000-05-30 | Pharmacia & Upjohn Company | Substituted aminophenyl isoxazoline derivatives useful as antimicrobials |
TW572757B (en) * | 1998-08-24 | 2004-01-21 | Bristol Myers Squibb Co | Novel isoxazolinone antibacterial agents |
GB9928568D0 (en) * | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
-
2001
- 2001-07-20 ES ES200101793A patent/ES2180456B1/en not_active Withdrawn - After Issue
-
2002
- 2002-07-17 EP EP02748888A patent/EP1437349B9/en not_active Expired - Lifetime
- 2002-07-17 CA CA002453846A patent/CA2453846A1/en not_active Abandoned
- 2002-07-17 BR BR0211588-3A patent/BR0211588A/en not_active IP Right Cessation
- 2002-07-17 PT PT02748888T patent/PT1437349E/en unknown
- 2002-07-17 CN CNA02818517XA patent/CN1556797A/en active Pending
- 2002-07-17 WO PCT/ES2002/000358 patent/WO2003008395A1/en active IP Right Grant
- 2002-07-17 JP JP2003513955A patent/JP2005502634A/en active Pending
- 2002-07-17 US US10/484,027 patent/US20050014806A1/en not_active Abandoned
- 2002-07-17 AT AT02748888T patent/ATE370129T1/en not_active IP Right Cessation
- 2002-07-17 DK DK02748888T patent/DK1437349T3/en active
- 2002-07-17 AU AU2002319320A patent/AU2002319320B2/en not_active Ceased
- 2002-07-17 KR KR1020047001066A patent/KR100882377B1/en not_active IP Right Cessation
- 2002-07-17 DE DE60221870T patent/DE60221870T2/en not_active Expired - Fee Related
- 2002-07-17 ES ES02748888T patent/ES2291481T3/en not_active Expired - Lifetime
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