AU2002314044A1 - Novel use of 2-phenyl-substituted imidazotriazinones - Google Patents
Novel use of 2-phenyl-substituted imidazotriazinonesInfo
- Publication number
- AU2002314044A1 AU2002314044A1 AU2002314044A AU2002314044A AU2002314044A1 AU 2002314044 A1 AU2002314044 A1 AU 2002314044A1 AU 2002314044 A AU2002314044 A AU 2002314044A AU 2002314044 A AU2002314044 A AU 2002314044A AU 2002314044 A1 AU2002314044 A1 AU 2002314044A1
- Authority
- AU
- Australia
- Prior art keywords
- phenyl
- novel use
- substituted imidazotriazinones
- imidazotriazinones
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- -1 2-phenyl-substituted imidazotriazinones Chemical class 0.000 title 1
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10122576.8 | 2001-05-09 | ||
DE10122576 | 2001-05-09 | ||
DE10126198.5 | 2001-05-30 | ||
DE10126198A DE10126198A1 (en) | 2001-05-09 | 2001-05-30 | New use of 2-phenyl-substituted imidazotriazinones |
PCT/EP2002/005002 WO2002089808A1 (en) | 2001-05-09 | 2002-05-07 | Novel use of 2-phenyl-substituted imidazotriazinones |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002314044A1 true AU2002314044A1 (en) | 2003-05-01 |
AU2002314044B2 AU2002314044B2 (en) | 2006-09-21 |
Family
ID=26009261
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002314044A Ceased AU2002314044B2 (en) | 2001-05-09 | 2002-05-07 | Novel use of 2-phenyl-substituted imidazotriazinones |
Country Status (15)
Country | Link |
---|---|
US (1) | US20040152700A1 (en) |
EP (1) | EP1392314B1 (en) |
JP (1) | JP4540295B2 (en) |
CN (1) | CN1633298A (en) |
AT (1) | ATE348618T1 (en) |
AU (1) | AU2002314044B2 (en) |
BR (1) | BR0209541A (en) |
CA (1) | CA2449163C (en) |
DE (1) | DE50209015D1 (en) |
DK (1) | DK1392314T3 (en) |
ES (1) | ES2278927T3 (en) |
IL (1) | IL158738A0 (en) |
MX (1) | MXPA03010119A (en) |
PL (1) | PL363679A1 (en) |
WO (1) | WO2002089808A1 (en) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK1049695T3 (en) * | 1997-11-12 | 2002-05-13 | Bayer Ag | 2-Phenyl-substituted imidazotriazinones as phosphodiesterase inhibitors |
DE10135815A1 (en) * | 2001-07-23 | 2003-02-06 | Bayer Ag | Use of imidazo-triazinone derivative phosphodiesterase 5 inhibitors e.g. for treatment of cardiac insufficiency, psoriasis, diabetes, cancer, glaucoma, bladder disease, Parkinson's disease or pain |
DE10232113A1 (en) * | 2002-07-16 | 2004-01-29 | Bayer Ag | Medicinal products containing vardenafil hydrochloride trihydrate |
JP4838792B2 (en) * | 2004-03-05 | 2011-12-14 | ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング | Novel uses for PDE5 inhibitors |
DE102004023069A1 (en) | 2004-05-11 | 2005-12-08 | Bayer Healthcare Ag | New dosage forms of the PDE 5 inhibitor vardenafil |
DE102004038328A1 (en) * | 2004-08-06 | 2006-03-16 | Bayer Healthcare Ag | New uses of 2-phenyl-substituted imidazotriazinone derivatives |
DE102005001989A1 (en) * | 2005-01-15 | 2006-07-20 | Bayer Healthcare Ag | Intravenous formulations of PDE inhibitors |
DE102005009241A1 (en) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Dosage forms with controlled bioavailability |
DE102005009240A1 (en) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Dosage forms with improved pharmacokinetic properties |
BRPI0616633A2 (en) * | 2005-09-29 | 2011-06-28 | Bayer Healthcare Ag | pde inhibitors and combinations thereof for the treatment of urological disorders |
US8841300B2 (en) | 2006-10-02 | 2014-09-23 | Jerry M. Held | Treatment for Parkinson's disease—combination high dose serotonergic synaptic reuptake inhibitor with phosphodiesterase inhibitor |
AU2008254424B2 (en) | 2007-05-18 | 2012-12-20 | Vivus, Inc. | Novel combinations comprising a phosphodiesterase-5 inhibitor and their use |
CA2689638A1 (en) * | 2007-06-13 | 2008-12-18 | Bayer Schering Pharma Aktiengesellschaft | Pde inhibitors for the treatment of hearing impairment |
CN101965348B (en) * | 2007-09-06 | 2013-11-13 | 上海特化医药科技有限公司 | Process for preparing vardenafil and intermediates thereof |
JP6120985B2 (en) * | 2012-12-04 | 2017-04-26 | アリビオ, インコーポレーテッド | Composition for suppressing apoptosis of nerve cells, comprising a phosphodiesterase type 5 activity inhibitor |
JP2022509815A (en) | 2018-11-28 | 2022-01-24 | トパデュール ファルマ アーゲー | New dual-acting soluble guanylate cyclase activators and phosphodiesterase inhibitors and their uses |
CN113493459B (en) * | 2020-04-07 | 2022-12-13 | 广州白云山医药集团股份有限公司白云山制药总厂 | PDE5 inhibitor compound, preparation method and application thereof |
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US6548490B1 (en) * | 1997-10-28 | 2003-04-15 | Vivus, Inc. | Transmucosal administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
DK1049695T3 (en) * | 1997-11-12 | 2002-05-13 | Bayer Ag | 2-Phenyl-substituted imidazotriazinones as phosphodiesterase inhibitors |
DE19812462A1 (en) * | 1998-03-23 | 1999-09-30 | Bayer Ag | New phosphodiesterase inhibiting 2-phenyl-imidazotriazinone derivatives useful for treating e.g. cardiovascular, cerebrovascular and/or urogenital diseases |
US6221402B1 (en) * | 1997-11-20 | 2001-04-24 | Pfizer Inc. | Rapidly releasing and taste-masking pharmaceutical dosage form |
GT199900061A (en) * | 1998-05-15 | 2000-10-14 | Pfizer | PHARMACEUTICAL FORMULATIONS. |
DE19827640A1 (en) * | 1998-06-20 | 1999-12-23 | Bayer Ag | New imidazotriazine derivatives useful as smooth muscle relaxants for treating e.g. cardiovascular disorders, cerebrovascular disorders, or erectile dysfunction |
JP2002528773A (en) * | 1998-10-27 | 2002-09-03 | コーニンクレッカ フィリップス エレクトロニクス エヌ ヴィ | Driving circuit and device for matrix display panel |
US6075028A (en) * | 1999-09-23 | 2000-06-13 | Graham; Richard | Method of treating Tourette's syndrome and related CNS disorders |
US6503908B1 (en) * | 1999-10-11 | 2003-01-07 | Pfizer Inc | Pharmaceutically active compounds |
GB9923968D0 (en) * | 1999-10-11 | 1999-12-15 | Pfizer Ltd | Therapeutic agents |
IL150022A0 (en) * | 1999-12-24 | 2002-12-01 | Bayer Ag | Imidazo [1,3,5] triazinones and the use thereof |
CN1630532A (en) * | 2000-04-19 | 2005-06-22 | 约翰斯霍普金斯大学 | Methods for prevention and treatment of gastrointestinal disorders |
WO2002009713A2 (en) * | 2000-08-01 | 2002-02-07 | Bayer Aktiengesellschaft | Selective pde 2 inhibitors, used as medicaments for improving cognition |
DE60103299T2 (en) * | 2000-10-30 | 2005-05-12 | Lupin Ltd., Mumbai | FAST-CRUSHING CEFUROXIM AXETIL-CONTAINING MEDICAMENT COMPOSITION WITH DELAYED ACTIVE INGREDIENTS |
WO2002064119A1 (en) * | 2001-02-15 | 2002-08-22 | Tanabe Seiyaku Co., Ltd. | Tablets quickly disintegrated in oral cavity |
DE10118306A1 (en) * | 2001-04-12 | 2002-10-17 | Bayer Ag | Composition for intranasal administration of imidazo-triazinone derivative cGMP PDE inhibitor for treatment of erectile dysfunction, also containing local anesthetic to prevent nasal blockage and improve absorption |
US7939102B2 (en) * | 2002-06-07 | 2011-05-10 | Torrent Pharmaceuticals Ltd. | Controlled release formulation of lamotrigine |
DE10232113A1 (en) * | 2002-07-16 | 2004-01-29 | Bayer Ag | Medicinal products containing vardenafil hydrochloride trihydrate |
DE10325813B4 (en) * | 2003-06-06 | 2007-12-20 | Universitätsklinikum Freiburg | Prophylaxis and / or therapy in portal hypertension |
DE102004023069A1 (en) * | 2004-05-11 | 2005-12-08 | Bayer Healthcare Ag | New dosage forms of the PDE 5 inhibitor vardenafil |
-
2002
- 2002-05-07 EP EP02740570A patent/EP1392314B1/en not_active Expired - Lifetime
- 2002-05-07 BR BR0209541-6A patent/BR0209541A/en not_active IP Right Cessation
- 2002-05-07 CN CNA028139267A patent/CN1633298A/en active Pending
- 2002-05-07 PL PL02363679A patent/PL363679A1/en not_active Application Discontinuation
- 2002-05-07 AT AT02740570T patent/ATE348618T1/en not_active IP Right Cessation
- 2002-05-07 CA CA2449163A patent/CA2449163C/en not_active Expired - Fee Related
- 2002-05-07 MX MXPA03010119A patent/MXPA03010119A/en unknown
- 2002-05-07 AU AU2002314044A patent/AU2002314044B2/en not_active Ceased
- 2002-05-07 WO PCT/EP2002/005002 patent/WO2002089808A1/en active IP Right Grant
- 2002-05-07 DE DE50209015T patent/DE50209015D1/en not_active Expired - Lifetime
- 2002-05-07 US US10/476,939 patent/US20040152700A1/en not_active Abandoned
- 2002-05-07 IL IL15873802A patent/IL158738A0/en unknown
- 2002-05-07 ES ES02740570T patent/ES2278927T3/en not_active Expired - Lifetime
- 2002-05-07 JP JP2002586943A patent/JP4540295B2/en not_active Expired - Fee Related
- 2002-05-07 DK DK02740570T patent/DK1392314T3/en active
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