AU2002216649A1 - Benzoxazole lpaat- beta inhibitors and uses thereof - Google Patents

Benzoxazole lpaat- beta inhibitors and uses thereof

Info

Publication number
AU2002216649A1
AU2002216649A1 AU2002216649A AU1664902A AU2002216649A1 AU 2002216649 A1 AU2002216649 A1 AU 2002216649A1 AU 2002216649 A AU2002216649 A AU 2002216649A AU 1664902 A AU1664902 A AU 1664902A AU 2002216649 A1 AU2002216649 A1 AU 2002216649A1
Authority
AU
Australia
Prior art keywords
lpaat
benzoxazole
beta inhibitors
inhibitors
beta
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002216649A
Inventor
Lynn Bonham
Robert E. Finney
David M. Hollenback
J. Peter Klein
David W Leung
Scott A. Shaffer
Norina M. Tang
Thayer H. White
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of AU2002216649A1 publication Critical patent/AU2002216649A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57—Aryl or substituted aryl radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/18—Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • C07D277/66—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2 with aromatic rings or ring systems directly attached in position 2
AU2002216649A 2000-10-31 2001-10-30 Benzoxazole lpaat- beta inhibitors and uses thereof Abandoned AU2002216649A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24419400P 2000-10-31 2000-10-31
US60/244,194 2000-10-31
PCT/US2001/042836 WO2002036580A2 (en) 2000-10-31 2001-10-30 Benzoxazole lpaat- beta inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
AU2002216649A1 true AU2002216649A1 (en) 2002-05-15

Family

ID=22921741

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002216649A Abandoned AU2002216649A1 (en) 2000-10-31 2001-10-30 Benzoxazole lpaat- beta inhibitors and uses thereof

Country Status (3)

Country Link
US (1) US20020107269A1 (en)
AU (1) AU2002216649A1 (en)
WO (1) WO2002036580A2 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003035602A1 (en) * 2001-10-25 2003-05-01 Sankyo Company, Limited Lipid modulators
EP1460067A4 (en) * 2001-11-26 2005-12-07 Takeda Pharmaceutical Bicyclic derivative, process for producing the same, and use
DE60322869D1 (en) * 2002-04-22 2008-09-25 Univ Johns Hopkins MODULATORS OF HEDGEHOG SIGNALING PATCHES, COMPOSITIONS AND RELATED USES
WO2004067480A2 (en) * 2003-01-25 2004-08-12 Oxford Glycosciences (Uk) Ltd Substituted phenylurea derivatives as hdac inhibitors
US20070185152A1 (en) * 2004-03-02 2007-08-09 Smithkline Beecham Corporation Inhibitors of akt activity
US7772271B2 (en) 2004-07-14 2010-08-10 Ptc Therapeutics, Inc. Methods for treating hepatitis C
US7868037B2 (en) 2004-07-14 2011-01-11 Ptc Therapeutics, Inc. Methods for treating hepatitis C
US7781478B2 (en) 2004-07-14 2010-08-24 Ptc Therapeutics, Inc. Methods for treating hepatitis C
BRPI0511834A (en) 2004-07-14 2008-01-08 Ptc Therapeutics Inc methods for treating hepatitis c
EP1781289A1 (en) 2004-07-22 2007-05-09 PTC Therapeutics, Inc. Thienopyridines for treating hepatitis c
BRPI0516110A (en) * 2004-10-13 2008-08-26 Ptc Therapeutics Inc senseless suppression compounds and methods for their use
US8334290B2 (en) 2005-10-31 2012-12-18 Merck Sharp & Dohme Corp. CETP inhibitors
AU2007351886A1 (en) * 2006-06-23 2008-10-30 Paratek Pharmaceuticals, Inc. Transcription factor modulating compounds and methods of use thereof
WO2014151630A2 (en) 2013-03-15 2014-09-25 Irm Llc Compounds and compositions for the treatment of parasitic diseases
US9186361B2 (en) 2013-03-15 2015-11-17 Novartis Ag Compounds and compositions for the treatment of parasitic diseases
US9296754B2 (en) 2013-03-15 2016-03-29 Novartis Ag Compounds and compositions for the treatment of parasitic diseases
AU2014364565B2 (en) 2013-12-19 2017-06-15 Novartis Ag [1,2,4]triazolo[1,5-a]pyrimidine derivatives as protozoan proteasome inhibitors for the treatment of parasitic diseases such as leishmaniasis
CN116813551A (en) * 2023-08-28 2023-09-29 齐鲁晟华制药有限公司 Preparation method of imidazole phenylurea dipropionate

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR208500A1 (en) * 1972-06-14 1977-02-15 Merck & Co Inc PROCEDURE FOR THE PREPARATION OF OXAZOLE (4,5-B) -PYRIDINES DERIVATIVES
US3974287A (en) * 1975-01-24 1976-08-10 Uniroyal Inc. Control of acarids using certain benzothiazoles or benzothiazolines
US4038396A (en) * 1975-02-24 1977-07-26 Merck & Co., Inc. Anti-inflammatory oxazole[4,5-b]pyridines

Also Published As

Publication number Publication date
WO2002036580A3 (en) 2002-09-06
WO2002036580A2 (en) 2002-05-10
US20020107269A1 (en) 2002-08-08
WO2002036580A9 (en) 2003-02-13

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