AU2002216107A1 - Substituted pyrrolidines as CCR-3 receptor antagonists - Google Patents

Substituted pyrrolidines as CCR-3 receptor antagonists

Info

Publication number
AU2002216107A1
AU2002216107A1 AU2002216107A AU1610702A AU2002216107A1 AU 2002216107 A1 AU2002216107 A1 AU 2002216107A1 AU 2002216107 A AU2002216107 A AU 2002216107A AU 1610702 A AU1610702 A AU 1610702A AU 2002216107 A1 AU2002216107 A1 AU 2002216107A1
Authority
AU
Australia
Prior art keywords
ccr
receptor antagonists
substituted pyrrolidines
pyrrolidines
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002216107A
Inventor
Denis John Kertesz
Michael Garret Roepel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of AU2002216107A1 publication Critical patent/AU2002216107A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2002216107A 2000-12-19 2001-12-13 Substituted pyrrolidines as CCR-3 receptor antagonists Abandoned AU2002216107A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25658500P 2000-12-19 2000-12-19
US60256585 2000-12-19
PCT/EP2001/014670 WO2002050064A1 (en) 2000-12-19 2001-12-13 Substituted pyrrolidines as ccr-3 receptor antagonists

Publications (1)

Publication Number Publication Date
AU2002216107A1 true AU2002216107A1 (en) 2002-07-01

Family

ID=22972794

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002216107A Abandoned AU2002216107A1 (en) 2000-12-19 2001-12-13 Substituted pyrrolidines as CCR-3 receptor antagonists

Country Status (15)

Country Link
US (2) US6552028B2 (en)
EP (1) EP1358181B1 (en)
JP (1) JP2004519443A (en)
KR (1) KR20030061455A (en)
CN (1) CN1239498C (en)
AR (1) AR035519A1 (en)
AT (1) ATE374198T1 (en)
AU (1) AU2002216107A1 (en)
BR (1) BR0116352A (en)
CA (1) CA2431767A1 (en)
DE (1) DE60130684T2 (en)
ES (1) ES2292530T3 (en)
MX (1) MXPA03005581A (en)
WO (1) WO2002050064A1 (en)
ZA (1) ZA200304530B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2004283842A1 (en) * 2003-10-24 2005-05-06 F. Hoffmann-La Roche Ag CCR3 receptor antagonists

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2143143A1 (en) * 1994-03-08 1995-09-09 Toshihiko Tanaka 3-phenylpyrrolidine derivatives
IL125658A0 (en) * 1997-08-18 1999-04-11 Hoffmann La Roche Ccr-3 receptor antagonists
TR200101397T2 (en) * 1998-11-20 2001-11-21 F.Hoffmann-La Roche Ag Piperidine CCR-3 receptor antagonists
AU763960B2 (en) 1998-11-20 2003-08-07 F. Hoffmann-La Roche Ag Pyrrolidine derivatives-CCR-3 receptor antagonists
EP1158980B1 (en) 1998-12-18 2005-08-24 Bristol-Myers Squibb Pharma Company N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
AU2056800A (en) 1998-12-18 2000-07-03 Du Pont Pharmaceuticals Company Heterocyclic piperidines as modulators of chemokine receptor activity
IL142768A0 (en) 1998-12-18 2002-03-10 Du Pont Pharm Co N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
AU2056700A (en) 1998-12-18 2000-07-03 Du Pont Pharmaceuticals Company 2-substituted-4-nitrogen heterocycles as modulators of chemokine receptor activity
EP1140087A4 (en) 1998-12-18 2002-04-03 Du Pont Pharm Co N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
AU2482100A (en) 1998-12-18 2000-07-03 Du Pont Pharmaceuticals Company N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
EP1140086A4 (en) 1998-12-18 2002-04-03 Du Pont Pharm Co N-ureidoalkyl-piperidines as modulators of chemokine receptor activity

Also Published As

Publication number Publication date
KR20030061455A (en) 2003-07-18
US20030199532A1 (en) 2003-10-23
WO2002050064A1 (en) 2002-06-27
AR035519A1 (en) 2004-06-02
CN1481379A (en) 2004-03-10
ZA200304530B (en) 2004-09-10
CN1239498C (en) 2006-02-01
DE60130684T2 (en) 2008-08-14
JP2004519443A (en) 2004-07-02
US20020198255A1 (en) 2002-12-26
EP1358181B1 (en) 2007-09-26
US6552028B2 (en) 2003-04-22
ATE374198T1 (en) 2007-10-15
ES2292530T3 (en) 2008-03-16
CA2431767A1 (en) 2002-06-27
EP1358181A1 (en) 2003-11-05
DE60130684D1 (en) 2007-11-08
BR0116352A (en) 2003-12-02
MXPA03005581A (en) 2003-10-06

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Legal Events

Date Code Title Description
MK4 Application lapsed section 142(2)(d) - no continuation fee paid for the application