AU2001252410A1 - Pyrazole derivatives and their use as gastrin and cholecystokin in receptor ligands - Google Patents
Pyrazole derivatives and their use as gastrin and cholecystokin in receptor ligandsInfo
- Publication number
- AU2001252410A1 AU2001252410A1 AU2001252410A AU5241001A AU2001252410A1 AU 2001252410 A1 AU2001252410 A1 AU 2001252410A1 AU 2001252410 A AU2001252410 A AU 2001252410A AU 5241001 A AU5241001 A AU 5241001A AU 2001252410 A1 AU2001252410 A1 AU 2001252410A1
- Authority
- AU
- Australia
- Prior art keywords
- cholecystokin
- gastrin
- receptor ligands
- pyrazole derivatives
- pyrazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0011095.7A GB0011095D0 (en) | 2000-05-08 | 2000-05-08 | astrin and cholecystokinin receptor ligands (III) |
GB0011095 | 2000-05-08 | ||
PCT/GB2001/001976 WO2001090078A1 (en) | 2000-05-08 | 2001-05-04 | Pyrazole derivatives and their use as gastrin and cholecystokin in receptor ligands |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001252410A1 true AU2001252410A1 (en) | 2001-12-03 |
Family
ID=9891194
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001252410A Abandoned AU2001252410A1 (en) | 2000-05-08 | 2001-05-04 | Pyrazole derivatives and their use as gastrin and cholecystokin in receptor ligands |
Country Status (4)
Country | Link |
---|---|
US (1) | US6956053B2 (en) |
AU (1) | AU2001252410A1 (en) |
GB (2) | GB0011095D0 (en) |
WO (1) | WO2001090078A1 (en) |
Families Citing this family (45)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA79804C2 (en) | 2002-07-03 | 2007-07-25 | Janssen Pharmaceutica Nv | Cck-1 receptor modulators |
CA2515119A1 (en) | 2003-02-07 | 2004-08-19 | Daiichi Pharmaceutical Co., Ltd. | Pyrazole derivative |
US7517900B2 (en) | 2003-10-10 | 2009-04-14 | Bristol-Myers Squibb Company | Pyrazole derivatives as cannabinoid receptor modulators |
US7250434B2 (en) | 2003-12-22 | 2007-07-31 | Janssen Pharmaceutica N.V. | CCK-1 receptor modulators |
EP2088681B1 (en) * | 2004-10-12 | 2018-08-08 | Maxlinear, Inc. | A receiver architecture with digitally generated intermediate frequency |
US7863330B2 (en) | 2006-06-14 | 2011-01-04 | Rottapharm S.P.A. | Deloxiglumide and proton pump inhibitor combination in the treatment of gastrointestinal disorders |
ES2551095T3 (en) | 2007-07-19 | 2015-11-16 | Lundbeck, H., A/S | 5-membered heterocyclic amides and related compounds |
HUP1000243A2 (en) | 2010-05-06 | 2012-01-30 | Avidin Kft | 8-hidroxy-quinoline derivatives |
US8815271B2 (en) | 2010-11-03 | 2014-08-26 | Dow Agrosciences, Llc. | Pesticidal compositions and processes related thereto |
MX355431B (en) | 2011-10-26 | 2018-04-18 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto. |
US9282739B2 (en) | 2012-04-27 | 2016-03-15 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
US9708288B2 (en) | 2012-04-27 | 2017-07-18 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
CN105732580B (en) | 2012-04-27 | 2018-12-07 | 陶氏益农公司 | Pesticidal combination and relative method |
WO2015058026A1 (en) | 2013-10-17 | 2015-04-23 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
JP2016539092A (en) | 2013-10-17 | 2016-12-15 | ダウ アグロサイエンシィズ エルエルシー | Method for producing pest control compound |
CA2925914A1 (en) | 2013-10-17 | 2015-04-23 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
CA2925952A1 (en) | 2013-10-17 | 2015-04-23 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
WO2015058021A1 (en) | 2013-10-17 | 2015-04-23 | Dow Agrosciences Llc | Processes for the preparation of pesticidal compounds |
CN105636443A (en) | 2013-10-17 | 2016-06-01 | 美国陶氏益农公司 | Processes for the preparation of pesticidal compounds |
BR112016008070B8 (en) | 2013-10-17 | 2022-08-23 | Dow Agrosciences Llc | PESTICIDE COMPOUNDS AND THEIR PREPARATION PROCESSES |
CN105848480A (en) | 2013-10-22 | 2016-08-10 | 美国陶氏益农公司 | Synergistic pesticidal compositions and related methods |
RU2016119560A (en) | 2013-10-22 | 2017-11-28 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | SYNERGETIC PESTICIDE COMPOSITIONS AND WAYS RELATED TO THEM |
RU2016119566A (en) | 2013-10-22 | 2017-11-28 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | SYNERGETIC PESTICIDE COMPOSITIONS AND WAYS RELATED TO THEM |
KR20160074637A (en) | 2013-10-22 | 2016-06-28 | 다우 아그로사이언시즈 엘엘씨 | Pesticidal compositions and related methods |
TW201517797A (en) | 2013-10-22 | 2015-05-16 | Dow Agrosciences Llc | Synergistic pesticidal compositions and related methods |
WO2015061151A1 (en) | 2013-10-22 | 2015-04-30 | Dow Agrosciences Llc | Pesticidal compositions and related methods |
CA2926647A1 (en) | 2013-10-22 | 2015-04-30 | Dow Agrosciences Llc | Pesticidal compositions and related methods |
US9788545B2 (en) | 2013-10-22 | 2017-10-17 | Dow Agrosciences Llc | Synergistic pesticidal compositions and related methods |
CA2927198A1 (en) | 2013-10-22 | 2015-04-30 | Dow Agrosciences Llc | Synergistic pesticidal compositions and related methods |
RU2016119531A (en) | 2013-10-22 | 2017-11-28 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | SYNERGIC PESTICIDAL COMPOSITIONS AND RELATED WAYS |
AU2014340422B2 (en) | 2013-10-22 | 2017-06-29 | Corteva Agriscience Llc | Pesticidal compositions and related methods |
JP2016538266A (en) | 2013-10-22 | 2016-12-08 | ダウ アグロサイエンシィズ エルエルシー | Synergistic pest control compositions and related methods |
EP3060054A4 (en) | 2013-10-22 | 2017-04-05 | Dow AgroSciences LLC | Synergistic pesticidal compositions and related methods |
NZ719952A (en) | 2013-10-22 | 2017-05-26 | Dow Agrosciences Llc | Pesticidal compositions and related methods |
WO2015061140A1 (en) | 2013-10-22 | 2015-04-30 | Dow Agrosciences Llc | Synergistic pesticidal compositions and related methods |
JP2016535026A (en) | 2013-10-22 | 2016-11-10 | ダウ アグロサイエンシィズ エルエルシー | Synergistic pest control compositions and related methods |
KR20160074640A (en) | 2013-10-22 | 2016-06-28 | 다우 아그로사이언시즈 엘엘씨 | Pesticidal compositions and related methods |
KR20170038785A (en) | 2014-07-31 | 2017-04-07 | 다우 아그로사이언시즈 엘엘씨 | Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine |
US9249122B1 (en) | 2014-07-31 | 2016-02-02 | Dow Agrosciences Llc | Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine |
JP2017523168A (en) | 2014-07-31 | 2017-08-17 | ダウ アグロサイエンシィズ エルエルシー | Method for producing 3- (3-chloro-1H-pyrazol-1-yl) pyridine |
JP2017525703A (en) | 2014-08-19 | 2017-09-07 | ダウ アグロサイエンシィズ エルエルシー | Method for preparing 3- (3-chloro-1H-pyrazol-1-yl) pyridine |
BR112017004613A2 (en) | 2014-09-12 | 2017-12-05 | Dow Agrosciences Llc | Process for the preparation of 3- (3-chloro-1h-pyrazol-1-yl) pyridine |
JP2020503336A (en) | 2016-12-29 | 2020-01-30 | ダウ アグロサイエンシィズ エルエルシー | Method for preparing pesticidal compounds |
CN110325036B (en) | 2016-12-29 | 2021-10-26 | 美国陶氏益农公司 | Process for preparing pesticidal compounds |
CN114591243B (en) * | 2022-01-11 | 2023-06-20 | 华南农业大学 | Antipyrine hapten, artificial antigen, antibody and preparation methods and application thereof |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2363139A1 (en) * | 1973-12-19 | 1975-07-10 | Bayer Ag | 1-Substd-pyrazol-5-ones - with diuretic, saluretic, antihypertensive and antithrombotic activity |
DK143684A (en) * | 1983-03-12 | 1984-09-13 | Bayer Ag | APPLICATION OF PYRAZOLONE DERIVATIVES AS LIPOXYGENASE INHIBITORS IN THE THERAPY OF ISAER ISCHAEMI AND HEART RHYTHM |
JPH0675749B2 (en) * | 1989-05-11 | 1994-09-28 | 吉田工業株式会社 | Horizontal continuous casting equipment |
US5300514A (en) * | 1990-07-17 | 1994-04-05 | Eli Lilly And Company | Pyrazolidinone CCK and gastrin antagonists and pharmaceutical formulations thereof |
IL98785A (en) | 1990-07-17 | 1995-11-27 | Lilly Co Eli | Pyrazolidinone and pyrazoline-3-ether derivatives as cck and gastrin antagonists and pharmaceutical formulations thereof |
US5399565A (en) * | 1990-07-17 | 1995-03-21 | Eli Lilly And Company | Pyrazolidinone CCK and gastrin antagonists and pharmaceutical formulations therof |
US5202344A (en) * | 1990-12-11 | 1993-04-13 | G. D. Searle & Co. | N-substituted lactams useful as cholecystokinin antagonists |
FR2773153A1 (en) * | 1997-12-29 | 1999-07-02 | Rhone Poulenc Agrochimie | NEW FUNGICIDE COMPOUNDS |
CA2346108A1 (en) * | 1998-11-09 | 2000-05-18 | James Black Foundation Limited | Gastrin and cholecystokinin receptor ligands |
-
2000
- 2000-05-08 GB GBGB0011095.7A patent/GB0011095D0/en not_active Ceased
-
2001
- 2001-05-04 US US10/275,614 patent/US6956053B2/en not_active Expired - Fee Related
- 2001-05-04 WO PCT/GB2001/001976 patent/WO2001090078A1/en active Application Filing
- 2001-05-04 GB GB0225710A patent/GB2378443B/en not_active Expired - Fee Related
- 2001-05-04 AU AU2001252410A patent/AU2001252410A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
GB2378443A (en) | 2003-02-12 |
GB2378443B (en) | 2004-08-04 |
GB0011095D0 (en) | 2000-06-28 |
WO2001090078A1 (en) | 2001-11-29 |
US20030207874A1 (en) | 2003-11-06 |
US6956053B2 (en) | 2005-10-18 |
GB0225710D0 (en) | 2002-12-11 |
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