AU2000246281A1 - Piperidine compounds and process for providing such - Google Patents
Piperidine compounds and process for providing suchInfo
- Publication number
- AU2000246281A1 AU2000246281A1 AU2000246281A AU4628100A AU2000246281A1 AU 2000246281 A1 AU2000246281 A1 AU 2000246281A1 AU 2000246281 A AU2000246281 A AU 2000246281A AU 4628100 A AU4628100 A AU 4628100A AU 2000246281 A1 AU2000246281 A1 AU 2000246281A1
- Authority
- AU
- Australia
- Prior art keywords
- providing
- piperidine compounds
- paroxetine
- piperidine
- synthesis
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Abstract
The tosylate ester of the formula (6) and its salts, are convenient intermediates in the synthesis of paroxetine.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/NL2000/000321 WO2001085689A1 (en) | 2000-05-12 | 2000-05-12 | Piperidine compounds and process for providing such |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2000246281A1 true AU2000246281A1 (en) | 2001-11-20 |
Family
ID=19760689
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2000246281A Abandoned AU2000246281A1 (en) | 2000-05-12 | 2000-05-12 | Piperidine compounds and process for providing such |
Country Status (11)
Country | Link |
---|---|
US (1) | US20020099219A1 (en) |
EP (1) | EP1286965B1 (en) |
AT (1) | ATE257823T1 (en) |
AU (1) | AU2000246281A1 (en) |
DE (1) | DE60007782T2 (en) |
DK (1) | DK1286965T3 (en) |
ES (1) | ES2209876T3 (en) |
NL (1) | NL1016013C1 (en) |
PT (1) | PT1286965E (en) |
SI (1) | SI1286965T1 (en) |
WO (1) | WO2001085689A1 (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1280775A1 (en) * | 2000-05-12 | 2003-02-05 | Synthon B.V. | TOSYLATE SALTS OF 4-(p-FLUOROPHENYL)-PIPERIDINE-3-CARBINOLS |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0190496A3 (en) * | 1984-12-13 | 1987-05-27 | Beecham Group Plc | Piperidine derivatives having a gastro-intestinal activity |
EP0812827B1 (en) * | 1996-06-13 | 2009-09-02 | Sumitomo Chemical Company, Limited | Piperidine derivative as intermediates for the preparation of paroxetine and process for their preparation |
HU221921B1 (en) * | 1996-07-08 | 2003-02-28 | Richter Gedeon Vegyészeti Gyár Rt. | N-benzyl-piperidine or tetrahydro-pyridine derivatives and processes for producing them |
DK0994872T3 (en) * | 1997-06-10 | 2001-05-28 | Synthon Bv | 4-phenylpiperidine compounds |
JP2000095780A (en) * | 1998-09-22 | 2000-04-04 | Asahi Glass Co Ltd | Production of crystal of carbamate compound |
-
2000
- 2000-05-12 DE DE60007782T patent/DE60007782T2/en not_active Revoked
- 2000-05-12 AU AU2000246281A patent/AU2000246281A1/en not_active Abandoned
- 2000-05-12 ES ES00927979T patent/ES2209876T3/en not_active Expired - Lifetime
- 2000-05-12 DK DK00927979T patent/DK1286965T3/en active
- 2000-05-12 AT AT00927979T patent/ATE257823T1/en not_active IP Right Cessation
- 2000-05-12 WO PCT/NL2000/000321 patent/WO2001085689A1/en not_active Application Discontinuation
- 2000-05-12 SI SI200030312T patent/SI1286965T1/en unknown
- 2000-05-12 PT PT00927979T patent/PT1286965E/en unknown
- 2000-05-12 EP EP00927979A patent/EP1286965B1/en not_active Revoked
- 2000-08-24 NL NL1016013A patent/NL1016013C1/en not_active IP Right Cessation
-
2001
- 2001-05-14 US US09/853,860 patent/US20020099219A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
PT1286965E (en) | 2004-04-30 |
SI1286965T1 (en) | 2004-04-30 |
WO2001085689A1 (en) | 2001-11-15 |
EP1286965B1 (en) | 2004-01-14 |
NL1016013C1 (en) | 2001-01-30 |
DE60007782T2 (en) | 2004-12-09 |
US20020099219A1 (en) | 2002-07-25 |
EP1286965A1 (en) | 2003-03-05 |
DE60007782D1 (en) | 2004-02-19 |
DK1286965T3 (en) | 2004-05-03 |
ATE257823T1 (en) | 2004-01-15 |
ES2209876T3 (en) | 2004-07-01 |
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