AU1858992A - 2-(1-piperidyl)ethanol derivatives, their preparation and their therapeutic application - Google Patents

2-(1-piperidyl)ethanol derivatives, their preparation and their therapeutic application

Info

Publication number
AU1858992A
AU1858992A AU18589/92A AU1858992A AU1858992A AU 1858992 A AU1858992 A AU 1858992A AU 18589/92 A AU18589/92 A AU 18589/92A AU 1858992 A AU1858992 A AU 1858992A AU 1858992 A AU1858992 A AU 1858992A
Authority
AU
Australia
Prior art keywords
piperidyl
preparation
therapeutic application
ethanol derivatives
ethanol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU18589/92A
Other versions
AU644296B2 (en
Inventor
Jonathan Frost
Patrick Lardenois
Maria-Carmen Renones
Corinne Rousselle
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9107936A external-priority patent/FR2678270B1/en
Priority claimed from FR9107934A external-priority patent/FR2678265B1/en
Priority claimed from FR9204507A external-priority patent/FR2689891B3/en
Application filed by Synthelabo SA filed Critical Synthelabo SA
Publication of AU1858992A publication Critical patent/AU1858992A/en
Application granted granted Critical
Publication of AU644296B2 publication Critical patent/AU644296B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
AU18589/92A 1991-06-27 1992-06-26 2-(1-piperidyl)ethanol derivatives, their preparation and their therapeutic application Ceased AU644296B2 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
FR9107936A FR2678270B1 (en) 1991-06-27 1991-06-27 DERIVATIVES OF 2- (PIPERIDIN-1-YL) ETHANOL, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9107934A FR2678265B1 (en) 1991-06-27 1991-06-27 DERIVATIVES OF 4- (2-PHENYLETHYL) PIPERIDINE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9107936 1992-04-13
FR9204507A FR2689891B3 (en) 1992-04-13 1992-04-13 DERIVATIVES OF 2- (PIPERIDIN-1-YL) ETHANOL, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR9204507 1992-04-13
FR9107934 1992-04-13

Publications (2)

Publication Number Publication Date
AU1858992A true AU1858992A (en) 1993-01-07
AU644296B2 AU644296B2 (en) 1993-12-02

Family

ID=27252473

Family Applications (1)

Application Number Title Priority Date Filing Date
AU18589/92A Ceased AU644296B2 (en) 1991-06-27 1992-06-26 2-(1-piperidyl)ethanol derivatives, their preparation and their therapeutic application

Country Status (14)

Country Link
EP (1) EP0524846A1 (en)
JP (1) JPH05186460A (en)
KR (1) KR930000505A (en)
CN (1) CN1069491A (en)
AU (1) AU644296B2 (en)
CA (1) CA2072520A1 (en)
CZ (1) CZ199992A3 (en)
FI (1) FI922979A (en)
HU (1) HUT61743A (en)
IE (1) IE922090A1 (en)
IL (1) IL102334A0 (en)
MX (1) MX9203452A (en)
NO (1) NO922521L (en)
NZ (1) NZ243337A (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994001403A1 (en) * 1992-07-08 1994-01-20 Shell Internationale Research Maatschappij B.V. Piperidine derivatives
CZ280669B6 (en) * 1992-10-30 1996-03-13 Pfizer Inc. Derivatives of 3,4-dihydro-2(1h)-quinolone and pharmaceutical composition based thereon
FR2727864B1 (en) * 1994-12-12 1997-04-04 Synthelabo USE OF LIGANDS FROM THE PERIPHERAL BINDING SITES FOR BENZODIAZEPINES FOR THE PREPARATION OF DRUGS USEFUL IN THE TREATMENT OF PERIPHERAL NEUROPATHIES
ZA9610738B (en) 1995-12-22 1997-06-24 Warner Lambert Co Subtype selective nmda receptor ligands and the use thereof
ZA9610736B (en) 1995-12-22 1997-06-27 Warner Lambert Co 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists
ZA9610741B (en) 1995-12-22 1997-06-24 Warner Lambert Co 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610745B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists
WO1999058117A1 (en) * 1998-05-13 1999-11-18 Sanofi-Synthelabo Use of compounds for reducing apoptosis
FR2778564B1 (en) * 1998-05-13 2001-07-13 Sanofi Sa USE OF COMPOUNDS REDUCING APOPTOSIS
ATE333281T1 (en) 1998-12-18 2006-08-15 Scios Inc AGONISTS AND ANTAGONISTS OF BENZODIAZEPINE RECEPTORS OF THE PERIPHERAL TYPE
JPWO2005097782A1 (en) * 2004-04-07 2007-08-16 協和醗酵工業株式会社 Piperidine derivatives
CN103896835A (en) * 2014-04-20 2014-07-02 武汉珈瑜科技有限公司 Quinolinone derivatives and application thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1030415A (en) * 1987-02-20 1989-01-18 山之内制药株式会社 Saturated heterocycle carboxamide derivatives and its preparation method
FR2640266B2 (en) * 1988-07-12 1992-07-10 Synthelabo INDOLONES-2, QUINOLEINONES-2, BENZO (B) AZEPINONES-2 AND BENZIMIDAZOLONES-2 DERIVATIVES OF (HYDROXY-1 PIPERIDINYL-2 ALKYL), THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
JP2969359B2 (en) * 1989-01-13 1999-11-02 武田薬品工業株式会社 Cyclic amine compounds
FR2644786B1 (en) * 1989-03-21 1993-12-31 Adir Cie NOVEL 4-FLUORO-4 BENZOIC DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
JPH03130263A (en) * 1989-07-19 1991-06-04 Eisai Co Ltd Optically active naphthylethanol derivative
FR2668149B1 (en) * 1990-10-18 1994-09-23 Synthelabo 1- (3,4-DIHYDRO-2-OXO-1H-QUINOLEIN-6-YL) -2- [4- (2-PHENYL-ETHYL) PIPERIDIN-1-YL] ETHANOL, ITS PREPARATION AND THERAPEUTIC APPLICATION .

Also Published As

Publication number Publication date
NO922521D0 (en) 1992-06-26
HUT61743A (en) 1993-03-01
FI922979A0 (en) 1992-06-26
IL102334A0 (en) 1993-01-14
CN1069491A (en) 1993-03-03
KR930000505A (en) 1993-01-15
NO922521L (en) 1992-12-28
EP0524846A1 (en) 1993-01-27
AU644296B2 (en) 1993-12-02
CA2072520A1 (en) 1992-12-28
NZ243337A (en) 1994-03-25
FI922979A (en) 1992-12-28
CZ199992A3 (en) 1993-01-13
HU9202138D0 (en) 1992-10-28
IE922090A1 (en) 1992-12-30
MX9203452A (en) 1994-01-31
JPH05186460A (en) 1993-07-27

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