ATE971T1 - HYDROCORTISON-ORTHOESTER, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND PROCESSES FOR THEIR MANUFACTURE. - Google Patents

HYDROCORTISON-ORTHOESTER, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND PROCESSES FOR THEIR MANUFACTURE.

Info

Publication number
ATE971T1
ATE971T1 AT79103870T AT79103870T ATE971T1 AT E971 T1 ATE971 T1 AT E971T1 AT 79103870 T AT79103870 T AT 79103870T AT 79103870 T AT79103870 T AT 79103870T AT E971 T1 ATE971 T1 AT E971T1
Authority
AT
Austria
Prior art keywords
hydrocortison
orthoester
manufacture
processes
pharmaceutical preparations
Prior art date
Application number
AT79103870T
Other languages
German (de)
Inventor
Manfred Dr. Chem. Baumgarth
Dieter Dr. Chem. Orth
Juergen Dr. Harting
Hans Prof. Dr. Chem. Schaefer
Achim Prof. Dr. Zesch
Original Assignee
Merck Patent Gesellschaft Mit Beschraenkter Haftung
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gesellschaft Mit Beschraenkter Haftung filed Critical Merck Patent Gesellschaft Mit Beschraenkter Haftung
Application granted granted Critical
Publication of ATE971T1 publication Critical patent/ATE971T1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

Hydrocortisone orthoesters of the formula <IMAGE> wherein R1 and R2 are independently each H or CH3 and n is 1 or 2 possess antiphlogistic activity.
AT79103870T 1978-11-09 1979-10-09 HYDROCORTISON-ORTHOESTER, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND PROCESSES FOR THEIR MANUFACTURE. ATE971T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19782848584 DE2848584A1 (en) 1978-11-09 1978-11-09 HYDROCORTISON ORTHOESTER, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF
EP79103870A EP0011134B1 (en) 1978-11-09 1979-10-09 Hydrocortisone-ortho ester, pharmaceutical compositions containing them and process for their preparation

Publications (1)

Publication Number Publication Date
ATE971T1 true ATE971T1 (en) 1982-05-15

Family

ID=6054216

Family Applications (1)

Application Number Title Priority Date Filing Date
AT79103870T ATE971T1 (en) 1978-11-09 1979-10-09 HYDROCORTISON-ORTHOESTER, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND PROCESSES FOR THEIR MANUFACTURE.

Country Status (11)

Country Link
US (1) US4264584A (en)
EP (1) EP0011134B1 (en)
JP (1) JPS5569600A (en)
AT (1) ATE971T1 (en)
AU (1) AU527561B2 (en)
CA (1) CA1146532A (en)
DE (2) DE2848584A1 (en)
ES (1) ES485785A1 (en)
HU (1) HU180875B (en)
IL (1) IL58641A (en)
ZA (1) ZA796007B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3516298A1 (en) * 1985-05-07 1986-11-13 Sartorius Gmbh METHOD FOR CONTROLLING A LIQUID CRYSTAL DISPLAY WITH FUNCTION ERROR DETECTABILITY

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3147249A (en) * 1961-06-13 1964-09-01 Vismara Francesco Spa 17alpha, 21-substituted methylenedioxy steroids and methods therefor
US3798217A (en) * 1970-05-14 1974-03-19 Syntex Corp Novel c-16,17 spiro-orthoester steroids and preparation
US3716529A (en) * 1970-05-14 1973-02-13 Syntex Corp Novel c-16,17 spiro-orthoester steroids and preparation

Also Published As

Publication number Publication date
ZA796007B (en) 1980-11-26
EP0011134B1 (en) 1982-05-05
AU5261479A (en) 1980-05-15
EP0011134A1 (en) 1980-05-28
IL58641A (en) 1983-07-31
US4264584A (en) 1981-04-28
DE2848584A1 (en) 1980-05-22
DE2962723D1 (en) 1982-06-24
JPS5569600A (en) 1980-05-26
AU527561B2 (en) 1983-03-10
HU180875B (en) 1983-04-29
CA1146532A (en) 1983-05-17
IL58641A0 (en) 1980-02-29
ES485785A1 (en) 1980-05-16

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