ATE484491T1 - NEW METHOD FOR THE SYNTHESIS OF ENAMIDE DERIVATIVES - Google Patents
NEW METHOD FOR THE SYNTHESIS OF ENAMIDE DERIVATIVESInfo
- Publication number
- ATE484491T1 ATE484491T1 AT04806523T AT04806523T ATE484491T1 AT E484491 T1 ATE484491 T1 AT E484491T1 AT 04806523 T AT04806523 T AT 04806523T AT 04806523 T AT04806523 T AT 04806523T AT E484491 T1 ATE484491 T1 AT E484491T1
- Authority
- AT
- Austria
- Prior art keywords
- synthesis
- new method
- hydrogen atom
- enamide derivatives
- aryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/10—Preparation of carboxylic acid amides from compounds not provided for in groups C07C231/02 - C07C231/08
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C233/04—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C233/06—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Compositions Of Macromolecular Compounds (AREA)
Abstract
Ene-amide derivative of formula (IIE)
wherein
R4 is a hydrogen atom, an alkyl, an aryl, an alkylaryl, said groups are substituted or not with a halogen atom as C1, Br, or F;
R7, R8, R9 and R10, identical or different, with not simultaneously an hydrogen atom, are an hydrogen atom, a functional group, an alkyl, an aryl, preferably R7, R8 and R10 are an hydrogen atom, R9 is a methoxy and R4 is a methyl.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP03293281A EP1547997A1 (en) | 2003-12-22 | 2003-12-22 | New process for the synthesis of enamide derivatives |
PCT/IB2004/004363 WO2005063687A2 (en) | 2003-12-22 | 2004-12-22 | New process for the synthesis of eneamide derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE484491T1 true ATE484491T1 (en) | 2010-10-15 |
Family
ID=34530825
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT04806523T ATE484491T1 (en) | 2003-12-22 | 2004-12-22 | NEW METHOD FOR THE SYNTHESIS OF ENAMIDE DERIVATIVES |
Country Status (14)
Country | Link |
---|---|
US (1) | US7884243B2 (en) |
EP (3) | EP1547997A1 (en) |
JP (1) | JP4597141B2 (en) |
KR (1) | KR101155389B1 (en) |
CN (2) | CN101265210A (en) |
AT (1) | ATE484491T1 (en) |
DE (1) | DE602004029611D1 (en) |
DK (1) | DK1716097T3 (en) |
ES (1) | ES2354294T3 (en) |
IL (1) | IL176346A (en) |
PL (1) | PL1716097T3 (en) |
PT (1) | PT1716097E (en) |
SI (1) | SI1716097T1 (en) |
WO (1) | WO2005063687A2 (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1797030A1 (en) | 2004-09-08 | 2007-06-20 | Teva Pharmaceuticals USA, Inc. | Improved process for the synthesis of indanylamine or aminotetralin derivatives and novel intermediates |
ES2643602T3 (en) * | 2006-03-31 | 2017-11-23 | Sunovion Pharmaceuticals Inc. | Amines and chiral |
CN101875590B (en) * | 2010-07-19 | 2013-09-18 | 西北大学 | Method for synthesizing acrylamide compound |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3375287A (en) * | 1961-08-30 | 1968-03-26 | Union Carbide Corp | Process for isomerizing ethylenically unsaturated compound possessing cycloaliphatic nucleus |
JPS52133905A (en) * | 1976-04-30 | 1977-11-09 | Sumitomo Chem Co Ltd | Preparation of enamides |
US4194050A (en) * | 1976-04-30 | 1980-03-18 | Sumitomo Chemical Company, Limited | Process for producing an enamide |
WO1999018065A1 (en) * | 1997-10-03 | 1999-04-15 | Chirotech Technology Limited | Chiral amines |
US6737547B1 (en) * | 1998-12-31 | 2004-05-18 | Teva Pharmaceutical Industries, Ltd. | Compositions containing and methods of using N-acyl-1H-aminoindenes |
US6635784B2 (en) * | 2000-09-29 | 2003-10-21 | Eastman Chemical Company | Process for the preparation of enantiomerically-enriched cyclopropylalanine derivates |
EP1574498A1 (en) * | 2004-02-19 | 2005-09-14 | PPG-Sipsy | Process for the synthesis of substituted alpha-aminoindan derivatives |
-
2003
- 2003-12-22 EP EP03293281A patent/EP1547997A1/en not_active Withdrawn
-
2004
- 2004-12-22 EP EP07018349A patent/EP1897868A1/en not_active Withdrawn
- 2004-12-22 AT AT04806523T patent/ATE484491T1/en active
- 2004-12-22 SI SI200431559T patent/SI1716097T1/en unknown
- 2004-12-22 KR KR1020067011858A patent/KR101155389B1/en active IP Right Grant
- 2004-12-22 EP EP04806523A patent/EP1716097B1/en active Active
- 2004-12-22 CN CNA2008100912952A patent/CN101265210A/en active Pending
- 2004-12-22 PL PL04806523T patent/PL1716097T3/en unknown
- 2004-12-22 US US10/583,902 patent/US7884243B2/en active Active
- 2004-12-22 JP JP2006546407A patent/JP4597141B2/en not_active Expired - Fee Related
- 2004-12-22 DE DE602004029611T patent/DE602004029611D1/en active Active
- 2004-12-22 CN CN2004800386020A patent/CN1898194B/en active Active
- 2004-12-22 WO PCT/IB2004/004363 patent/WO2005063687A2/en not_active Application Discontinuation
- 2004-12-22 PT PT04806523T patent/PT1716097E/en unknown
- 2004-12-22 ES ES04806523T patent/ES2354294T3/en active Active
- 2004-12-22 DK DK04806523.9T patent/DK1716097T3/en active
-
2006
- 2006-06-15 IL IL176346A patent/IL176346A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
CN1898194B (en) | 2010-12-29 |
CN101265210A (en) | 2008-09-17 |
DE602004029611D1 (en) | 2010-11-25 |
WO2005063687A2 (en) | 2005-07-14 |
EP1547997A1 (en) | 2005-06-29 |
EP1716097A2 (en) | 2006-11-02 |
ES2354294T3 (en) | 2011-03-11 |
PL1716097T3 (en) | 2011-04-29 |
DK1716097T3 (en) | 2011-01-24 |
WO2005063687A3 (en) | 2005-10-27 |
US7884243B2 (en) | 2011-02-08 |
EP1897868A1 (en) | 2008-03-12 |
US20070129573A1 (en) | 2007-06-07 |
JP4597141B2 (en) | 2010-12-15 |
CN1898194A (en) | 2007-01-17 |
KR101155389B1 (en) | 2012-06-20 |
JP2007517017A (en) | 2007-06-28 |
KR20070057693A (en) | 2007-06-07 |
SI1716097T1 (en) | 2011-01-31 |
PT1716097E (en) | 2011-01-17 |
IL176346A (en) | 2011-01-31 |
EP1716097B1 (en) | 2010-10-13 |
IL176346A0 (en) | 2006-10-05 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1108924T1 (en) | Pyrrolidine and Pepperidine Derivatives as NK1 Antagonists | |
CO4970713A1 (en) | DERIVATIVES OF CARBOXAMIDOTIAZOLES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM | |
DE59807486D1 (en) | METHOD FOR PRODUCING (HETERO) AROMATIC HYDROXYLAMINE | |
CO4970780A1 (en) | NEW PIRIDAZINE HETERO-CYCLE COMPOUNDS | |
MEP7808A (en) | Process for preparing 4-trifluoromethylsulphinylpyrazole derivative | |
NO331165B1 (en) | Derivatives of dioxane-2-alkylcarbamates, processes for their preparation and use thereof for the preparation of medicaments | |
ATE425136T1 (en) | METHOD FOR PRODUCING SUBSTITUTED 3-ARYL-BUTYL AMINE COMPOUNDS | |
CO4520230A1 (en) | DERIVATIVES OF [3- (4-PHENYLPIPERACIN-1-IL) PROPYLAMINE, UNCLE AND OXYL] -PIRIDINE, PYRIMIDINE AND BENZENE AS ALPHA ANTAGONISTS 1- ADRENOCEPTORS | |
TW200607828A (en) | Polymer, polymer film and polymer film device using same | |
MX9806246A (en) | NOVEL PIPERIDINES DERIVED FROM 1-/(PIPERAZIN-1-YL)ARYL(OXY/AMINO)CARBONYL/-4-ARYL-PIPERIDIN E AS SELECTIVE 5-HT1Db RECEPTOR ANTAGONISTS. | |
EA200600485A1 (en) | Method of producing 2-oxo-1-pyrrolidine derivatives | |
DE602005026827D1 (en) | PROCESS FOR THE PREPARATION OF ISOINDOL DERIVATIVES | |
ATE484491T1 (en) | NEW METHOD FOR THE SYNTHESIS OF ENAMIDE DERIVATIVES | |
DK1362040T3 (en) | Process for preparing mesylates of piperidine derivatives | |
ATE299877T1 (en) | METHOD FOR PRODUCING ARYLACETYLAMINOTHIAZOLES | |
PT1140761E (en) | BENZOFENONAS AND THEIR USE AS PHOTO-INITIATORS | |
DE59906807D1 (en) | METHOD FOR RACEMIZING OPTICALLY ACTIVE AMINES | |
DE60125378D1 (en) | PROCESS FOR THE PREPARATION OF 2-AMINOMETHYL-HALOGEN-PYRIDINES | |
DE69808771D1 (en) | A METHOD FOR PRODUCING TETRAAZA MACROCYCLEN | |
YU74201A (en) | Novel synthesis of piperazine ring | |
ATE310735T1 (en) | METHOD FOR PRODUCING SPIROCYCLIC TETRONSIC ACID DERIVATIVES | |
DE60003169D1 (en) | METHOD FOR PRODUCING [S- (R *, S *)] - G (B) - [[1- [1-OXO-3- (4-PIPERIDINYL) PROPYL] -3-PIPERIDINYL] CARBONYL] AMINO] -3 -PYRIDINPROPANSÄUREDERIVATE | |
ATE280769T1 (en) | METHOD FOR PRODUCING VITRONECTIN RECEPTOR ANTAGONISTS | |
DE59712632D1 (en) | PROCESS FOR THE PREPARATION OF 3-PYRROLINE-2-CARBOXYLIC ACID DERIVATIVES | |
ATE241594T1 (en) | N-PHENYLACETOACETAMIDE AND METHOD FOR THE PRODUCTION THEREOF |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification |
Ref document number: 1716097 Country of ref document: EP |