ATE414060T1 - Verfahren und zwischenprodukte zur herstellung von pyrrolidinen - Google Patents

Verfahren und zwischenprodukte zur herstellung von pyrrolidinen

Info

Publication number
ATE414060T1
ATE414060T1 AT01935453T AT01935453T ATE414060T1 AT E414060 T1 ATE414060 T1 AT E414060T1 AT 01935453 T AT01935453 T AT 01935453T AT 01935453 T AT01935453 T AT 01935453T AT E414060 T1 ATE414060 T1 AT E414060T1
Authority
AT
Austria
Prior art keywords
pyrrolidines
producing
intermediate products
ribofuranoside
erythro
Prior art date
Application number
AT01935453T
Other languages
English (en)
Inventor
Rawle Hollingsworth
Original Assignee
Univ Michigan State
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Michigan State filed Critical Univ Michigan State
Application granted granted Critical
Publication of ATE414060T1 publication Critical patent/ATE414060T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/08Preparation of carboxylic acid esters by reacting carboxylic acids or symmetrical anhydrides with the hydroxy or O-metal group of organic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms
    • C07D207/262-Pyrrolidones
    • C07D207/2732-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/67Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
    • C07C69/716Esters of keto-carboxylic acids or aldehydo-carboxylic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12Oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/02Acyclic radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biotechnology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT01935453T 2000-08-02 2001-05-14 Verfahren und zwischenprodukte zur herstellung von pyrrolidinen ATE414060T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US09/630,765 US6414163B1 (en) 2000-08-02 2000-08-02 Process and intermediate compounds for the preparation of pyrrolidines

Publications (1)

Publication Number Publication Date
ATE414060T1 true ATE414060T1 (de) 2008-11-15

Family

ID=24528483

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01935453T ATE414060T1 (de) 2000-08-02 2001-05-14 Verfahren und zwischenprodukte zur herstellung von pyrrolidinen

Country Status (9)

Country Link
US (8) US6414163B1 (de)
EP (3) EP1947084A2 (de)
JP (2) JP3934047B2 (de)
KR (2) KR100536981B1 (de)
AT (1) ATE414060T1 (de)
AU (2) AU6154701A (de)
CA (1) CA2415097C (de)
DE (1) DE60136544D1 (de)
WO (1) WO2002010130A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6161439A (en) 1997-05-12 2000-12-19 Stanley; James Gregory Seat belt tension prediction
US6679855B2 (en) * 2000-11-07 2004-01-20 Gerald Horn Method and apparatus for the correction of presbyopia using high intensity focused ultrasound
KR100543478B1 (ko) * 2002-12-31 2006-01-20 엘지.필립스 엘시디 주식회사 유기전계 발광소자와 그 제조방법
DE10301806A1 (de) * 2003-01-20 2004-07-29 Bayer Cropscience Ag Selektive Herbizide auf Basis von substituierten, cyclischen Dicarbonylverbindungen und Safenern
CA2621717A1 (en) * 2005-09-08 2007-03-15 Michigan State University Pyrrolo-thiazines and processes for the preparation and use thereof
US8353402B2 (en) 2008-10-06 2013-01-15 Rehrig Pacific Company Stackable low depth tray
EP2248780A1 (de) 2009-05-06 2010-11-10 BK Giulini GmbH Abbinde- und Enthärtungsbeschleuniger
JP2012184190A (ja) * 2011-03-04 2012-09-27 Yamaguchi Univ 4−ケト−d−リボン酸、4−ケト−d−リボース及びそれらの製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4973602A (en) * 1988-11-03 1990-11-27 G. D. Searle & Co. Antiviral compounds and a method of use thereas
US5461071A (en) * 1994-10-21 1995-10-24 Merck & Co., Inc. Anti-fungal agents
EP0884050A1 (de) * 1995-09-08 1998-12-16 Novo Nordisk A/S Verwendung von 3,4-dihydroxy-2-hydroxymethylpyrrolidin zur behandlung von diabetes
US5801247A (en) * 1997-01-23 1998-09-01 Temple University-Of The Commonwealth System Of Higher Education Process for the enantioselective synthesis of hydroxypyrrolidines from amino acids and products thereof
JPH11255742A (ja) * 1998-03-13 1999-09-21 Sumitomo Chem Co Ltd 光学活性ヒドロキシラクタム化合物の製造方法

Also Published As

Publication number Publication date
JP2004505108A (ja) 2004-02-19
US6492534B2 (en) 2002-12-10
DE60136544D1 (de) 2008-12-24
KR100570410B1 (ko) 2006-04-11
US20020026072A1 (en) 2002-02-28
US20020026073A1 (en) 2002-02-28
US6518437B1 (en) 2003-02-11
US20020019542A1 (en) 2002-02-14
JP2007126464A (ja) 2007-05-24
WO2002010130A1 (en) 2002-02-07
US20020019561A1 (en) 2002-02-14
EP1947082A3 (de) 2009-04-29
EP1305284A1 (de) 2003-05-02
EP1305284A4 (de) 2005-08-03
US6583297B2 (en) 2003-06-24
US20020026071A1 (en) 2002-02-28
CA2415097C (en) 2007-09-18
EP1947082A2 (de) 2008-07-23
EP1947084A2 (de) 2008-07-23
CA2415097A1 (en) 2002-02-07
US6414163B1 (en) 2002-07-02
AU6154701A (en) 2002-02-13
US6423867B1 (en) 2002-07-23
US20020026074A1 (en) 2002-02-28
JP3934047B2 (ja) 2007-06-20
KR100536981B1 (ko) 2005-12-14
AU2001261547B2 (en) 2004-08-12
KR20050095917A (ko) 2005-10-04
KR20030019574A (ko) 2003-03-06
US6482974B2 (en) 2002-11-19
US6482973B2 (en) 2002-11-19
EP1305284B1 (de) 2008-11-12

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Legal Events

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