ATE410171T1 - Graduierte östrogen-kontrazeptiva - Google Patents

Graduierte östrogen-kontrazeptiva

Info

Publication number
ATE410171T1
ATE410171T1 AT04819121T AT04819121T ATE410171T1 AT E410171 T1 ATE410171 T1 AT E410171T1 AT 04819121 T AT04819121 T AT 04819121T AT 04819121 T AT04819121 T AT 04819121T AT E410171 T1 ATE410171 T1 AT E410171T1
Authority
AT
Austria
Prior art keywords
graduated
contraceptives
estrogen contraceptives
graduated estrogen
estrogen
Prior art date
Application number
AT04819121T
Other languages
English (en)
Inventor
Roger Boissonneault
Original Assignee
Warner Chilcott Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Chilcott Co Inc filed Critical Warner Chilcott Co Inc
Application granted granted Critical
Publication of ATE410171T1 publication Critical patent/ATE410171T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Nutrition Science (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT04819121T 2003-11-14 2004-11-12 Graduierte östrogen-kontrazeptiva ATE410171T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US52018203P 2003-11-14 2003-11-14

Publications (1)

Publication Number Publication Date
ATE410171T1 true ATE410171T1 (de) 2008-10-15

Family

ID=34619442

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04819121T ATE410171T1 (de) 2003-11-14 2004-11-12 Graduierte östrogen-kontrazeptiva

Country Status (9)

Country Link
US (2) US8124595B2 (de)
EP (1) EP1689411B1 (de)
JP (1) JP2007511533A (de)
CN (1) CN1878558A (de)
AT (1) ATE410171T1 (de)
CA (1) CA2542854C (de)
DE (1) DE602004017045D1 (de)
IL (1) IL174893A (de)
WO (1) WO2005049142A2 (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1735056B1 (de) * 2004-03-19 2012-10-24 Warner Chilcott Company, LLC Mehrphasige orale kontrazeptionsmethode mit verlängertem zyklus
CA2609336C (en) 2005-06-29 2013-12-10 Warner Chilcott Company, Inc. Quadraphasic continuous graduated estrogen contraceptive
MX2008011074A (es) 2006-03-02 2008-09-10 Warner Chilcott Co Inc Metodo anticonceptivo oral multifasico de ciclo prolongado.
WO2009112231A2 (en) * 2008-03-10 2009-09-17 Schuermann Rolf New drospirenone/17beta-estradil regimen, pharmaceutical combination product and kit for performing this regimen
TW200946542A (en) * 2008-03-10 2009-11-16 Vladimir Hanes New drospirenone/17β-estradiol regimen, pharmaceutical combination product and kit for performing this regimen
KR20130097073A (ko) 2010-04-15 2013-09-02 바이엘 인텔렉쳐 프로퍼티 게엠베하 초저-용량의 ｈｒｔ용 고체 경구 투여 형태
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
EP2782584B1 (de) 2011-11-23 2021-06-09 TherapeuticsMD, Inc. Natürliche kombinierte hormonersatzformulierungen und -therapien
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
AR100562A1 (es) 2014-05-22 2016-10-12 Therapeuticsmd Inc Composición farmacéutica de estradiol y progesterona para terapia de reemplazo hormonal
US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
WO2017173044A1 (en) 2016-04-01 2017-10-05 Therapeuticsmd Inc. Steroid hormone compositions in medium chain oils
KR20180126582A (ko) 2016-04-01 2018-11-27 쎄러퓨틱스엠디, 인코퍼레이티드 스테로이드 호르몬 약제학적 조성물
US11633405B2 (en) 2020-02-07 2023-04-25 Therapeuticsmd, Inc. Steroid hormone pharmaceutical formulations
US20230135376A1 (en) * 2020-06-25 2023-05-04 Millicent Pharma Limited Multiphasic contraceptive and/or hormone replacement therapy
CA3234836A1 (en) 2021-09-07 2023-03-16 Millicent Pharma Limited Contraceptive regimen including reduced level of estrogen
US12138270B2 (en) 2021-09-07 2024-11-12 Millicent Pharma Limited Contraceptive regimen including reduced level of estrogen

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4292315A (en) * 1977-12-30 1981-09-29 Nichols Vorys Follicular phase estrogen or progestin with physiologic estrogen/progestin luteal phase replacement drug delivery system
US4921843A (en) 1988-10-20 1990-05-01 Pasquale Samuel A Contraception system and method
US4962098A (en) * 1987-06-15 1990-10-09 Warner-Lambert Company Graduated estrogen contraceptive
DK174724B1 (da) 1986-07-15 2003-10-06 Wyeth Corp Anvendelse af et præparat omfattende et østrogen og et progestogen til fremstilling af en dosisform til tilvejebringelse af hormonerstatningsterapi og kontraception til kvinder i præmenopausen samt pakning til tilvejebringelse af præparatet
DE4313926A1 (de) 1993-04-28 1994-11-03 Jenapharm Gmbh Pharmazeutisches Mehrphasenpräparat zur hormonalen Kontrazeption
US5552394A (en) * 1994-07-22 1996-09-03 The Medical College Of Hampton Roads Low dose oral contraceptives with less breakthrough bleeding and sustained efficacy
US5888543A (en) 1996-07-26 1999-03-30 American Home Products Corporation Oral contraceptives
US6479475B1 (en) * 1996-07-26 2002-11-12 Wyeth Oral contraceptive
US6511970B1 (en) * 1996-09-13 2003-01-28 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of products that induce transforming growth factor-beta and/or apoptosis in the ovarian epithelium
EP1735056B1 (de) * 2004-03-19 2012-10-24 Warner Chilcott Company, LLC Mehrphasige orale kontrazeptionsmethode mit verlängertem zyklus
US7704984B2 (en) * 2005-04-22 2010-04-27 Warner Chilcott Company, Llc Extended estrogen dosing contraceptive regimen
CA2609336C (en) * 2005-06-29 2013-12-10 Warner Chilcott Company, Inc. Quadraphasic continuous graduated estrogen contraceptive
MX2008011074A (es) * 2006-03-02 2008-09-10 Warner Chilcott Co Inc Metodo anticonceptivo oral multifasico de ciclo prolongado.

Also Published As

Publication number Publication date
EP1689411A2 (de) 2006-08-16
IL174893A0 (en) 2009-02-11
CA2542854C (en) 2012-04-17
EP1689411B1 (de) 2008-10-08
CA2542854A1 (en) 2005-06-02
WO2005049142A2 (en) 2005-06-02
CN1878558A (zh) 2006-12-13
US8124595B2 (en) 2012-02-28
WO2005049142A3 (en) 2005-09-29
JP2007511533A (ja) 2007-05-10
IL174893A (en) 2011-11-30
US20110059928A1 (en) 2011-03-10
DE602004017045D1 (de) 2008-11-20
US9132137B2 (en) 2015-09-15
US20050107351A1 (en) 2005-05-19

Similar Documents

Publication Publication Date Title
DE602004017045D1 (de) Graduierte östrogen-kontrazeptiva
SG166107A1 (en) Quadraphasic continuous graduated estrogen contraceptive
TW200603813A (en) Cyclic progestin regimens and kits
IL172959A0 (en) Methods for contraception using estrogen and progestin
TR200001460T2 (tr) Çok düşük estrojen dozları kullanılarak menopoz sonrası kadınların tedavisine yönelik metodlar
ATE311204T1 (de) Estrogen-zyklodextrin komplexe-zusammensetzungen
BRPI0512993A (pt) uso de um antagonista de pr, kit farmaceuticamente últil, e, método de contracepção em uma fêmea em idade de parto
BRPI0214716B8 (pt) kit, preparos, e uso de estrogênio e progestina na fabricação de um medicamento para uso na prevenção de gravidez
DK1623711T3 (da) Eksternt plaster indeholdende östrogen og/eller progestogen
MXPA02012896A (es) Combinaciones de estatinas, agentes estrogenicos y opcionalmente estrogenos.
MXPA03004499A (es) Kit de repinotan.
DK1293210T3 (da) Midler og fremgangsmåde til hormonal prævention
BR0008437A (pt) Inibidores esteróides de sulfatase e métodos parafabricação e uso dos mesmos
MX2007004120A (es) Metodos de tratamiento hormonal utilizando regimentes de ciclo prolongado de dosis ascendente.
AR043013A1 (es) Composicion farmaceutica destinada al tratamiento de la endometriosis
FR2819395B1 (fr) Implant dentaire transitoire de preparation d'une alveole
ATE303397T1 (de) 9-alpha-substituierte estratriene als selektiv wirksame estrogene
BR0111509A (pt) Kit iniciante para contraceptivos orais de baixa dose
DK1635843T3 (da) Terapi, der omfatter dienogest for hormonerstatning og depression
DE60202954D1 (de) Tetrahydrochinolin-derivate zur behandlung von krankheiten ausgelöst durch zu hohem oder zu niedrigem oestrogenspiegel
WO2004011029A3 (en) Pharmaceutical compositions for penis enlargement
GB0201284D0 (en) Screening methods for contraceptive and fertility agents
DK1286666T3 (da) Starterkit for lavdoseret oralt antikonceptionsmiddel
EA200100745A1 (ru) СПОСОБ ПОЛУЧЕНИЯ 6β,7β;15β,16β- ДИМЕТИЛЕН-5β-ГИДРОКСИ-3-ОКСО-17α-АНДРОСТАН-21,17-КАРБАЛАКТОНА
DK200100065U3 (da) Penisekspander

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties