ATA525275A - PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALTS AND OPTICALLY ACTIVE FORMS - Google Patents

PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALTS AND OPTICALLY ACTIVE FORMS

Info

Publication number
ATA525275A
ATA525275A AT525275A AT525275A ATA525275A AT A525275 A ATA525275 A AT A525275A AT 525275 A AT525275 A AT 525275A AT 525275 A AT525275 A AT 525275A AT A525275 A ATA525275 A AT A525275A
Authority
AT
Austria
Prior art keywords
production
acid addition
addition salts
optically active
active forms
Prior art date
Application number
AT525275A
Other languages
German (de)
Other versions
AT344178B (en
Inventor
John Christopher Dr Danilewicz
Anthony Garth Evans
Allan Leslie Ham
Colin Dr Thomson
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Priority to AT453077A priority Critical patent/AT344184B/en
Priority to AT453277A priority patent/AT344186B/en
Priority to AT453177A priority patent/AT344185B/en
Publication of ATA525275A publication Critical patent/ATA525275A/en
Application granted granted Critical
Publication of AT344178B publication Critical patent/AT344178B/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
AT525275A 1974-07-25 1975-07-08 PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALT AND OPTICALLY ACTIVE FORMS AT344178B (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
AT453077A AT344184B (en) 1974-07-25 1977-06-27 PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALT AND OPTICALLY ACTIVE FORMS
AT453277A AT344186B (en) 1974-07-25 1977-06-27 PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALT AND OPTICALLY ACTIVE FORMS
AT453177A AT344185B (en) 1974-07-25 1977-06-27 PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALT AND OPTICALLY ACTIVE FORMS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3280574 1974-07-25

Publications (2)

Publication Number Publication Date
ATA525275A true ATA525275A (en) 1977-11-15
AT344178B AT344178B (en) 1978-07-10

Family

ID=10344259

Family Applications (1)

Application Number Title Priority Date Filing Date
AT525275A AT344178B (en) 1974-07-25 1975-07-08 PROCESS FOR THE PRODUCTION OF NEW QUINAZOLINE COMPOUNDS AND THEIR ACID ADDITION SALT AND OPTICALLY ACTIVE FORMS

Country Status (7)

Country Link
AT (1) AT344178B (en)
BE (1) BE831654A (en)
CS (1) CS192549B2 (en)
ES (4) ES439690A1 (en)
HU (1) HU174961B (en)
PL (6) PL104615B1 (en)
SU (5) SU578874A3 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070004763A1 (en) * 2005-06-10 2007-01-04 Nand Baindur Aminoquinoline and aminoquinazoline kinase modulators

Also Published As

Publication number Publication date
PL103791B1 (en) 1979-07-31
PL103798B1 (en) 1979-07-31
SU625606A3 (en) 1978-09-25
ES439690A1 (en) 1977-07-01
PL103797B1 (en) 1979-07-31
PL99427B1 (en) 1978-07-31
PL193423A1 (en) 1978-04-24
ES455984A1 (en) 1978-06-01
AT344178B (en) 1978-07-10
SU858563A3 (en) 1981-08-23
ES455985A1 (en) 1978-06-16
ES455986A1 (en) 1978-06-01
CS192549B2 (en) 1979-08-31
SU578874A3 (en) 1977-10-30
PL193422A1 (en) 1978-06-05
PL103789B1 (en) 1979-07-31
SU613723A3 (en) 1978-06-30
PL104615B1 (en) 1979-08-31
SU634671A3 (en) 1978-11-25
PL193419A1 (en) 1978-04-24
HU174961B (en) 1980-04-28
PL193420A1 (en) 1978-04-24
PL193421A1 (en) 1978-04-24
BE831654A (en) 1976-01-23

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