AT351545B - PROCESS FOR THE PREPARATION OF BENZODIAZEPINE DERIVATIVES - Google Patents

PROCESS FOR THE PREPARATION OF BENZODIAZEPINE DERIVATIVES

Info

Publication number
AT351545B
AT351545B AT224775A AT224775A AT351545B AT 351545 B AT351545 B AT 351545B AT 224775 A AT224775 A AT 224775A AT 224775 A AT224775 A AT 224775A AT 351545 B AT351545 B AT 351545B
Authority
AT
Austria
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
AT224775A
Other languages
German (de)
Other versions
ATA224775A (en
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of ATA224775A publication Critical patent/ATA224775A/en
Application granted granted Critical
Publication of AT351545B publication Critical patent/AT351545B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/28Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
AT224775A 1974-03-25 1975-03-24 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE DERIVATIVES AT351545B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH414974A CH596173A5 (en) 1974-03-25 1974-03-25 CNS Depressant 5-aryl-benzodiazepine prepn.

Publications (2)

Publication Number Publication Date
ATA224775A ATA224775A (en) 1979-01-15
AT351545B true AT351545B (en) 1979-07-25

Family

ID=4270728

Family Applications (1)

Application Number Title Priority Date Filing Date
AT224775A AT351545B (en) 1974-03-25 1975-03-24 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE DERIVATIVES

Country Status (12)

Country Link
JP (1) JPS50130777A (en)
AT (1) AT351545B (en)
CA (1) CA1055491A (en)
CH (1) CH596173A5 (en)
DD (1) DD118644A5 (en)
DK (1) DK123675A (en)
ES (1) ES435935A1 (en)
FI (1) FI750380A7 (en)
NL (1) NL7502283A (en)
NO (1) NO751008L (en)
SE (1) SE7503301L (en)
YU (1) YU57775A (en)

Also Published As

Publication number Publication date
FI750380A7 (en) 1975-09-26
CA1055491A (en) 1979-05-29
DK123675A (en) 1975-09-26
JPS50130777A (en) 1975-10-16
ES435935A1 (en) 1976-12-16
NO751008L (en) 1975-09-26
SE7503301L (en) 1975-09-26
DD118644A5 (en) 1976-03-12
CH596173A5 (en) 1978-02-28
NL7502283A (en) 1975-09-29
ATA224775A (en) 1979-01-15
YU57775A (en) 1982-05-31

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties