AT343802B - Verfahren zur herstellung von derivaten von 4,6-di-0- (aminoglycosyl)-2-deoxystreptaminen - Google Patents
Verfahren zur herstellung von derivaten von 4,6-di-0- (aminoglycosyl)-2-deoxystreptaminenInfo
- Publication number
- AT343802B AT343802B AT895075A AT895075A AT343802B AT 343802 B AT343802 B AT 343802B AT 895075 A AT895075 A AT 895075A AT 895075 A AT895075 A AT 895075A AT 343802 B AT343802 B AT 343802B
- Authority
- AT
- Austria
- Prior art keywords
- deoxystreptamines
- aminoglycosyl
- derivatives
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- C07H15/236—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US52859374A | 1974-11-29 | 1974-11-29 | |
US05/611,289 US4000261A (en) | 1974-11-29 | 1975-09-08 | 5-epi-4,6-di-o-(aminoglycosyl)-2-deoxystreptamines, methods for their manufacture and intermediates useful therein, methods for their use as antibacterial agents and compositions useful therefor |
Publications (2)
Publication Number | Publication Date |
---|---|
ATA895075A ATA895075A (de) | 1977-10-15 |
AT343802B true AT343802B (de) | 1978-06-26 |
Family
ID=27062767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT895075A AT343802B (de) | 1974-11-29 | 1975-11-25 | Verfahren zur herstellung von derivaten von 4,6-di-0- (aminoglycosyl)-2-deoxystreptaminen |
Country Status (2)
Country | Link |
---|---|
US (1) | US4000261A (de) |
AT (1) | AT343802B (de) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4217446A (en) * | 1974-10-26 | 1980-08-12 | Pfizer Inc. | ωAmino-2-hydroxyalkyl derivatives of aminoglycoside antibiotics |
NZ184213A (en) * | 1976-06-16 | 1980-05-27 | Pfizer | 2-deoxystreptamine aminoglycosides and antibacterial pharmaceutical compositions |
DE2647807A1 (de) * | 1976-10-22 | 1978-04-27 | Merck Patent Gmbh | Verfahren zur herstellung von garamin und garaminderivaten |
DE2840907A1 (de) * | 1978-09-20 | 1980-04-03 | Bayer Ag | Selektiv geschuetzte 4,6-di-o-(aminoglykosyl)-1,3-diaminocyclitole |
US4272626A (en) * | 1979-09-26 | 1981-06-09 | Abbott Laboratories | Method of producing 1-epi-2-deoxyfortimicin A and intermediates therefor |
US4387219A (en) * | 1979-11-13 | 1983-06-07 | Sterling Drug Inc. | 2-Hydroxy gentamicin compounds |
US4288547A (en) * | 1979-11-13 | 1981-09-08 | Haruo Yamamoto | Fermentative process for preparing antibiotics of the gentamicin class |
EP1710248A4 (de) * | 2004-01-21 | 2009-05-27 | Meiji Seika Kaisha | Neues aminoglycosid-antibiotikum mit wirkung gegen methicillin-resistentes staphylococcus aureus (mrsa) |
PT2217610T (pt) | 2007-11-21 | 2017-02-10 | Achaogen Inc | Análogos de aminoglicosido antibacterianos |
WO2010132765A2 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
WO2010132757A2 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
WO2010132760A1 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial derivatives of tobramycin |
WO2010132759A1 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial derivatives of dibekacin |
WO2010132768A1 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial derivatives of sisomicin |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3828021A (en) * | 1972-06-14 | 1974-08-06 | Merck & Co Inc | Gentamicin c1 derivatives |
US3920628A (en) * | 1972-10-24 | 1975-11-18 | Schering Corp | 2{41 -Deoxyaminoglycosides and 2{41 -epi-amino-3{41 -desamino derivatives thereof, methods for their manufacture and novel intermediates useful therein |
-
1975
- 1975-09-08 US US05/611,289 patent/US4000261A/en not_active Expired - Lifetime
- 1975-11-25 AT AT895075A patent/AT343802B/de not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ATA895075A (de) | 1977-10-15 |
US4000261A (en) | 1976-12-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AT333777B (de) | Verfahren zur herstellung von 1,2-benzothiazin-3-carboxamiden | |
DD127731A5 (de) | Verfahren zur herstellung von cephalosporansaeurederivaten | |
ATA966275A (de) | Verfahren zur herstellung von p-benzochinondiketalen | |
AT343802B (de) | Verfahren zur herstellung von derivaten von 4,6-di-0- (aminoglycosyl)-2-deoxystreptaminen | |
AT336613B (de) | Verfahren zur herstellung von 2,2,6,6-tetramethyl-4-oxopiperidin | |
AT338262B (de) | Verfahren zur herstellung von 2,2,6,6-tetramethyl-4-oxopiperidin | |
AT333774B (de) | Verfahren zur herstellung von 3-phenylpyridazonen | |
DD129334A5 (de) | Verfahren zur herstellung von 4-androsten-3,17-dion-derivaten | |
AT338263B (de) | Verfahren zur herstellung von 2,2,6,6-tetramethyl-4-oxopiperidin | |
ATA904575A (de) | Verfahren zur herstellung von neuen 1,3-dialkyl-7-aminoalkylxanthinen | |
ATA751376A (de) | Verfahren zur herstellung von 24,25-dihydroxy- cholesterinderivaten | |
AT333749B (de) | Verfahren zur herstellung von neuen 2-arylamino-2-imidazolinderivaten | |
AT346842B (de) | Verfahren zur herstellung von 1,2-benz- isothiazolen | |
AT344702B (de) | Verfahren zur herstellung von neuen chinoxalin-1,4-dioxyd-derivaten | |
DD122962A5 (de) | Verfahren zur herstellung von halogenanthrachinonen | |
AT350558B (de) | Verfahren zur herstellung von 2,4-dioxo- oxazolidinen | |
AT334909B (de) | Verfahren zur herstellung von substituierten thiocarbaminsaure-s-alkylestern | |
AT341672B (de) | Verfahren zur herstellung von 3-methylencephamsulfoxiden | |
AT343120B (de) | Verfahren zur herstellung von 6-chlor-2-chlormethyl-4-phenylchinazolin-3-oxid | |
DD122986A1 (de) | Verfahren zur herstellung von polyesteralkoholen | |
AT350199B (de) | Verfahren zur herstellung von 17-monoestern von 17alfa,21-dihydroxysteroiden | |
DD129333A5 (de) | Verfahren zur herstellung von 4-androsten-3,17-dion-derivaten | |
AT344675B (de) | Verfahren zur herstellung von 3-fluor-dl-alanin | |
DD122973A5 (de) | Verfahren zur herstellung von 4a-aryl-transdecahydroisochinolinen | |
AT334336B (de) | Verfahren zur herstellung von 1-phenyl -2- glycinamidoathanolen-(1) |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
ELJ | Ceased due to non-payment of the annual fee |