AT259565B - Verfahren zur Herstellung von neuen Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von neuen Benzodiazepin-Derivaten

Info

Publication number
AT259565B
AT259565B AT176066A AT176066A AT259565B AT 259565 B AT259565 B AT 259565B AT 176066 A AT176066 A AT 176066A AT 176066 A AT176066 A AT 176066A AT 259565 B AT259565 B AT 259565B
Authority
AT
Austria
Prior art keywords
preparation
benzodiazepine derivatives
new benzodiazepine
new
derivatives
Prior art date
Application number
AT176066A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AT259565B publication Critical patent/AT259565B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • HELECTRICITY
    • H01ELECTRIC ELEMENTS
    • H01RELECTRICALLY-CONDUCTIVE CONNECTIONS; STRUCTURAL ASSOCIATIONS OF A PLURALITY OF MUTUALLY-INSULATED ELECTRICAL CONNECTING ELEMENTS; COUPLING DEVICES; CURRENT COLLECTORS
    • H01R33/00Coupling devices specially adapted for supporting apparatus and having one part acting as a holder providing support and electrical connection via a counterpart which is structurally associated with the apparatus, e.g. lamp holders; Separate parts thereof
    • H01R33/05Two-pole devices
    • H01R33/06Two-pole devices with two current-carrying pins, blades or analogous contacts, having their axes parallel to each other
    • H01R33/08Two-pole devices with two current-carrying pins, blades or analogous contacts, having their axes parallel to each other for supporting tubular fluorescent lamp

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT176066A 1965-03-22 1966-02-25 Verfahren zur Herstellung von neuen Benzodiazepin-Derivaten AT259565B (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US441863A US3320239A (en) 1965-03-22 1965-03-22 Certain 2, 3-bis(substituted amino)-5-aryl-3h-1, 4-benzodiazepine-4-oxide compounds and their preparation

Publications (1)

Publication Number Publication Date
AT259565B true AT259565B (de) 1968-01-25

Family

ID=23754595

Family Applications (1)

Application Number Title Priority Date Filing Date
AT176066A AT259565B (de) 1965-03-22 1966-02-25 Verfahren zur Herstellung von neuen Benzodiazepin-Derivaten

Country Status (12)

Country Link
US (1) US3320239A (de)
AT (1) AT259565B (de)
BE (1) BE677983A (de)
BR (1) BR6677950D0 (de)
CH (1) CH460791A (de)
DE (1) DE1695129A1 (de)
ES (1) ES324458A1 (de)
FR (1) FR5307M (de)
GB (1) GB1095220A (de)
IL (1) IL25374A (de)
NL (1) NL6603736A (de)
SE (1) SE322782B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3933794A (en) * 1971-08-04 1976-01-20 The Upjohn Company 2-(2-Alkynylamino)-3H-1,4-benzodiazepines
US4755508A (en) * 1984-06-26 1988-07-05 Merck & Co., Inc. Benzodiazepine analogs and use as antogonists of gastrin and cholecystokinin
DK287185A (da) * 1984-06-26 1986-02-24 Merck & Co Inc Benzodiazepinderivat og farmaceutisk praeparat indeholdende et saadantderivat
AU678503B2 (en) * 1993-09-24 1997-05-29 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds and their use as squalene synthetase inhibitors

Also Published As

Publication number Publication date
US3320239A (en) 1967-05-16
CH460791A (de) 1968-08-15
FR5307M (de) 1967-08-21
ES324458A1 (es) 1967-03-16
BR6677950D0 (pt) 1973-09-11
SE322782B (de) 1970-04-20
DE1695129A1 (de) 1970-02-12
IL25374A (en) 1970-01-29
BE677983A (de) 1966-09-19
NL6603736A (de) 1966-09-23
GB1095220A (en) 1967-12-13

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