AR225181A1 - Procedimiento para obtener nuevos derivados de 3-(((fosfonoxi-alquil)-hidrazono)metil)rifamicina sv - Google Patents

Procedimiento para obtener nuevos derivados de 3-(((fosfonoxi-alquil)-hidrazono)metil)rifamicina sv

Info

Publication number
AR225181A1
AR225181A1 AR281548A AR28154880A AR225181A1 AR 225181 A1 AR225181 A1 AR 225181A1 AR 281548 A AR281548 A AR 281548A AR 28154880 A AR28154880 A AR 28154880A AR 225181 A1 AR225181 A1 AR 225181A1
Authority
AR
Argentina
Prior art keywords
rifamicina
phosphonoxy
hydrazone
alkyl
methyl
Prior art date
Application number
AR281548A
Other languages
English (en)
Spanish (es)
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Application granted granted Critical
Publication of AR225181A1 publication Critical patent/AR225181A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AR281548A 1979-06-28 1980-06-26 Procedimiento para obtener nuevos derivados de 3-(((fosfonoxi-alquil)-hidrazono)metil)rifamicina sv AR225181A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7922461 1979-06-28

Publications (1)

Publication Number Publication Date
AR225181A1 true AR225181A1 (es) 1982-02-26

Family

ID=10506154

Family Applications (1)

Application Number Title Priority Date Filing Date
AR281548A AR225181A1 (es) 1979-06-28 1980-06-26 Procedimiento para obtener nuevos derivados de 3-(((fosfonoxi-alquil)-hidrazono)metil)rifamicina sv

Country Status (18)

Country Link
US (1) US4271155A (it)
JP (1) JPS5618993A (it)
KR (1) KR830002533B1 (it)
AR (1) AR225181A1 (it)
AU (1) AU536524B2 (it)
CA (1) CA1114814A (it)
DE (1) DE3024304A1 (it)
DK (1) DK155742C (it)
FR (1) FR2460304A1 (it)
GB (1) GB2051815B (it)
HK (1) HK23684A (it)
IE (1) IE49930B1 (it)
IT (1) IT1209333B (it)
NL (1) NL8003527A (it)
NZ (1) NZ194144A (it)
PH (1) PH15769A (it)
SE (1) SE451842B (it)
ZA (1) ZA803635B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004096285A2 (en) * 2003-04-25 2004-11-11 Gilead Sciences, Inc. Anti-infective phosphonate conjugates
EP1928890B1 (en) * 2005-08-11 2013-04-03 Targanta Therapeutics Inc. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR208F (it) * 1964-07-31
FR5223M (it) * 1965-11-12 1967-07-10
US4005076A (en) * 1971-06-24 1977-01-25 Gruppo Lepetit S.P.A. Hydrazones of 3-formylrifamycin SV
BE794100A (fr) * 1972-02-23 1973-05-16 Lepetit Spa Derives 3-hydrazonomethyles de rifamycine et leur preparation
AR205434A1 (es) * 1972-03-27 1976-05-07 Lepetit Spa Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv
GB1486118A (en) * 1975-03-05 1977-09-21 Lepetit Spa Rifamycin derivatives
GB1478563A (en) * 1975-03-05 1977-07-06 Lepetit Spa Rifamycin derivatives
GR64108B (en) * 1977-04-15 1980-01-24 Dso Pharmachim Method for the preparation of azomethine-derivatives of rifamycin s.v

Also Published As

Publication number Publication date
DK155742B (da) 1989-05-08
SE451842B (sv) 1987-11-02
IE49930B1 (en) 1986-01-08
PH15769A (en) 1983-03-24
NZ194144A (en) 1984-05-31
FR2460304A1 (fr) 1981-01-23
US4271155A (en) 1981-06-02
AU536524B2 (en) 1984-05-10
SE8004739L (sv) 1980-12-29
AU5918880A (en) 1981-01-08
IT1209333B (it) 1989-07-16
GB2051815A (en) 1981-01-21
NL8003527A (nl) 1980-12-30
HK23684A (en) 1984-03-23
IE801346L (en) 1980-12-28
JPS5618993A (en) 1981-02-23
FR2460304B1 (it) 1984-07-27
CA1114814A (en) 1981-12-22
KR830002533B1 (ko) 1983-11-12
KR830002767A (ko) 1983-05-30
JPS6348877B2 (it) 1988-09-30
ZA803635B (en) 1981-06-24
DK155742C (da) 1989-09-18
DE3024304A1 (de) 1981-02-05
DK269380A (da) 1980-12-29
GB2051815B (en) 1983-07-06
DE3024304C2 (it) 1991-10-31
IT8022817A0 (it) 1980-06-17

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