AR216288A1 - PROCEDURE FOR OBTAINING 1,1-DIOXIDO-4-HYDROXY-2H-HAVE- (3,4-E) -1,2-TIACIN-3-CARBOXAMIDE COMPOUNDS - Google Patents

PROCEDURE FOR OBTAINING 1,1-DIOXIDO-4-HYDROXY-2H-HAVE- (3,4-E) -1,2-TIACIN-3-CARBOXAMIDE COMPOUNDS

Info

Publication number
AR216288A1
AR216288A1 AR260104A AR26010475A AR216288A1 AR 216288 A1 AR216288 A1 AR 216288A1 AR 260104 A AR260104 A AR 260104A AR 26010475 A AR26010475 A AR 26010475A AR 216288 A1 AR216288 A1 AR 216288A1
Authority
AR
Argentina
Prior art keywords
tiacin
dioxido
hydroxy
procedure
obtaining
Prior art date
Application number
AR260104A
Other languages
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1158274A external-priority patent/CH608500A5/en
Priority claimed from CH1215774A external-priority patent/CH608501A5/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR216288A1 publication Critical patent/AR216288A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/34Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Manufacturing Of Printed Wiring (AREA)
  • Electroplating Methods And Accessories (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AR260104A 1974-08-26 1975-08-22 PROCEDURE FOR OBTAINING 1,1-DIOXIDO-4-HYDROXY-2H-HAVE- (3,4-E) -1,2-TIACIN-3-CARBOXAMIDE COMPOUNDS AR216288A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1158274A CH608500A5 (en) 1974-08-26 1974-08-26 Process for the preparation of thiazine derivatives
CH1215774A CH608501A5 (en) 1974-09-09 1974-09-09 Process for the preparation of thiazine derivatives

Publications (1)

Publication Number Publication Date
AR216288A1 true AR216288A1 (en) 1979-12-14

Family

ID=25708582

Family Applications (1)

Application Number Title Priority Date Filing Date
AR260104A AR216288A1 (en) 1974-08-26 1975-08-22 PROCEDURE FOR OBTAINING 1,1-DIOXIDO-4-HYDROXY-2H-HAVE- (3,4-E) -1,2-TIACIN-3-CARBOXAMIDE COMPOUNDS

Country Status (20)

Country Link
JP (1) JPS5826758B2 (en)
AR (1) AR216288A1 (en)
AT (1) AT350064B (en)
BR (1) BR7505463A (en)
DD (1) DD124119A5 (en)
DE (1) DE2537070A1 (en)
DK (1) DK137835B (en)
FI (1) FI59253C (en)
FR (3) FR2282893A1 (en)
GB (1) GB1519811A (en)
HU (1) HU173739B (en)
IE (1) IE41457B1 (en)
IL (1) IL47877A (en)
LU (2) LU73257A1 (en)
NL (2) NL183582C (en)
NO (1) NO146096C (en)
PL (1) PL106076B1 (en)
SE (1) SE412066B (en)
SU (1) SU603338A3 (en)
YU (1) YU40266B (en)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2704485A1 (en) * 1977-02-03 1978-08-10 Thomae Gmbh Dr K NEW 2,5-DIHYDRO-1,2-THIAZINO ANGLE CLAMP ON 5,6-B ANGLE CLAMP ON INDOL-3-CARBOXAMID-1,1-DIOXIDE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THEM
LU78009A1 (en) * 1977-08-22 1979-05-23 Hoffmann La Roche METHOD FOR PRODUCING THIAZINE DERIVATIVES
ZA784958B (en) * 1977-09-06 1979-08-29 Hoffmann La Roche Thiazine derivatives
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
DE2838377A1 (en) * 1978-09-02 1980-03-20 Thomae Gmbh Dr K NEW 4-HYDROXY-2H SQUARE CLAMP ON 1 SQUARE CLAMP ON BENZOTHIENO SQUARE CLAMP ON 2.3-S SQUARE CLAMP ON -1,2- THIAZINE-3-CARBOXAMIDE-1,1-DIOXIDE AND THEIR SALES, THEIR USE AND METHOD FOR THEM YOUR PRODUCTION
AU5811280A (en) * 1979-06-13 1980-12-18 F. Hoffmann-La Roche Ag Thiazine derivatives
JPS58109492A (en) * 1981-12-22 1983-06-29 Mitsui Toatsu Chem Inc Thienothiazine derivative and drug composition containing it
ATE26720T1 (en) * 1982-09-09 1987-05-15 Hoffmann La Roche THIENO(2,3-E)-1,2-THIAZINE DERIVATIVES.
JPS60163533U (en) * 1984-04-02 1985-10-30 ホシデン株式会社 Braking device for reel stand
JPH0318748Y2 (en) * 1985-12-18 1991-04-19
ATA39088A (en) 1988-02-18 1990-06-15 Binder Dieter Dr BASICALLY SUBSTITUTED THIENOISOTHIAZOL-3 (2H) -ON-1,1-DIOXIDES AND THEIR PHARMACEUTICALLY COMPATIBLE SALTS, METHOD FOR THE PRODUCTION AND THEIR USE
AT400437B (en) * 1993-12-14 1995-12-27 Chem Pharm Forsch Gmbh Novel N-heterocyclic thienothiazinecarboxamides, process for their preparation and their use
AT400568B (en) * 1994-05-18 1996-01-25 Chem Pharm Forsch Gmbh Novel N-heterocyclic thienothiazinecarboxamides, process for their preparation and their use
EP0658559A1 (en) * 1993-12-14 1995-06-21 Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. Thienothiazin derivatives, process for their preparation and their use as 5-dipoxygenase and cyclooxygenase inhibitors
US5538966A (en) * 1994-01-21 1996-07-23 Alcon Laboratories, Inc. Carbonic anhydrase inhibitors
IT1308633B1 (en) 1999-03-02 2002-01-09 Nicox Sa NITROSSIDERIVATI.
CN1171892C (en) * 2001-06-25 2004-10-20 李晶 Thienothiazine compound with anti-inflammatory and antalgic activity and its preparing process and usage

Also Published As

Publication number Publication date
NL183582B (en) 1988-07-01
ATA655975A (en) 1978-10-15
FR2282893B1 (en) 1980-05-16
DE2537070A1 (en) 1976-03-18
BR7505463A (en) 1976-08-03
SU603338A3 (en) 1978-04-15
PL106076B1 (en) 1979-11-30
YU40266B (en) 1985-12-31
AU8418675A (en) 1977-02-24
LU88312I2 (en) 1994-09-09
HU173739B (en) 1979-08-28
DE2537070C2 (en) 1987-06-25
DK137835C (en) 1978-10-16
DD124119A5 (en) 1977-02-02
YU216675A (en) 1982-08-31
DK381175A (en) 1976-02-27
SE412066B (en) 1980-02-18
FR2303803B1 (en) 1979-07-13
FI59253B (en) 1981-03-31
NL7510057A (en) 1976-03-01
FI59253C (en) 1981-07-10
FR2309558B1 (en) 1979-05-04
DK137835B (en) 1978-05-16
AT350064B (en) 1979-05-10
NO752932L (en) 1976-02-27
GB1519811A (en) 1978-08-02
NO146096B (en) 1982-04-19
FR2282893A1 (en) 1976-03-26
NL930080I1 (en) 1993-09-16
IE41457B1 (en) 1980-01-02
IE41457L (en) 1976-02-26
FR2309558A1 (en) 1976-11-26
IL47877A0 (en) 1975-11-25
LU73257A1 (en) 1977-04-15
IL47877A (en) 1978-10-31
FR2303803A1 (en) 1976-10-08
SE7509446L (en) 1976-02-27
NO146096C (en) 1982-07-28
JPS5148694A (en) 1976-04-26
FI752398A (en) 1976-02-27
JPS5826758B2 (en) 1983-06-04
NL930080I2 (en) 1994-01-03
NL183582C (en) 1988-12-01

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