AR209436A1 - Procedimiento para la fabricacion de derivados de 2-(beta-(fenilo opcionalmente sustituido) vinil)morfolina y 2-(-beta-(fenilo opcionalmente sustituido) etil) morfolina - Google Patents

Procedimiento para la fabricacion de derivados de 2-(beta-(fenilo opcionalmente sustituido) vinil)morfolina y 2-(-beta-(fenilo opcionalmente sustituido) etil) morfolina

Info

Publication number
AR209436A1
AR209436A1 AR258562A AR25856276A AR209436A1 AR 209436 A1 AR209436 A1 AR 209436A1 AR 258562 A AR258562 A AR 258562A AR 25856276 A AR25856276 A AR 25856276A AR 209436 A1 AR209436 A1 AR 209436A1
Authority
AR
Argentina
Prior art keywords
morpholine
beta
optionally substituted
substituted phenyl
vinyl
Prior art date
Application number
AR258562A
Other languages
English (en)
Spanish (es)
Inventor
Bernard J Mcloughlin
Allen J Guildford
Original Assignee
Ici Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Ltd filed Critical Ici Ltd
Application granted granted Critical
Publication of AR209436A1 publication Critical patent/AR209436A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C07D265/321,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/04Compounds containing oxirane rings containing only hydrogen and carbon atoms in addition to the ring oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07F9/6533Six-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR258562A 1974-05-07 1976-04-29 Procedimiento para la fabricacion de derivados de 2-(beta-(fenilo opcionalmente sustituido) vinil)morfolina y 2-(-beta-(fenilo opcionalmente sustituido) etil) morfolina AR209436A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB2001374A GB1452701A (en) 1974-05-07 1974-05-07 Morpholine derivatives
JP2495676A JPS52139074A (en) 1974-05-07 1976-03-08 Morpholine derivative and mental version drug composition containing same

Publications (1)

Publication Number Publication Date
AR209436A1 true AR209436A1 (es) 1977-04-29

Family

ID=26254367

Family Applications (1)

Application Number Title Priority Date Filing Date
AR258562A AR209436A1 (es) 1974-05-07 1976-04-29 Procedimiento para la fabricacion de derivados de 2-(beta-(fenilo opcionalmente sustituido) vinil)morfolina y 2-(-beta-(fenilo opcionalmente sustituido) etil) morfolina

Country Status (20)

Country Link
US (1) US4010266A (fr)
JP (2) JPS50154273A (fr)
AR (1) AR209436A1 (fr)
AT (1) AT344188B (fr)
BE (1) BE828822A (fr)
CA (1) CA1067075A (fr)
CH (2) CH610894A5 (fr)
DD (1) DD121641A5 (fr)
DE (1) DE2519101A1 (fr)
DK (1) DK198675A (fr)
FI (1) FI751344A (fr)
FR (1) FR2269953B1 (fr)
GB (1) GB1452701A (fr)
HK (1) HK5580A (fr)
IN (1) IN141021B (fr)
KE (1) KE3021A (fr)
LU (1) LU72408A1 (fr)
NL (1) NL7505140A (fr)
SE (1) SE425312B (fr)
ZA (1) ZA752388B (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4088814A (en) * 1974-05-07 1978-05-09 Imperial Chemical Industries Limited Morpholine derivatives
JPS5266991U (fr) * 1975-11-13 1977-05-18
DE2731668A1 (de) * 1976-07-14 1978-01-19 Ici Ltd Appetitzuegler
IE50355B1 (en) * 1979-10-20 1986-04-02 Wyeth John & Brother Ltd Morpholine derivatives
WO1993015052A1 (fr) * 1992-01-28 1993-08-05 Smithkline Beecham Plc Composes utilises comme antagonistes des canaux calciques
US5637699A (en) * 1992-06-29 1997-06-10 Merck & Co., Inc. Process for preparing morpholine tachykinin receptor antagonists
US6048859A (en) 1992-06-29 2000-04-11 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
US5719147A (en) * 1992-06-29 1998-02-17 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
IL112778A0 (en) * 1994-03-04 1995-05-26 Merck & Co Inc Substituted heterocycles, their preparation and pharmaceutical compositions containing them
ATE287878T1 (de) * 1996-08-23 2005-02-15 Neurosearch As Disubstituierte morpholin-, oxazepin- oder thiazepinderivate, deren herstellung und verwendung als dopamin-d4-rezeptorantagonisten
US7294637B2 (en) 2000-09-11 2007-11-13 Sepracor, Inc. Method of treating addiction or dependence using a ligand for a monamine receptor or transporter
AU9087301A (en) 2000-09-11 2002-03-26 Sepracor Inc Ligands for monoamine receptors and transporters, and methods of use thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2255077A (en) * 1938-03-21 1941-09-09 Du Pont Film Mfg Corp Filter dyes for color photography

Also Published As

Publication number Publication date
DE2519101A1 (de) 1975-11-20
CH610894A5 (fr) 1979-05-15
FI751344A (fr) 1975-11-08
CA1067075A (fr) 1979-11-27
ZA752388B (en) 1976-03-31
IN141021B (fr) 1977-01-08
AU8021575A (en) 1976-10-21
CH634569A5 (de) 1983-02-15
BE828822A (fr) 1975-11-07
GB1452701A (en) 1976-10-13
ATA341575A (de) 1977-11-15
NL7505140A (nl) 1975-11-11
SE425312B (sv) 1982-09-20
JPS52139074A (en) 1977-11-19
KE3021A (en) 1980-03-14
LU72408A1 (fr) 1976-11-11
DK198675A (da) 1975-11-08
AT344188B (de) 1978-07-10
JPS50154273A (fr) 1975-12-12
FR2269953B1 (fr) 1978-10-06
DD121641A5 (fr) 1976-08-12
FR2269953A1 (fr) 1975-12-05
HK5580A (en) 1980-02-29
US4010266A (en) 1977-03-01
SE7505237L (sv) 1975-11-10

Similar Documents

Publication Publication Date Title
AR211097A1 (es) Procedimiento para la preparacionde nuevos derivados de 3-(carbamil o tiocarbamil)-sulfamido-piridina-4-sustituida.
AR206339A1 (es) Procedimiento para la preparacion de derivados de 1-(metoxifenil)-4-(3-(naft-1-il-oxi)-2-hidroxi-propil)-piperazina
FI65617B (fi) Mellanprodukt foer framstaellning av magsyrasekretionsinhiberande 2-(2-pyridylmetylsulfinyl)-benzimidazolderivat
AR210990A1 (es) Procedimiento para preparar derivados de 1,1-dihideoperflujoroalcobenzamidas n-pirrolidin- o piperidin- sustituidas
AR209436A1 (es) Procedimiento para la fabricacion de derivados de 2-(beta-(fenilo opcionalmente sustituido) vinil)morfolina y 2-(-beta-(fenilo opcionalmente sustituido) etil) morfolina
AR207869A1 (es) Procedimiento para la produccion de nuevos derivados de 2-(4-alquil-1-piperacinil)-metil-1-bencil-benzimidazol
DK588575A (da) Morpholinderivater
AR213287A1 (es) Procedimiento para preparar derivados de 4-(2-hidroxi-3-aminopropoxi)-indol
IT1041201B (it) Procedimento per la produzione di 2 metil tetraidro pirimidine i sostituite
SE7708692L (sv) Forfarande for framstellning av fiberarmerade cementprodukter
NO143625C (no) Analogifremgangsmaate for fremstilling av 2-metoksy-benzamider
AR206234A1 (es) Procedimiento para preparar 2-mercaptobenzotiazol
FI772629A (fi) Foerfarande foer framstaellning av blodtryckssaenkande 2-(aroylpiperazin-1-yl)-4-amino-6 7-dimetoxikinazoliner
AR208184A1 (es) Procedimiento para la fabricacion de derivados de 2-(aminocarbonil-aza-alcanamido)-benzofenoma
NO146357C (no) Fremgangsmaate ved fremstilling av nye prostaglandiner
AR219283A1 (es) Procedimiento para preparar derivados de 2-aminoalquil-3-(fenilo opcionalmente substituido)-isoindol-1-carboxilico y esteres y amidas opcionalmente substituidos en posicion 4,5,6,o 7
IT1033234B (it) Procedimento per la fabbricazione di isobutano
IT1043016B (it) Procedimento per la polimerizza zione dei cloroclofosfazenni
AR206658A1 (es) Procedimiento para la produccion de nuevos diariloxi-imidazolilacetales
AR213412A1 (es) Procedimiento para obtener derivados de 9-aminoalquil-9,10-dihidro-9,10-metanoantraceno y sus sales
SE421793B (sv) Analogiforfarande for framstellning naftyridinsubstituerade pyrrolderivat
NO143314C (no) Fremgangsmaate for fremstilling av akrylamid
AR213082A1 (es) Procedimiento para preparar nuevos derivados de las 5-(2-morfolinitmetil)-dibenzazepinas
AR202966A1 (es) Procedimiento para la preparacion de derivados de 1-(3-(naft-1-il-oxi)-propil)-piperazina
AR216894A1 (es) Procedimiento para la obtencion de derivados de 1,3-diisocianatopropano y dichos derivados